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Publikationer i urvalet

11 träffar

Bibliografisk träff 2022-12-15

Wiskostatin and other carbazole scaffolds as off target inhibitors of dynamin I GTPase activity and endocytosis.

Cossar PJ, Cardoso D, Mathwin D, Russell CC, Chiew B, Hamilton MP, Baker JR, Young KA, Chau N, Robinson PJ, McCluskey A.

Eur J Med Chem · journal article · DOI 10.1016/j.ejmech.2022.115001

Bibliografisk träff 2020-09-01

Development of Highly Potent Carbazole Amphiphiles as Membrane-Targeting Antimicrobials for Treating Gram-Positive Bacterial Infections.

Lin S, Liu J, Li H, Liu Y, Chen Y, Luo J, Liu S.

J Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1021/acs.jmedchem.0c00433

Bibliografisk träff 2020-03-03

Drug repurposing and rediscovery: Design, synthesis and preliminary biological evaluation of 1-arylamino-3-aryloxypropan-2-ols as anti-melanoma agents.

Chang Q, Long J, Hu L, Chen Z, Li Q, Hu G.

Bioorg Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1016/j.bmc.2020.115404

Bibliografisk träff 2019-05-13

Hybridization of β-Adrenergic Agonists and Antagonists Confers G Protein Bias.

Stanek M, Picard LP, Schmidt MF, Kaindl JM, Hübner H, Bouvier M, Weikert D, Gmeiner P.

J Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1021/acs.jmedchem.9b00349

Bibliografisk träff 2013-11-19

Comparison of the accuracy of experimental and predicted pKa values of basic and acidic compounds.

Settimo L, Bellman K, Knegtel RM.

Pharm Res · comparative study; journal article · DOI 10.1007/s11095-013-1232-z

Bibliografisk träff 2009-05-01

Lipophilicity of basic drugs measured by hydrophilic interaction chromatography.

Bard B, Carrupt PA, Martel S.

J Med Chem · journal article · DOI 10.1021/jm9003945

Bibliografisk träff 2008-09-14

Use of the X-ray structure of the beta2-adrenergic receptor for drug discovery. Part 2: Identification of active compounds.

Sabio M, Jones K, Topiol S.

Bioorg Med Chem Lett · journal article · DOI 10.1016/j.bmcl.2008.09.046

Bibliografisk träff 2008-07-26

Facile radiosynthesis of fluorine-18 labeled beta-blockers. Synthesis, radiolabeling, and ex vivo biodistribution of [18F]-(2S and 2R)-1-(1-fluoropropan-2-ylamino)-3-(m-tolyloxy)propan-2-ol.

Stephenson KA, Wilson AA, Meyer JH, Houle S, Vasdev N.

J Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1021/jm800227h

Bibliografisk träff 2008-01-12

High-throughput log P determination by ultraperformance liquid chromatography: a convenient tool for medicinal chemists.

Henchoz Y, Guillarme D, Rudaz S, Veuthey JL, Carrupt PA.

J Med Chem · journal article · DOI 10.1021/jm7014809

Bibliografisk träff 1994-09-01

Synthesis, binding properties, and 18F labeling of fluorocarazolol, a high-affinity beta-adrenergic receptor antagonist.

Zheng L, Berridge MS, Ernsberger P.

J Med Chem · journal article · DOI 10.1021/jm00046a005

Bibliografisk träff 1983-06-01

Synthesis of iodine-125 labeled (+/-)-15-(4-azidobenzyl)carazolol: a potent beta-adrenergic photoaffinity probe.

Heald SL, Jeffs PW, Lavin TN, Nambi P, Lefkowitz RJ, Caron MG.

J Med Chem · research support, u.s. gov't, p.h.s.; journal article · DOI 10.1021/jm00360a009