Enzymatic Synthesis of Austroeupatol Esters with Enhanced Antiprotozoal Activity.
Elso OG, Bivona AE, Aguilera E, Alvarez G, Sülsen VP, García Liñares GE.
ACS Med Chem Lett · rapid-communication; journal article · DOI 10.1021/acsmedchemlett.4c00070 PUBLIKATIONSREGISTRET
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39 träffarAntiparasitic Activity of Two Natural Terpenes from <i>Salvia cuspidata</i> against <i>Leishmania amazonensis</i>.
Troncoso ME, Germanó MJ, Arrieta VJ, García Bustos MF, Cifuente D, Cargnelutti DE, Lozano ES.
J Nat Prod · research support, non-u.s. gov't; journal article · DOI 10.1021/acs.jnatprod.2c00976Natural and synthetic coumarins as antileishmanial agents: A review.
Gonçalves GA, Spillere AR, das Neves GM, Kagami LP, von Poser GL, Canto RFS, Eifler-Lima V.
Eur J Med Chem · review; journal article · DOI 10.1016/j.ejmech.2020.112514<i>Leishmania infantum</i> isolates exhibit high infectivity and reduced susceptibility to amphotericin B.
Faral-Tello P, Greif G, Satragno D, Basmadjián Y, Robello C.
RSC Med Chem · research-article; journal article · DOI 10.1039/d0md00073f<i>O</i>-Alkyl Hydroxamates Display Potent and Selective Antileishmanial Activity.
Corpas-López V, Tabraue-Chávez M, Sixto-López Y, Panadero-Fajardo S, Alves de Lima Franco F, Domínguez-Seglar JF, Morillas-Márquez F, Franco-Montalbán F, Díaz-Gavilán M, Correa-Basurto J, López-Viota J, López-Viota M, Pérez Del Palacio J, de la Cruz M, de Pedro N, Martín-Sánchez J, Gómez-Vidal JA.
J Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1021/acs.jmedchem.9b02016Antileishmanial activity and cytotoxicity of ent-beyerene diterpenoids.
Murillo JA, Gil JF, Upegui YA, Restrepo AM, Robledo SM, Quiñones W, Echeverri F, San Martin A, Olivo HF, Escobar G.
Bioorg Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1016/j.bmc.2018.11.030Synthesis and leishmanicidal activity of eugenol derivatives bearing 1,2,3-triazole functionalities.
Teixeira RR, Gazolla PAR, da Silva AM, Borsodi MPG, Bergmann BR, Ferreira RS, Vaz BG, Vasconcelos GA, Lima WP.
Eur J Med Chem · journal article · DOI 10.1016/j.ejmech.2018.01.046Antileishmanial activity of new thiophene-indole hybrids: Design, synthesis, biological and cytotoxic evaluation, and chemometric studies.
Félix MB, de Souza ER, de Lima MDCA, Frade DKG, Serafim VL, Rodrigues KADF, Néris PLDN, Ribeiro FF, Scotti L, Scotti MT, de Aquino TM, Mendonça Junior FJB, de Oliveira MR.
Bioorg Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1016/j.bmc.2016.04.057Synthesis, leishmanicidal, trypanocidal and cytotoxic activity of quinoline-hydrazone hybrids.
Coa JC, Castrillón W, Cardona W, Carda M, Ospina V, Muñoz JA, Vélez ID, Robledo SM.
Eur J Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1016/j.ejmech.2015.07.018(-)-α-Bisabolol, a Promising Oral Compound for the Treatment of Visceral Leishmaniasis.
Corpas-López V, Morillas-Márquez F, Navarro-Moll MC, Merino-Espinosa G, Díaz-Sáez V, Martín-Sánchez J.
J Nat Prod · research support, non-u.s. gov't; journal article · DOI 10.1021/np5008697Design, synthesis and biological evaluation of quinazoline derivatives as anti-trypanosomatid and anti-plasmodial agents.
