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Publikationer i urvalet

8 träffar

Bibliografisk träff 2021-04-28

Targeting the FtsZ Allosteric Binding Site with a Novel Fluorescence Polarization Screen, Cytological and Structural Approaches for Antibacterial Discovery.

Huecas S, Araújo-Bazán L, Ruiz FM, Ruiz-Ávila LB, Martínez RF, Escobar-Peña A, Artola M, Vázquez-Villa H, Martín-Fontecha M, Fernández-Tornero C, López-Rodríguez ML, Andreu JM.

J Med Chem · research support, non-u.s. gov't; research-article; journal article · DOI 10.1021/acs.jmedchem.0c02207

Bibliografisk träff 2021-03-02

Small-Molecule Drug Discovery in Triple Negative Breast Cancer: Current Situation and Future Directions.

Liao M, Zhang J, Wang G, Wang L, Liu J, Ouyang L, Liu B.

J Med Chem · research support, non-u.s. gov't; review; journal article · DOI 10.1021/acs.jmedchem.0c01180

Bibliografisk träff 2017-08-22

New application of tiplaxtinin as an effective FtsZ-targeting chemotype for an antimicrobial study.

Sun N, Zheng YY, Du RL, Cai SY, Zhang K, So LY, Cheung KC, Zhuo C, Lu YJ, Wong KY.

Medchemcomm · research-article; journal article · DOI 10.1039/c7md00387k

Bibliografisk träff 2011-08-11

Discovery of inhibitors of plasminogen activator inhibitor-1: structure-activity study of 5-nitro-2-phenoxybenzoic acid derivatives.

Pandya V, Jain M, Chakrabarti G, Soni H, Parmar B, Chaugule B, Patel J, Joshi J, Joshi N, Rath A, Raviya M, Shaikh M, Sairam KV, Patel H, Patel P.

Bioorg Med Chem Lett · journal article · DOI 10.1016/j.bmcl.2011.08.031

Bibliografisk träff 2007-06-03

In vitro PAI-1 inhibitory activity of oxalamide derivatives.

Jain MR, Shetty S, Chakrabarti G, Pandya V, Sharma A, Parmar B, Srivastava S, Raviya M, Soni H, Patel PR.

Eur J Med Chem · journal article · DOI 10.1016/j.ejmech.2007.05.011

Bibliografisk träff 2007-02-02

Mechanism of inactivation of plasminogen activator inhibitor-1 by a small molecule inhibitor.

Gorlatova NV, Cale JM, Elokdah H, Li D, Fan K, Warnock M, Crandall DL, Lawrence DA.

J Biol Chem · research support, non-u.s. gov't; journal article; research support, n.i.h., extramural · DOI 10.1074/jbc.m611642200

Bibliografisk träff 2005-08-01

Synthesis and SAR of 2-carboxylic acid indoles as inhibitors of plasminogen activator inhibitor-1.

Hu B, Jetter JW, Wrobel JE, Antrilli TM, Bauer JS, Di L, Polakowski S, Jain U, Crandall DL.

Bioorg Med Chem Lett · journal article · DOI 10.1016/j.bmcl.2005.05.095

Bibliografisk träff 2004-07-01

Tiplaxtinin, a novel, orally efficacious inhibitor of plasminogen activator inhibitor-1: design, synthesis, and preclinical characterization.

Elokdah H, Abou-Gharbia M, Hennan JK, McFarlane G, Mugford CP, Krishnamurthy G, Crandall DL.

J Med Chem · journal article · DOI 10.1021/jm049766q