ActiQs / Forskning

PUBLIKATIONSREGISTRET

Gå till forskningen.

Publikationsdata från Europe PMC och PubMed. Följ källhänvisningar från ämnesregistret till originalpublikationerna.

Publikationer som ChEBI hänvisar till för Terfenadine. Visa hela publikationsregistret

En publikationsträff är inte en slutsats. Publikationslistan visar bibliografiska uppgifter. Eventuella forskningsutdrag visas separat med originalunderlag. En källhänvisning visar inte i sig effekt, dosering eller säkerhet.

Publikationer i urvalet

50 träffar

Bibliografisk träff 2005-03-01

Novel indolylindazolylmaleimides as inhibitors of protein kinase C-beta: synthesis, biological activity, and cardiovascular safety.

Zhang HC, Derian CK, McComsey DF, White KB, Ye H, Hecker LR, Li J, Addo MF, Croll D, Eckardt AJ, Smith CE, Li Q, Cheung WM, Conway BR, Emanuel S, Demarest KT, Andrade-Gordon P, Damiano BP, Maryanoff BE.

J Med Chem · journal article · DOI 10.1021/jm049478u

Bibliografisk träff 2004-12-01

Assessment of the health effects of chemicals in humans: II. Construction of an adverse effects database for QSAR modeling.

Matthews EJ, Kruhlak NL, Weaver JL, Benz RD, Contrera JF.

Curr Drug Discov Technol · journal article · DOI 10.2174/1570163043334794

Bibliografisk träff 2004-09-01

The pharmacophore hypotheses of I(Kr) potassium channel blockers: novel class III antiarrhythmic agents.

Du LP, Tsai KC, Li MY, You QD, Xia L.

Bioorg Med Chem Lett · comparative study; research support, non-u.s. gov't; journal article · DOI 10.1016/j.bmcl.2004.06.070

Bibliografisk träff 2004-08-01

[Drug-induced liver injury; fourteenth updated edition of the bibliographic database of liver injuries and related drugs].

Biour M, Ben Salem C, Chazouillères O, Grangé JD, Serfaty L, Poupon R.

Gastroenterol Clin Biol · bibliography; journal article · DOI 10.1016/s0399-8320(04)95062-2

Bibliografisk träff 2003-08-01

Prediction of hERG potassium channel affinity by traditional and hologram qSAR methods.

Keserü GM.

Bioorg Med Chem Lett · comparative study; journal article · DOI 10.1016/s0960-894x(03)00492-x

Bibliografisk träff 2003-05-01

Characterization of HERG potassium channel inhibition using CoMSiA 3D QSAR and homology modeling approaches.

Pearlstein RA, Vaz RJ, Kang J, Chen XL, Preobrazhenskaya M, Shchekotikhin AE, Korolev AM, Lysenkova LN, Miroshnikova OV, Hendrix J, Rampe D.

Bioorg Med Chem Lett · journal article · DOI 10.1016/s0960-894x(03)00196-3

Bibliografisk träff 2003-05-01

Understanding the structure-activity relationship of the human ether-a-go-go-related gene cardiac K+ channel. A model for bad behavior.

Pearlstein R, Vaz R, Rampe D.

J Med Chem · review; journal article · DOI 10.1021/jm0205651

Bibliografisk träff 2003-04-01

Comparison of in vitro P-glycoprotein screening assays: recommendations for their use in drug discovery.

Schwab D, Fischer H, Tabatabaei A, Poli S, Huwyler J.

J Med Chem · comparative study; validation study; journal article · DOI 10.1021/jm021012t

Bibliografisk träff 2002-08-01

Toward a pharmacophore for drugs inducing the long QT syndrome: insights from a CoMFA study of HERG K(+) channel blockers.

Cavalli A, Poluzzi E, De Ponti F, Recanatini M.

J Med Chem · journal article · DOI 10.1021/jm0208875

Bibliografisk träff 2001-11-01

Rational use of in vitro P-glycoprotein assays in drug discovery.