Mendoza-Martínez C, Correa-Basurto J, Nieto-Meneses R, Márquez-Navarro A, Aguilar-Suárez R, Montero-Cortes MD, Nogueda-Torres B, Suárez-Contreras E, Galindo-Sevilla N, Rojas-Rojas Á, Rodriguez-Lezama A, Hernández-Luis F.
Eur J Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1016/j.ejmech.2015.04.028Antileishmanial activity of quinazoline derivatives: synthesis, docking screens, molecular dynamic simulations and electrochemical studies.
Mendoza-Martínez C, Galindo-Sevilla N, Correa-Basurto J, Ugalde-Saldivar VM, Rodríguez-Delgado RG, Hernández-Pineda J, Padierna-Mota C, Flores-Alamo M, Hernández-Luis F.
Eur J Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1016/j.ejmech.2014.12.051Thymol and eugenol derivatives as potential antileishmanial agents.
de Morais SM, Vila-Nova NS, Bevilaqua CM, Rondon FC, Lobo CH, de Alencar Araripe Noronha Moura A, Sales AD, Rodrigues AP, de Figuereido JR, Campello CC, Wilson ME, de Andrade HF.
Bioorg Med Chem · research-article; journal article · DOI 10.1016/j.bmc.2014.08.020Recent developments in biological activities of chalcones: a mini review.
Singh P, Anand A, Kumar V.
Eur J Med Chem · research support, non-u.s. gov't; review; journal article · DOI 10.1016/j.ejmech.2014.08.033In vitro activity of scorpiand-like azamacrocycle derivatives in promastigotes and intracellular amastigotes of Leishmania infantum and Leishmania braziliensis.
Marín C, Clares MP, Ramírez-Macías I, Blasco S, Olmo F, Soriano C, Verdejo B, Rosales MJ, Gomez-Herrera D, García-España E, Sánchez-Moreno M.
Eur J Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1016/j.ejmech.2013.01.001Synthesis and anti-leishmanial activity of 5-(5-nitrofuran-2-yl)-1,3,4-thiadiazol-2-amines containing N-[(1-benzyl-1H-1,2,3-triazol-4-yl)methyl] moieties.
Tahghighi A, Razmi S, Mahdavi M, Mahdavi M, Foroumadi P, Ardestani SK, Emami S, Kobarfard F, Dastmalchi S, Shafiee A, Foroumadi A.
Eur J Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1016/j.ejmech.2012.01.046Synthesis and antileishmanial activity of novel 5-(5-nitrofuran-2-y1)-1,3,4-thiadiazoles with piperazinyl-linked benzamidine substituents.
Tahghighi A, Marznaki FR, Kobarfard F, Dastmalchi S, Mojarrad JS, Razmi S, Ardestani SK, Emami S, Shafiee A, Foroumadi A.
Eur J Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1016/j.ejmech.2011.03.053Anti-leishmanial and anti-trypanosomal activities of 1,4-dihydropyridines: In vitro evaluation and structure-activity relationship study.
Reimão JQ, Scotti MT, Tempone AG, Tempone AG.
Bioorg Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1016/j.bmc.2010.09.015Trypanoside, anti-tuberculosis, leishmanicidal, and cytotoxic activities of tetrahydrobenzothienopyrimidines.
Aponte JC, Vaisberg AJ, Castillo D, Gonzalez G, Estevez Y, Arevalo J, Quiliano M, Zimic M, Verástegui M, Málaga E, Gilman RH, Bustamante JM, Tarleton RL, Wang Y, Franzblau SG, Pauli GF, Sauvain M, Hammond GB.
Bioorg Med Chem · research support, non-u.s. gov't; research support, u.s. gov't, non-p.h.s.; journal article; research support, n.i.h., extramural · DOI 10.1016/j.bmc.2010.03.018Novel antileishmanial chalconoids: synthesis and biological activity of 1- or 3-(6-chloro-2H-chromen-3-yl)propen-1-ones.
Nazarian Z, Emami S, Heydari S, Ardestani SK, Nakhjiri M, Poorrajab F, Shafiee A, Foroumadi A.
Eur J Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1016/j.ejmech.2009.12.046In vitro and in vivo anti-Leishmania activity of polysubstituted synthetic chalcones.
