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Publikationer i urvalet

50 träffar

Bibliografisk träff 2012-11-19

Synthesis and biological characterization of 3-substituted 1H-indoles as ligands of GluN2B-containing N-methyl-D-aspartate receptors. Part 2.

Gitto R, De Luca L, Ferro S, Buemi MR, Russo E, De Sarro G, Chisari M, Ciranna L, Chimirri A.

J Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1021/jm301508d

Bibliografisk träff 2012-10-17

Combining galantamine and memantine in multitargeted, new chemical entities potentially useful in Alzheimer's disease.

Simoni E, Daniele S, Bottegoni G, Pizzirani D, Trincavelli ML, Goldoni L, Tarozzo G, Reggiani A, Martini C, Piomelli D, Melchiorre C, Rosini M, Cavalli A.

J Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1021/jm3009458

Bibliografisk träff 2011-10-17

Synthesis and binding assays of novel 3,3-dimethylpiperidine derivatives with various lipophilicities as σ₁ receptor ligands.

Ferorelli S, Abate C, Pedone MP, Colabufo NA, Contino M, Perrone R, Berardi F.

Bioorg Med Chem · journal article · DOI 10.1016/j.bmc.2011.10.023

Bibliografisk träff 2011-03-15

Synthesis, evaluation and metabolic studies of radiotracers containing a 4-(4-[18F]-fluorobenzyl)piperidin-1-yl moiety for the PET imaging of NR2B NMDA receptors.

Labas R, Gilbert G, Nicole O, Dhilly M, Abbas A, Tirel O, Buisson A, Henry J, Barré L, Debruyne D, Sobrio F.

Eur J Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1016/j.ejmech.2011.03.013

Bibliografisk träff 2010-12-08

Predicting hERG activities of compounds from their 3D structures: development and evaluation of a global descriptors based QSAR model.

Sinha N, Sen S.

Eur J Med Chem · journal article · DOI 10.1016/j.ejmech.2010.11.042

Bibliografisk träff 2010-09-25

Synthesis and biological evaluation of radio-iodinated benzimidazoles as SPECT imaging agents for NR2B subtype of NMDA receptor.

Fuchigami T, Yamaguchi H, Ogawa M, Biao L, Nakayama M, Haratake M, Magata Y.

Bioorg Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1016/j.bmc.2010.08.053

Bibliografisk träff 2010-09-24

Conformationally constrained NR2B selective NMDA receptor antagonists derived from ifenprodil: Synthesis and biological evaluation of tetrahydro-3-benzazepine-1,7-diols.

Tewes B, Frehland B, Schepmann D, Schmidtke KU, Winckler T, Wünsch B.

Bioorg Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1016/j.bmc.2010.09.026

Bibliografisk träff 2010-07-15

Identification of a novel NR2B-selective NMDA receptor antagonist using a virtual screening approach.

Mony L, Triballeau N, Paoletti P, Acher FC, Bertrand HO.

Bioorg Med Chem Lett · research support, non-u.s. gov't; journal article · DOI 10.1016/j.bmcl.2010.07.043

Bibliografisk träff 2009-12-01

Exploring the importance of piperazine N-atoms for sigma(2) receptor affinity and activity in a series of analogs of 1-cyclohexyl-4-[3-(5-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)propyl]piperazine (PB28).

Berardi F, Abate C, Ferorelli S, Uricchio V, Colabufo NA, Niso M, Perrone R.

J Med Chem · journal article · DOI 10.1021/jm9007505

Bibliografisk träff 2009-09-01

Synthesis, biological evaluation, and three-dimensional in silico pharmacophore model for sigma(1) receptor ligands based on a series of substituted benzo[d]oxazol-2(3H)-one derivatives.

Zampieri D, Mamolo MG, Laurini E, Florio C, Zanette C, Fermeglia M, Posocco P, Paneni MS, Pricl S, Vio L.

J Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1021/jm900366z

Bibliografisk träff 2008-12-31

Development of 3-substituted-1H-indole derivatives as NR2B/NMDA receptor antagonists.

