Sleep modulating agents.
Choi Y, Raymer BK.
Bioorg Med Chem Lett · review; journal article · DOI 10.1016/j.bmcl.2019.06.043 PUBLIKATIONSREGISTRET
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Publikationer i urvalet
8 träffarActivation of the γ-Aminobutyric Acid Type B (GABA(B)) Receptor by Agonists and Positive Allosteric Modulators.
Brown KM, Roy KK, Hockerman GH, Doerksen RJ, Colby DA.
J Med Chem · research support, non-u.s. gov't; research-article; review; journal article; research support, n.i.h., extramural · DOI 10.1021/jm5018913Evaluation of difluoromethyl ketones as agonists of the γ-aminobutyric acid type B (GABAB) receptor.
Han C, Salyer AE, Kim EH, Jiang X, Jarrard RE, Powers MS, Kirchhoff AM, Salvador TK, Chester JA, Hockerman GH, Colby DA.
J Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1021/jm301805eDiscovery of a novel potent GABA(B) receptor agonist.
Xu F, Peng G, Phan T, Dilip U, Chen JL, Chernov-Rogan T, Zhang X, Grindstaff K, Annamalai T, Koller K, Gallop MA, Wustrow DJ.
Bioorg Med Chem Lett · journal article · DOI 10.1016/j.bmcl.2011.08.006QSAR and molecular modeling studies of baclofen analogues as GABA(B) agonists. Insights into the role of the aromatic moiety in GABA(B) binding and activation.
Costantino G, Macchiarulo A, Entrena Guadix A, Pellicciari R.
J Med Chem · journal article · DOI 10.1021/jm0100133Synthesis and pharmacology of the baclofen homologues 5-amino-4-(4-chlorophenyl)pentanoic acid and the R- and S-enantiomers of 5-amino-3-(4-chlorophenyl)pentanoic acid.
Karla R, Ebert B, Thorkildsen C, Herdeis C, Johansen TN, Nielsen B, Krogsgaard-Larsen P.
J Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1021/jm990076+Phosphinic acid analogues of GABA. 1. New potent and selective GABAB agonists.
Froestl W, Mickel SJ, Hall RG, von Sprecher G, Strub D, Baumann PA, Brugger F, Gentsch C, Jaekel J, Olpe HR.
J Med Chem · journal article · DOI 10.1021/jm00017a015[3H]Batrachotoxinin A 20 alpha-benzoate binding to voltage-sensitive sodium channels: a rapid and quantitative assay for local anesthetic activity in a variety of drugs.
McNeal ET, Lewandowski GA, Daly JW, Creveling CR.
J Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1021/jm00381a019