Aponte JC, Castillo D, Estevez Y, Gonzalez G, Arevalo J, Hammond GB, Sauvain M.
Bioorg Med Chem Lett · research support, non-u.s. gov't; journal article · DOI 10.1016/j.bmcl.2009.11.033Comparative efficacies of two antimony regimens to treat Leishmania braziliensis-induced cutaneous Leishmaniasis in rhesus macaques (Macaca mulatta).
Grimaldi G, Porrozzi R, Friedrich K, Teva A, Marchevsky RS, Vieira F, Miekeley N, Paumgartten FJ.
Antimicrob Agents Chemother · comparative study; research support, non-u.s. gov't; research-article; journal article · DOI 10.1128/aac.00858-09Antileishmaniasis activity of flavonoids from Consolida oliveriana.
Marín C, Boutaleb-Charki S, Díaz JG, Huertas O, Rosales MJ, Pérez-Cordon G, Guitierrez-Sánchez R, Sánchez-Moreno M.
J Nat Prod · research support, non-u.s. gov't; journal article · DOI 10.1021/np8008122Antileishmanial activity of 1,3,4-thiadiazolium-2-aminide in mice infected with Leishmania amazonensis.
Rodrigues RF, Charret KS, da Silva EF, Echevarria A, Amaral VF, Leon LL, Canto-Cavalheiro MM.
Antimicrob Agents Chemother · research support, non-u.s. gov't; research-article; journal article · DOI 10.1128/aac.00062-08Activity of hydroxyurea against Leishmania mexicana.
Martinez-Rojano H, Mancilla-Ramirez J, Quiñonez-Diaz L, Galindo-Sevilla N.
Antimicrob Agents Chemother · research support, non-u.s. gov't; research-article; journal article · DOI 10.1128/aac.00124-08Nitroimidazolyl-1,3,4-thiadiazole-based anti-leishmanial agents: synthesis and in vitro biological evaluation.
Poorrajab F, Ardestani SK, Emami S, Behrouzi-Fardmoghadam M, Shafiee A, Foroumadi A.
Eur J Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1016/j.ejmech.2008.03.039Improved synthesis of seven aromatic Baylis-Hillman adducts (BHA): evaluation against Artemia salina Leach. and Leishmania chagasi.
Barbosa TP, Junior CG, Silva FP, Lopes HM, Figueiredo LR, Sousa SC, Batista GN, da Silva TG, Silva TM, de Oliveira MR, Vasconcellos ML.
Eur J Med Chem · journal article · DOI 10.1016/j.ejmech.2008.03.016Synthesis and in vitro anti-leishmanial activity of 1-[5-(5-nitrofuran-2-yl)-1,3,4-thiadiazol-2-yl]- and 1-[5-(5-nitrothiophen-2-yl)-1,3,4-thiadiazol-2-yl]-4-aroylpiperazines.
Behrouzi-Fardmoghadam M, Poorrajab F, Ardestani SK, Emami S, Shafiee A, Foroumadi A.
Bioorg Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1016/j.bmc.2008.02.052Antiparasitic, antineuroinflammatory, and cytotoxic polyketides from the marine sponge Plakortis angulospiculatus collected in Brazil.
Kossuga MH, Nascimento AM, Reimão JQ, Tempone AG, Tempone AG, Taniwaki NN, Veloso K, Ferreira AG, Cavalcanti BC, Pessoa C, Moraes MO, Mayer AM, Hajdu E, Berlinck RG.
J Nat Prod · research support, non-u.s. gov't; journal article; research support, n.i.h., extramural · DOI 10.1021/np0705256Activity of a hydroxybibenzyl bryophyte constituent against Leishmania spp. and Trypanosoma cruzi: in silico, in vitro and in vivo activity studies.
Roldos V, Nakayama H, Rolón M, Montero-Torres A, Trucco F, Torres S, Vega C, Marrero-Ponce Y, Heguaburu V, Yaluff G, Gómez-Barrio A, Sanabria L, Ferreira ME, Rojas de Arias A, Pandolfi E.
Eur J Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1016/j.ejmech.2007.11.007