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Publikationer i urvalet

8 träffar

Bibliografisk träff 2021-05-18

Designing Out PXR Activity on Drug Discovery Projects: A Review of Structure-Based Methods, Empirical and Computational Approaches.

Hall A, Chanteux H, Ménochet K, Ledecq M, Schulze MED.

J Med Chem · review; journal article · DOI 10.1021/acs.jmedchem.0c02245

Bibliografisk träff 2014-08-14

From human immunodeficiency virus non-nucleoside reverse transcriptase inhibitors to potent and selective antitrypanosomal compounds.

Venkatraj M, Ariën KK, Heeres J, Joossens J, Dirié B, Lyssens S, Michiels J, Cos P, Lewi PJ, Vanham G, Maes L, Van der Veken P, Augustyns K.

Bioorg Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1016/j.bmc.2014.08.005

Bibliografisk träff 2012-02-15

Strategies for the design of HIV-1 non-nucleoside reverse transcriptase inhibitors: lessons from the development of seven representative paradigms.

Li D, Zhan P, De Clercq E, Liu X.

J Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1021/jm200990c

Bibliografisk träff 2011-10-17

Design and synthesis of pyridone inhibitors of non-nucleoside reverse transcriptase.

Gomez R, Jolly S, Williams T, Tucker T, Tynebor R, Vacca J, McGaughey G, Lai MT, Felock P, Munshi V, DeStefano D, Touch S, Miller M, Yan Y, Sanchez R, Liang Y, Paton B, Wan BL, Anthony N.

Bioorg Med Chem Lett · journal article · DOI 10.1016/j.bmcl.2011.10.027

Bibliografisk träff 2010-08-30

Nitrile-containing pharmaceuticals: efficacious roles of the nitrile pharmacophore.

Fleming FF, Yao L, Ravikumar PC, Funk L, Shook BC.

J Med Chem · research-article; review; research support, u.s. gov't, non-p.h.s.; journal article; research support, n.i.h., extramural · DOI 10.1021/jm100762r

Bibliografisk träff 2010-07-26

Lersivirine, a nonnucleoside reverse transcriptase inhibitor with activity against drug-resistant human immunodeficiency virus type 1.

Corbau R, Mori J, Phillips C, Fishburn L, Martin A, Mowbray C, Panton W, Smith-Burchnell C, Thornberry A, Ringrose H, Knöchel T, Irving S, Westby M, Wood A, Perros M.

Antimicrob Agents Chemother · research support, non-u.s. gov't; research-article; journal article · DOI 10.1128/aac.01455-09

Bibliografisk träff 2010-02-16

Lack of a clinically relevant effect of an antacid on the pharmacokinetics of lersivirine.

Vourvahis M, Banerjee S, LaBadie R, Gore D, Mayer H.

Antimicrob Agents Chemother · research support, non-u.s. gov't; research-article; randomized controlled trial; journal article · DOI 10.1128/aac.01110-09

Bibliografisk träff 2009-08-27

Pyrazole NNRTIs 4: selection of UK-453,061 (lersivirine) as a development candidate.

Mowbray CE, Burt C, Corbau R, Gayton S, Hawes M, Perros M, Tran I, Price DA, Quinton FJ, Selby MD, Stupple PA, Webster R, Wood A.

Bioorg Med Chem Lett · journal article · DOI 10.1016/j.bmcl.2009.08.080