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Publikationer i urvalet

18 träffar

Bibliografisk träff 2023-07-17

Lipophilic modification of salirasib modulates the antiproliferative and antimigratory activity.

Ballari MS, O J Porta E, Zalazar EA, Etichetti CMB, Padrón JM, Girardini JE, Labadie GR.

Bioorg Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1016/j.bmc.2023.117417

Bibliografisk träff 2023-01-26

Screening through Lead Optimization of High Affinity, Allosteric Cyclin-Dependent Kinase 2 (CDK2) Inhibitors as Male Contraceptives That Reduce Sperm Counts in Mice.

Faber EB, Wang N, John K, Sun L, Wong HL, Burban D, Francis R, Tian D, Hong KH, Yang A, Wang L, Elsaid M, Khalid H, Levinson NM, Schönbrunn E, Hawkinson JE, Georg GI.

J Med Chem · research-article; research support, u.s. gov't, non-p.h.s.; journal article; research support, n.i.h., extramural · DOI 10.1021/acs.jmedchem.2c01731

Bibliografisk träff 2020-11-17

Targeting KRAS mutant cancers by preventing signaling transduction in the MAPK pathway.

Korzeniecki C, Priefer R.

Eur J Med Chem · review; journal article · DOI 10.1016/j.ejmech.2020.113006

Bibliografisk träff 2020-09-17

Paradigm shift of "classical" HDAC inhibitors to "hybrid" HDAC inhibitors in therapeutic interventions.

Vaidya GN, Rana P, Venkatesh A, Chatterjee DR, Contractor D, Satpute DP, Nagpure M, Jain A, Kumar D.

Eur J Med Chem · review; journal article · DOI 10.1016/j.ejmech.2020.112844

Bibliografisk träff 2020-08-01

Hydroxamic acid hybrids as the potential anticancer agents: An Overview.

Liu W, Liang Y, Si X.

Eur J Med Chem · review; journal article · DOI 10.1016/j.ejmech.2020.112679

Bibliografisk träff 2019-06-21

Repositioning Salirasib as a new antimalarial agent.

Porta EOJ, Bofill Verdaguer I, Perez C, Banchio C, Ferreira de Azevedo M, Katzin AM, Labadie GR.

Medchemcomm · research-article; journal article · DOI 10.1039/c9md00298g

Bibliografisk träff 2019-03-04

N-Cinnamoylanthranilates as human TRPA1 modulators: Structure-activity relationships and channel binding sites.

Chandrabalan A, McPhillie MJ, Morice AH, Boa AN, Sadofsky LR.

Eur J Med Chem · journal article · DOI 10.1016/j.ejmech.2019.02.074

Bibliografisk träff 2014-05-09

Polyisoprenylated methylated protein methyl esterase: a putative biomarker and therapeutic target for pancreatic cancer.

Aguilar BJ, Nkembo AT, Duverna R, Poku RA, Amissah F, Ablordeppey SY, Lamango NS.

Eur J Med Chem · research-article; journal article; research support, n.i.h., extramural · DOI 10.1016/j.ejmech.2014.05.018

Bibliografisk träff 2013-11-15

Synthesis and biological evaluation of farnesylthiosalicylamides as potential anti-tumor agents.

Ling Y, Wang Z, Zhu H, Wang X, Zhang W, Wang X, Chen L, Huang Z, Zhang Y.

Bioorg Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1016/j.bmc.2013.11.013

Bibliografisk träff 2012-02-07

Species comparison and pharmacological characterization of human, monkey, rat, and mouse TRPA1 channels.

Bianchi BR, Zhang XF, Reilly RM, Kym PR, Yao BB, Chen J.

J Pharmacol Exp Ther · journal article · DOI 10.1124/jpet.111.189902

Bibliografisk träff 2011-11-28

S-Farnesyl-Thiopropionic Acid (FTPA) Triazoles as Potent Inhibitors of Isoprenylcysteine Carboxyl Methyltransferase.

Bergman JA, Hahne K, Song J, Hrycyna CA, Gibbs RA.

ACS Med Chem Lett · rapid-communication; journal article · DOI 10.1021/ml200106d

Bibliografisk träff 2011-04-19

Novel nitric oxide-releasing derivatives of farnesylthiosalicylic acid: synthesis and evaluation of antihepatocellular carcinoma activity.

Ling Y, Ye X, Zhang Z, Zhang Y, Lai Y, Ji H, Peng S, Tian J.

J Med Chem · journal article · DOI 10.1021/jm1014814

Bibliografisk träff 2010-07-01

Transient receptor potential ankyrin 1 (TRPA1) channel as emerging target for novel analgesics and anti-inflammatory agents.

Baraldi PG, Preti D, Materazzi S, Geppetti P.

J Med Chem · review; journal article · DOI 10.1021/jm100062h

Bibliografisk träff 2010-04-03

Synthesis and evaluation of nitric oxide-releasing derivatives of farnesylthiosalicylic acid as anti-tumor agents.

Ling Y, Ye X, Ji H, Zhang Y, Lai Y, Peng S, Tian J.

Bioorg Med Chem · journal article · DOI 10.1016/j.bmc.2010.03.077

Bibliografisk träff 2009-09-06

Genetic mapping of targets mediating differential chemical phenotypes in Plasmodium falciparum.

Yuan J, Johnson RL, Huang R, Wichterman J, Jiang H, Hayton K, Fidock DA, Wellems TE, Inglese J, Austin CP, Su XZ.

Nat Chem Biol · research support, n.i.h., intramural; research-article; journal article; research support, n.i.h., extramural · DOI 10.1038/nchembio.215

Bibliografisk träff 2009-01-01

New derivatives of farnesylthiosalicylic acid (salirasib) for cancer treatment: farnesylthiosalicylamide inhibits tumor growth in nude mice models.

Goldberg L, Haklai R, Bauer V, Heiss A, Kloog Y.

J Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1021/jm801165r

Bibliografisk träff 2007-04-08

Chemical genetics reveals a complex functional ground state of neural stem cells.

Diamandis P, Wildenhain J, Clarke ID, Sacher AG, Graham J, Bellows DS, Ling EK, Ward RJ, Jamieson LG, Tyers M, Dirks PB.

Nat Chem Biol · research support, non-u.s. gov't; journal article · DOI 10.1038/nchembio873

Bibliografisk träff 1995-04-01

Farnesyl derivatives of rigid carboxylic acids-inhibitors of ras-dependent cell growth.

Marciano D, Ben-Baruch G, Marom M, Egozi Y, Haklai R, Kloog Y.

J Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1021/jm00008a004