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Publikationer i urvalet

50 träffar

Bibliografisk träff 2003-09-01

Carbonic anhydrase inhibitors: topically acting antiglaucoma sulfonamides incorporating esters and amides of 3- and 4-carboxybenzolamide.

Casini A, Scozzafava A, Mincione F, Menabuoni L, Starnotti M, Supuran CT.

Bioorg Med Chem Lett · comparative study; research support, non-u.s. gov't; journal article · DOI 10.1016/s0960-894x(03)00580-8

Bibliografisk träff 2003-05-01

Carbonic anhydrase inhibitors. Inhibition of tumor-associated isozyme IX by halogenosulfanilamide and halogenophenylaminobenzolamide derivatives.

Ilies MA, Vullo D, Pastorek J, Scozzafava A, Ilies M, Caproiu MT, Pastorekova S, Supuran CT.

J Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1021/jm021123s

Bibliografisk träff 2003-05-01

Carbonic anhydrase inhibitors. Inhibition of cytosolic isozymes I and II and transmembrane, tumor-associated isozyme IX with sulfamates including EMATE also acting as steroid sulfatase inhibitors.

Winum JY, Vullo D, Casini A, Montero JL, Scozzafava A, Supuran CT.

J Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1021/jm021124k

Bibliografisk träff 2003-03-01

Carbonic anhydrase inhibitors: inhibition of cytosolic isozymes I and II with sulfamide derivatives.

Casini A, Winum JY, Montero JL, Scozzafava A, Supuran CT.

Bioorg Med Chem Lett · research support, non-u.s. gov't; journal article · DOI 10.1016/s0960-894x(03)00028-3

Bibliografisk träff 2003-03-01

Carbonic anhydrase inhibitors: SAR and X-ray crystallographic study for the interaction of sugar sulfamates/sulfamides with isozymes I, II and IV.

Casini A, Antel J, Abbate F, Scozzafava A, David S, Waldeck H, Schäfer S, Supuran CT.

Bioorg Med Chem Lett · journal article · DOI 10.1016/s0960-894x(03)00029-5

Bibliografisk träff 2003-03-01

Carbonic anhydrase inhibitors: inhibition of the tumor-associated isozyme IX with aromatic and heterocyclic sulfonamides.

Vullo D, Franchi M, Gallori E, Pastorek J, Scozzafava A, Pastorekova S, Supuran CT.

Bioorg Med Chem Lett · research support, non-u.s. gov't; journal article · DOI 10.1016/s0960-894x(03)00091-x

Bibliografisk träff 2002-08-01

Successful virtual screening for novel inhibitors of human carbonic anhydrase: strategy and experimental confirmation.

Grüneberg S, Stubbs MT, Klebe G.

J Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1021/jm011112j

Bibliografisk träff 2002-06-01

Carbonic anhydrase inhibitors. Preparation of potent sulfonamides inhibitors incorporating bile acid tails.

Scozzafava A, Supuran CT.

Bioorg Med Chem Lett · journal article · DOI 10.1016/s0960-894x(02)00252-4

Bibliografisk träff 2002-03-01

Carbonic anhydrase inhibitors. A general approach for the preparation of water-soluble sulfonamides incorporating polyamino-polycarboxylate tails and of their metal complexes possessing long-lasting, topical intraocular pressure-lowering properties.

Scozzafava A, Menabuoni L, Mincione F, Supuran CT.

J Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1021/jm0108202

Bibliografisk träff 2002-01-01

Carbonic anhydrase inhibitors: anticonvulsant sulfonamides incorporating valproyl and other lipophilic moieties.

Masereel B, Rolin S, Abbate F, Scozzafava A, Supuran CT.

J Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1021/jm0109199

Bibliografisk träff 2001-02-01

Carbonic anhydrase inhibitors: synthesis of sulfonamides incorporating dtpa tails and of their zinc complexes with powerful topical antiglaucoma properties.

Scozzafava A, Menabuoni L, Mincione F, Mincione G, Supuran CT.

Bioorg Med Chem Lett · research support, non-u.s. gov't; journal article · DOI 10.1016/s0960-894x(00)00722-8

Bibliografisk träff 2000-12-01

Carbonic anhydrase inhibitors: water-soluble 4-sulfamoylphenylthioureas as topical intraocular pressure-lowering agents with long-lasting effects.

Casini A, Scozzafava A, Mincione F, Menabuoni L, Ilies MA, Supuran CT.

J Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1021/jm001051+

Bibliografisk träff 2000-11-01

Carbonic anhydrase inhibitors: perfluoroalkyl/aryl-substituted derivatives of aromatic/heterocyclic sulfonamides as topical intraocular pressure-lowering agents with prolonged duration of action.

Scozzafava A, Menabuoni L, Mincione F, Briganti F, Mincione G, Supuran CT.

J Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1021/jm000296j

Bibliografisk träff 2000-10-01

Interaction and transport of thiazide diuretics, loop diuretics, and acetazolamide via rat renal organic anion transporter rOAT1.

Uwai Y, Saito H, Hashimoto Y, Inui KI.

J Pharmacol Exp Ther · research support, non-u.s. gov't; journal article · DOI 10.1016/s0022-3565(24)38896-2

Bibliografisk träff 2000-01-01

Carbonic anhydrase inhibitors: synthesis of membrane-impermeant low molecular weight sulfonamides possessing in vivo selectivity for the membrane-bound versus cytosolic isozymes.

Scozzafava A, Briganti F, Ilies MA, Supuran CT.

J Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1021/jm990479+

Bibliografisk träff 1999-09-01

Carbonic anhydrase inhibitors: synthesis of water-soluble, aminoacyl/dipeptidyl sulfonamides possessing long-lasting intraocular pressure-lowering properties via the topical route.

Scozzafava A, Briganti F, Mincione G, Menabuoni L, Mincione F, Supuran CT.

J Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1021/jm9901879

Bibliografisk träff 1989-12-01

Topically active carbonic anhydrase inhibitors. 2. Benzo[b]thiophenesulfonamide derivatives with ocular hypotensive activity.

Graham SL, Shepard KL, Anderson PS, Baldwin JJ, Best DB, Christy ME, Freedman MB, Gautheron P, Habecker CN, Hoffman JM.

J Med Chem · journal article · DOI 10.1021/jm00132a009

Bibliografisk träff 1989-11-01

Topically active carbonic anhydrase inhibitors. 1. O-acyl derivatives of 6-hydroxybenzothiazole-2-sulfonamide.

Woltersdorf OW, Schwam H, Bicking JB, Brown SL, deSolms SJ, Fishman DR, Graham SL, Gautheron PD, Hoffman JM, Larson RD.

J Med Chem · journal article · DOI 10.1021/jm00131a011

Bibliografisk träff 1987-11-01

Synthesis and physicochemical properties of thiadiazolo[3,2-a]pyrimidinesulfonamides and thiadiazolo[3,2-a]triazinesulfonamides as candidates for topically effective carbonic anhydrase inhibitors.

Katritzky AR, Caster KC, Maren TH, Conroy CW, Bar-Ilan A.

J Med Chem · research support, u.s. gov't, p.h.s.; journal article · DOI 10.1021/jm00394a021

Bibliografisk träff 1980-02-01

Cerebrovasodilatation through selective inhibition of the enzyme carbonic anhydrase. 2. Imidazo[2,1-b]thiadiazole and imidazo[2,1-b]thiazolesulfonamides.

Barnish IT, Cross PE, Dickinson RP, Gadsby B, Parry MJ, Randall MJ, Sinclair IW.

J Med Chem · journal article · DOI 10.1021/jm00176a003