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Publikationer i urvalet

50 träffar

Bibliografisk träff 1993-11-01

Development of high-affinity 5-HT3 receptor antagonists. Structure-affinity relationships of novel 1,7-annelated indole derivatives.

van Wijngaarden I, Hamminga D, van Hes R, Standaar PJ, Tipker J, Tulp MT, Mol F, Olivier B, de Jonge A.

J Med Chem · comparative study; journal article · DOI 10.1021/jm00075a026

Bibliografisk träff 1993-10-01

5-HT3 receptor antagonists. 3. Quinoline derivatives which may be effective in the therapy of irritable bowel syndrome.

Kishibayashi N, Miwa Y, Hayashi H, Ishii A, Ichikawa S, Nonaka H, Yokoyama T, Suzuki F.

J Med Chem · journal article · DOI 10.1021/jm00074a009

Bibliografisk träff 1993-09-01

2-(Quinuclidin-3-yl)pyrido[4,3-b]indol-1-ones and isoquinolin-1-ones. Potent conformationally restricted 5-HT3 receptor antagonists.

Clark RD, Miller AB, Berger J, Repke DB, Weinhardt KK, Kowalczyk BA, Eglen RM, Bonhaus DW, Lee CH, Michel AD.

J Med Chem · comparative study; journal article · DOI 10.1021/jm00070a008

Bibliografisk träff 1993-09-01

Novel antagonists of 5-HT3 receptors. Synthesis and biological evaluation of piperazinylquinoxaline derivatives.

Monge A, Palop JA, Del Castillo JC, Calderó JM, Roca J, Romero G, Del Río J, Lasheras B.

J Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1021/jm00071a005

Bibliografisk träff 1993-03-01

5-HT3 receptor antagonists. 2. 4-Hydroxy-3-quinolinecarboxylic acid derivatives.

Hayashi H, Miwa Y, Ichikawa S, Yoda N, Miki I, Ishii A, Kono M, Yasuzawa T, Suzuki F.

J Med Chem · comparative study; journal article · DOI 10.1021/jm00057a011

Bibliografisk träff 1992-12-01

5-HT3 receptor antagonists. 1. New quinoline derivatives.

Hayashi H, Miwa Y, Miki I, Ichikawa S, Yoda N, Ishii A, Kono M, Suzuki F.

J Med Chem · journal article · DOI 10.1021/jm00104a016

Bibliografisk träff 1992-09-01

Novel 5-HT3 antagonists. Isoquinolinones and 3-aryl-2-pyridones.

Matsui T, Sugiura T, Nakai H, Iguchi S, Shigeoka S, Takada H, Odagaki Y, Nagao Y, Ushio Y, Ohmoto K.

J Med Chem · journal article · DOI 10.1021/jm00096a001

Bibliografisk träff 1992-05-01

Novel antagonists of the 5-HT3 receptor. Synthesis and structure-activity relationships of (2-alkoxybenzoyl)ureas.

Bradley G, Ward TJ, White JC, Coleman J, Taylor A, Rhodes KF.

J Med Chem · journal article · DOI 10.1021/jm00087a003

Bibliografisk träff 1992-03-01

Development of high-affinity 5-HT3 receptor antagonists. 1. Initial structure-activity relationship of novel benzamides.

Youssefyeh RD, Campbell HF, Klein S, Airey JE, Darkes P, Powers M, Schnapper M, Neuenschwander K, Fitzpatrick LR, Pendley CE.

J Med Chem · comparative study; journal article · DOI 10.1021/jm00083a014

Bibliografisk träff 1992-03-01

Development of high-affinity 5-HT3 receptor antagonists. 2. Two novel tricyclic benzamides.

Youssefyeh RD, Campbell HF, Airey JE, Klein S, Schnapper M, Powers M, Woodward R, Rodriguez W, Golec S, Studt W.

J Med Chem · comparative study; journal article · DOI 10.1021/jm00083a015

Bibliografisk träff 1992-03-01

Novel 5-HT3 antagonists: indol-3-ylspiro(azabicycloalkane-3,5'(4'H)-oxazoles).

Swain CJ, Baker R, Kneen C, Herbert R, Moseley J, Saunders J, Seward EM, Stevenson GI, Beer M, Stanton J.

J Med Chem · journal article · DOI 10.1021/jm00084a007

Bibliografisk träff 1992-01-01

Zatosetron, a potent, selective, and long-acting 5HT3 receptor antagonist: synthesis and structure-activity relationships.

Robertson DW, Lacefield WB, Bloomquist W, Pfeifer W, Simon RL, Cohen ML.

J Med Chem · journal article · DOI 10.1021/jm00080a016

Bibliografisk träff 1991-01-01

Novel 5-HT3 antagonists. Indole oxadiazoles.

Swain CJ, Baker R, Kneen C, Moseley J, Saunders J, Seward EM, Stevenson G, Beer M, Stanton J, Watling K.

J Med Chem · comparative study; journal article · DOI 10.1021/jm00105a021

Bibliografisk träff 1990-12-01

Synthesis and biochemical evaluation of tritium-labeled 1-methyl-N-(8-methyl-8-azabicyclo[3.2.1]oct-3-yl)-1H-indazole-3-carboxa mide, a useful radioligand for 5HT3 receptors.

Robertson DW, Bloomquist W, Cohen ML, Reid LR, Schenck K, Wong DT.

J Med Chem · journal article · DOI 10.1021/jm00174a013

Bibliografisk träff 1990-11-01

Synthesis, in vitro binding profile, and central nervous system penetrability of the highly potent 5-HT3 receptor antagonist [3H]-4-(2-methoxyphenyl)-2-[4(5)-methyl-5(4)-imidazolylmethyl]thiazole.

Rosen T, Seeger TF, McLean S, Nagel AA, Ives JL, Guarino KJ, Bryce D, Furman J, Roth RW, Chalabi PM.

J Med Chem · journal article · DOI 10.1021/jm00173a017

Bibliografisk träff 1990-10-01

An initial three-component pharmacophore for specific serotonin-3 receptor ligands.

Rizzi JP, Nagel AA, Rosen T, McLean S, Seeger T.

J Med Chem · journal article · DOI 10.1021/jm00172a007

Bibliografisk träff 1990-10-01

Thiazole as a carbonyl bioisostere. A novel class of highly potent and selective 5-HT3 receptor antagonists.

Rosen T, Nagel AA, Rizzi JP, Ives JL, Daffeh JB, Ganong AH, Guarino K, Heym J, McLean S, Nowakowski JT.

J Med Chem · journal article · DOI 10.1021/jm00172a006

Bibliografisk träff 1990-07-01

5-Hydroxytryptamine (5-HT3) receptor antagonists. 1. Indazole and indolizine-3-carboxylic acid derivatives.

Bermudez J, Fake CS, Joiner GF, Joiner KA, King FD, Miner WD, Sanger GJ.

J Med Chem · journal article · DOI 10.1021/jm00169a016

Bibliografisk träff 1990-06-01

Conformation-activity relationship study of 5-HT3 receptor antagonists and a definition of a model for this receptor site.

Hibert MF, Hoffmann R, Miller RC, Carr AA.

J Med Chem · journal article · DOI 10.1021/jm00168a011

Bibliografisk träff 1990-01-01

Aromatic thiazole derivatives: structurally novel and selective serotonin-3 receptor antagonists.

Nagel AA, Rosen T, Rizzi J, Daffeh J, Guarino K, Nowakowski J, Vincent LA, Heym J, McLean S, Seeger T.

J Med Chem · journal article · DOI 10.1021/jm00163a003