Polli JW, Wring SA, Humphreys JE, Huang L, Morgan JB, Webster LO, Serabjit-Singh CS.

J Pharmacol Exp Ther · journal article · DOI 10.1016/s0022-3565(24)29270-3

Bibliografisk träff 2001-11-01

Active transport of fluorescent P-glycoprotein substrates: evaluation as markers and interaction with inhibitors.

Wang EJ, Casciano CN, Clement RP, Johnson WW.

Biochem Biophys Res Commun · journal article · DOI 10.1006/bbrc.2001.6000

Bibliografisk träff 2000-01-01

Human UDP-glucuronosyltransferases: metabolism, expression, and disease.

Tukey RH, Strassburg CP.

Annu Rev Pharmacol Toxicol · research support, u.s. gov't, p.h.s.; research support, non-u.s. gov't; review; journal article · DOI 10.1146/annurev.pharmtox.40.1.581

Bibliografisk träff 1999-03-01

Interrelationship between substrates and inhibitors of human CYP3A and P-glycoprotein.

Kim RB, Wandel C, Leake B, Cvetkovic M, Fromm MF, Dempsey PJ, Roden MM, Belas F, Chaudhary AK, Roden DM, Wood AJ, Wilkinson GR.

Pharm Res · research support, u.s. gov't, p.h.s.; research support, non-u.s. gov't; journal article · DOI 10.1023/a:1018877803319

Bibliografisk träff 1999-02-01

New N-(pyridin-4-yl)-(indol-3-yl)acetamides and propanamides as antiallergic agents.

Menciu C, Duflos M, Fouchard F, Le Baut G, Emig P, Achterrath U, Szelenyi I, Nickel B, Schmidt J, Kutscher B, Günther E.

J Med Chem · journal article · DOI 10.1021/jm981079+

Bibliografisk träff 1998-03-01

Molecular properties and pharmacokinetic behavior of cetirizine, a zwitterionic H1-receptor antagonist.

Pagliara A, Testa B, Carrupt PA, Jolliet P, Morin C, Morin D, Urien S, Tillement JP, Rihoux JP.

J Med Chem · comparative study; research support, non-u.s. gov't; journal article · DOI 10.1021/jm9704311

Bibliografisk träff 1995-09-01

New antihistamines: substituted piperazine and piperidine derivatives as novel H1-antagonists.

Abou-Gharbia M, Moyer JA, Nielsen ST, Webb M, Patel U.

J Med Chem · journal article · DOI 10.1021/jm00020a018

Bibliografisk träff 1995-06-01

(Piperidinylalkoxy)chromones: novel antihistamines with additional antagonistic activity against leukotriene D4.

Zhang MQ, Wada Y, Sato F, Timmerman H.

J Med Chem · journal article · DOI 10.1021/jm00013a023

Bibliografisk träff 1994-08-01

[(3-Pyridylalkyl)piperidylidene]benzocycloheptapyridine derivatives as dual antagonists of PAF and histamine.

Carceller E, Merlos M, Giral M, Balsa D, Almansa C, Bartrolí J, García-Rafanell J, Forn J.

J Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1021/jm00043a009

Bibliografisk träff 1993-01-01

Terfenadine (Seldane): a new drug for restoring sensitivity to multidrug resistant cancer cells.

Hait WN, Gesmonde JF, Murren JR, Yang JM, Chen HX, Reiss M.

Biochem Pharmacol · comparative study; research support, u.s. gov't, p.h.s.; research support, non-u.s. gov't; journal article · DOI 10.1016/0006-2952(93)90076-9

Bibliografisk träff 1989-01-01

Synthesis and antiallergy activity of 4-(diarylhydroxymethyl)-1-[3-(aryloxy)propyl]piperidines and structurally related compounds.

Walsh DA, Franzyshen SK, Yanni JM.

J Med Chem · journal article · DOI 10.1021/jm00121a022