Gitto R, De Luca L, Ferro S, Citraro R, De Sarro G, Costa L, Ciranna L, Chimirri A.

Bioorg Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1016/j.bmc.2008.12.058

Bibliografisk träff 2008-12-01

Novel 4-(4-aryl)cyclohexyl-1-(2-pyridyl)piperazines as Delta(8)-Delta(7) sterol isomerase (emopamil binding protein) selective ligands with antiproliferative activity.

Berardi F, Abate C, Ferorelli S, de Robertis AF, Leopoldo M, Colabufo NA, Niso M, Perrone R.

J Med Chem · journal article · DOI 10.1021/jm800965b

Bibliografisk träff 2008-09-01

Enantiomeric propanolamines as selective N-methyl-D-aspartate 2B receptor antagonists.

Tahirovic YA, Geballe M, Gruszecka-Kowalik E, Myers SJ, Lyuboslavsky P, Le P, French A, Irier H, Choi WB, Easterling K, Yuan H, Wilson LJ, Kotloski R, McNamara JO, Dingledine R, Liotta DC, Traynelis SF, Snyder JP.

J Med Chem · research support, non-u.s. gov't; research-article; journal article; research support, n.i.h., extramural · DOI 10.1021/jm8002153

Bibliografisk träff 2008-04-11

Reactive derivatives for affinity labeling in the ifenprodil site of NMDA receptors.

Alarcon K, Martz A, Mony L, Neyton J, Paoletti P, Goeldner M, Foucaud B.

Bioorg Med Chem Lett · research support, non-u.s. gov't; journal article · DOI 10.1016/j.bmcl.2008.04.019

Bibliografisk träff 2007-08-22

Design and evaluation of naphthol- and carbazole-containing fluorescent sigma ligands as potential probes for receptor binding studies.

Ferorelli S, Abate C, Colabufo NA, Niso M, Inglese C, Berardi F, Perrone R.

J Med Chem · journal article · DOI 10.1021/jm070373b

Bibliografisk träff 2007-04-08

Chemical genetics reveals a complex functional ground state of neural stem cells.

Diamandis P, Wildenhain J, Clarke ID, Sacher AG, Graham J, Bellows DS, Ling EK, Ward RJ, Jamieson LG, Tyers M, Dirks PB.

Nat Chem Biol · research support, non-u.s. gov't; journal article · DOI 10.1038/nchembio873

Bibliografisk träff 2005-12-01

Methyl substitution on the piperidine ring of N-[omega-(6-methoxynaphthalen-1-yl)alkyl] derivatives as a probe for selective binding and activity at the sigma(1) receptor.

Berardi F, Ferorelli S, Abate C, Pedone MP, Colabufo NA, Contino M, Perrone R.

J Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1021/jm050654o

Bibliografisk träff 2003-05-01

Synthesis of chiral 1-[omega-(4-chlorophenoxy)alkyl]-4-methylpiperidines and their biological evaluation at sigma1, sigma2, and sterol delta8-delta7 isomerase sites.

Berardi F, Loiodice F, Fracchiolla G, Colabufo NA, Perrone R, Tortorella V.

J Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1021/jm021014d

Bibliografisk träff 1999-12-01

A series of 6- and 7-piperazinyl- and -piperidinylmethylbenzoxazinones with dopamine D4 antagonist activity: discovery of a potential atypical antipsychotic agent.

Belliotti TR, Wustrow DJ, Brink WA, Zoski KT, Shih YH, Whetzel SZ, Georgic LM, Corbin AE, Akunne HC, Heffner TG, Pugsley TA, Wise LD.

J Med Chem · journal article · DOI 10.1021/jm990277d

Bibliografisk träff 1991-10-01

Separation of alpha 1 adrenergic and N-methyl-D-aspartate antagonist activity in a series of ifenprodil compounds.

Chenard BL, Shalaby IA, Koe BK, Ronau RT, Butler TW, Prochniak MA, Schmidt AW, Fox CB.

J Med Chem · comparative study; journal article · DOI 10.1021/jm00114a018