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Publikationer i urvalet

44 träffar

Bibliografisk träff 2011-08-05

Discovery of 7-hydroxy-6-methoxy-2-methyl-3-(3,4,5-trimethoxybenzoyl)benzo[b]furan (BNC105), a tubulin polymerization inhibitor with potent antiproliferative and tumor vascular disrupting properties.

Flynn BL, Gill GS, Grobelny DW, Chaplin JH, Paul D, Leske AF, Lavranos TC, Chalmers DK, Charman SA, Kostewicz E, Shackleford DM, Morizzi J, Hamel E, Jung MK, Kremmidiotis G.

J Med Chem · research-article; journal article · DOI 10.1021/jm200454y

Bibliografisk träff 2010-11-04

Synthesis of antimitotic polyalkoxyphenyl derivatives of combretastatin using plant allylpolyalkoxybenzenes.

Semenov VV, Kiselyov AS, Titov IY, Sagamanova IK, Ikizalp NN, Chernysheva NB, Tsyganov DV, Konyushkin LD, Firgang SI, Semenov RV, Karmanova IB, Raihstat MM, Semenova MN.

J Nat Prod · research support, non-u.s. gov't; journal article · DOI 10.1021/np1004278

Bibliografisk träff 2010-09-01

Identification of CKD-516: a potent tubulin polymerization inhibitor with marked antitumor activity against murine and human solid tumors.

Lee J, Kim SJ, Choi H, Kim YH, Lim IT, Yang HM, Lee CS, Kang HR, Ahn SK, Moon SK, Kim DH, Lee S, Choi NS, Lee KJ.

J Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1021/jm1002414

Bibliografisk träff 2010-01-14

Novel derivatives of 1,3,4-oxadiazoles are potent mitostatic agents featuring strong microtubule depolymerizing activity in the sea urchin embryo and cell culture assays.

Kiselyov AS, Semenova MN, Chernyshova NB, Leitao A, Samet AV, Kislyi KA, Raihstat MM, Oprea T, Lemcke H, Lantow M, Weiss DG, Ikizalp NN, Kuznetsov SA, Semenov VV.

Eur J Med Chem · journal article · DOI 10.1016/j.ejmech.2009.12.072

Bibliografisk träff 2009-10-20

Synthesis and antitumor-evaluation of cyclopropyl-containing combretastatin analogs.

Fürst R, Zupkó I, Berényi A, Ecker GF, Rinner U.

Bioorg Med Chem Lett · research support, non-u.s. gov't; journal article · DOI 10.1016/j.bmcl.2009.10.064

Bibliografisk träff 2009-09-25

Combretastatin-like chalcones as inhibitors of microtubule polymerization. Part 1: synthesis and biological evaluation of antivascular activity.

Ducki S, Rennison D, Woo M, Kendall A, Chabert JF, McGown AT, Lawrence NJ.

Bioorg Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1016/j.bmc.2009.09.039

Bibliografisk träff 2009-03-01

Antineoplastic agents. 578. Synthesis of stilstatins 1 and 2 and their water-soluble prodrugs.

Pettit GR, Thornhill A, Melody N, Knight JC.

J Nat Prod · research support, non-u.s. gov't; journal article; research support, n.i.h., extramural · DOI 10.1021/np800608c

Bibliografisk träff 2008-02-28

Combretastatin dinitrogen-substituted stilbene analogues as tubulin-binding and vascular-disrupting agents.

Siles R, Ackley JF, Hadimani MB, Hall JJ, Mugabe BE, Guddneppanavar R, Monk KA, Chapuis JC, Pettit GR, Chaplin DJ, Edvardsen K, Trawick ML, Garner CM, Pinney KG.

J Nat Prod · research support, non-u.s. gov't; research support, u.s. gov't, non-p.h.s.; journal article; research support, n.i.h., extramural · DOI 10.1021/np070377j

Bibliografisk träff 2005-10-01

Antineoplastic agents. 509: synthesis of fluorcombstatin phosphate and related 3-halostilbenes(1).

Pettit GR, Minardi MD, Rosenberg HJ, Hamel E, Bibby MC, Martin SW, Jung MK, Pettit RK, Cuthbertson TJ, Chapuis JC.

J Nat Prod · research support, u.s. gov't, p.h.s.; research support, non-u.s. gov't; journal article; research support, n.i.h., extramural · DOI 10.1021/np058038i

Bibliografisk träff 2005-06-01

Antineoplastic agents. 445. Synthesis and evaluation of structural modifications of (Z)- and (E)-combretastatin A-41.

Pettit GR, Rhodes MR, Herald DL, Hamel E, Schmidt JM, Pettit RK.

J Med Chem · research support, u.s. gov't, p.h.s.; research support, non-u.s. gov't; journal article; research support, n.i.h., extramural · DOI 10.1021/jm0205797

Bibliografisk träff 2003-05-01

Synthesis, in vitro, and in vivo evaluation of phosphate ester derivatives of combretastatin A-4.

Hadimani MB, Hua J, Jonklaas MD, Kessler RJ, Sheng Y, Olivares A, Tanpure RP, Weiser A, Zhang J, Edvardsen K, Kane RR, Pinney KG.

Bioorg Med Chem Lett · comparative study; research support, non-u.s. gov't; journal article · DOI 10.1016/s0960-894x(03)00206-3

Bibliografisk träff 2000-07-01

Antineoplastic agents. 443. Synthesis of the cancer cell growth inhibitor hydroxyphenstatin and its sodium diphosphate prodrug.

Pettit GR, Grealish MP, Herald DL, Boyd MR, Hamel E, Pettit RK.

J Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1021/jm000045a

Bibliografisk träff 2000-07-01

Antineoplastic agents 440. Asymmetric synthesis and evaluation of the combretastatin A-1 SAR probes (1S,2S)- and (1R,2R)-1, 2-dihydroxy- 1-(2',3'-dihydroxy-4'-methoxyphenyl)-2-(3' ',4' ',5' '-trimethoxyphenyl)-ethane.

Pettit GR, Lippert JW, Herald DL, Hamel E, Pettit RK.

J Nat Prod · research support, u.s. gov't, p.h.s.; journal article · DOI 10.1021/np0000623

Bibliografisk träff 1998-05-01

Antineoplastic agents. 379. Synthesis of phenstatin phosphate.

Pettit GR, Toki B, Herald DL, Verdier-Pinard P, Boyd MR, Hamel E, Pettit RK.

J Med Chem · comparative study; research support, u.s. gov't, non-p.h.s.; journal article · DOI 10.1021/jm970644q