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Publikationer i urvalet

50 träffar

Bibliografisk träff 2005-12-01

Carbonic anhydrase inhibitors. The mitochondrial isozyme VB as a new target for sulfonamide and sulfamate inhibitors.

Nishimori I, Vullo D, Innocenti A, Scozzafava A, Mastrolorenzo A, Supuran CT.

J Med Chem · comparative study; journal article · DOI 10.1021/jm050483n

Bibliografisk träff 2005-11-01

Carbonic anhydrase inhibitors: inhibition of cytosolic/tumor-associated carbonic anhydrase isozymes I, II, and IX with benzo[b]thiophene 1,1-dioxide sulfonamides.

Innocenti A, Villar R, Martinez-Merino V, Gil MJ, Scozzafava A, Vullo D, Supuran CT.

Bioorg Med Chem Lett · research support, non-u.s. gov't; journal article · DOI 10.1016/j.bmcl.2005.04.078

Bibliografisk träff 2005-07-01

Carbonic anhydrase inhibitors. Design of fluorescent sulfonamides as probes of tumor-associated carbonic anhydrase IX that inhibit isozyme IX-mediated acidification of hypoxic tumors.

Cecchi A, Hulikova A, Pastorek J, Pastoreková S, Scozzafava A, Winum JY, Montero JL, Supuran CT.

J Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1021/jm0501073

Bibliografisk träff 2005-06-01

Carbonic anhydrase inhibitors: novel sulfonamides incorporating 1,3,5-triazine moieties as inhibitors of the cytosolic and tumour-associated carbonic anhydrase isozymes I, II and IX.

Garaj V, Puccetti L, Fasolis G, Winum JY, Montero JL, Scozzafava A, Vullo D, Innocenti A, Supuran CT.

Bioorg Med Chem Lett · research support, non-u.s. gov't; journal article · DOI 10.1016/j.bmcl.2005.04.056

Bibliografisk träff 2005-06-01

Carbonic anhydrase inhibitors. Inhibition of cytosolic/tumor-associated carbonic anhydrase isozymes I, II, IX, and XII with Schiff's bases incorporating chromone and aromatic sulfonamide moieties, and their zinc complexes.

Puccetti L, Fasolis G, Vullo D, Chohan ZH, Scozzafava A, Supuran CT.

Bioorg Med Chem Lett · research support, non-u.s. gov't; journal article · DOI 10.1016/j.bmcl.2005.04.055

Bibliografisk träff 2005-05-01

Carbonic anhydrase inhibitors. Zonisamide is an effective inhibitor of the cytosolic isozyme II and mitochondrial isozyme V: solution and X-ray crystallographic studies.

De Simone G, Di Fiore A, Menchise V, Pedone C, Antel J, Casini A, Scozzafava A, Wurl M, Supuran CT.

Bioorg Med Chem Lett · journal article · DOI 10.1016/j.bmcl.2005.03.032

Bibliografisk träff 2005-05-01

Carbonic anhydrase inhibitors: synthesis and inhibition of cytosolic/tumor-associated carbonic anhydrase isozymes I, II, and IX with sulfonamides incorporating thioureido-sulfanilyl scaffolds.

Puccetti L, Fasolis G, Cecchi A, Winum JY, Gamberi A, Montero JL, Scozzafava A, Supuran CT.

Bioorg Med Chem Lett · research support, non-u.s. gov't; journal article · DOI 10.1016/j.bmcl.2005.02.087

Bibliografisk träff 2005-03-01

Carbonic anhydrase inhibitors: synthesis and inhibition of cytosolic/membrane-associated carbonic anhydrase isozymes I, II, and IX with sulfonamides incorporating hydrazino moieties.

Winum JY, Dogné JM, Casini A, de Leval X, Montero JL, Scozzafava A, Vullo D, Innocenti A, Supuran CT.

J Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1021/jm0494826

Bibliografisk träff 2005-02-01

Carbonic anhydrase inhibitors: synthesis and inhibition of cytosolic/tumor-associated carbonic anhydrase isozymes I, II, and IX with bis-sulfamates.

Winum JY, Pastorekova S, Jakubickova L, Montero JL, Scozzafava A, Pastorek J, Vullo D, Innocenti A, Supuran CT.

Bioorg Med Chem Lett · research support, non-u.s. gov't; journal article · DOI 10.1016/j.bmcl.2004.11.058

Bibliografisk träff 2005-02-01

Carbonic anhydrase inhibitors. Inhibition of the human cytosolic isozyme VII with aromatic and heterocyclic sulfonamides.

Vullo D, Voipio J, Innocenti A, Rivera C, Ranki H, Scozzafava A, Kaila K, Supuran CT.

Bioorg Med Chem Lett · journal article · DOI 10.1016/j.bmcl.2004.12.052

Bibliografisk träff 2005-02-01

Carbonic anhydrase inhibitors. Inhibition of the membrane-bound human and bovine isozymes IV with sulfonamides.

Innocenti A, Firnges MA, Antel J, Wurl M, Scozzafava A, Supuran CT.

Bioorg Med Chem Lett · journal article · DOI 10.1016/j.bmcl.2004.12.009

Bibliografisk träff 2005-01-01

Carbonic anhydrase inhibitors. Novel sulfanilamide/acetazolamide derivatives obtained by the tail approach and their interaction with the cytosolic isozymes I and II, and the tumor-associated isozyme IX.

Turkmen H, Durgun M, Yilmaztekin S, Emul M, Innocenti A, Vullo D, Scozzafava A, Supuran CT.

Bioorg Med Chem Lett · research support, non-u.s. gov't; journal article · DOI 10.1016/j.bmcl.2004.10.070

Bibliografisk träff 2004-12-01

Carbonic anhydrase inhibitors: synthesis and inhibition of cytosolic/tumor-associated carbonic anhydrase isozymes I, II, and IX with sulfonamides derived from 4-isothiocyanato-benzolamide.

Cecchi A, Winum JY, Innocenti A, Vullo D, Montero JL, Scozzafava A, Supuran CT.

Bioorg Med Chem Lett · research support, non-u.s. gov't; journal article · DOI 10.1016/j.bmcl.2004.09.062

Bibliografisk träff 2004-12-01

Carbonic anhydrase inhibitors. Design of anticonvulsant sulfonamides incorporating indane moieties.

Chazalette C, Masereel B, Rolin S, Thiry A, Scozzafava A, Innocenti A, Supuran CT.

Bioorg Med Chem Lett · journal article · DOI 10.1016/j.bmcl.2004.09.061

Bibliografisk träff 2004-12-01

Carbonic anhydrase inhibitors. Inhibition of the prokariotic beta and gamma-class enzymes from Archaea with sulfonamides.

Zimmerman S, Innocenti A, Casini A, Ferry JG, Scozzafava A, Supuran CT.

Bioorg Med Chem Lett · research support, u.s. gov't, p.h.s.; research support, non-u.s. gov't; research support, u.s. gov't, non-p.h.s.; journal article · DOI 10.1016/j.bmcl.2004.09.085

Bibliografisk träff 2004-11-01

Carbonic anhydrase inhibitors: synthesis and inhibition of cytosolic/tumor-associated carbonic anhydrase isozymes I, II, and IX with sulfonamides incorporating 1,2,4-triazine moieties.

Garaj V, Puccetti L, Fasolis G, Winum JY, Montero JL, Scozzafava A, Vullo D, Innocenti A, Supuran CT.

Bioorg Med Chem Lett · research support, non-u.s. gov't; journal article · DOI 10.1016/j.bmcl.2004.07.087

Bibliografisk träff 2004-10-01

Carbonic anhydrase inhibitors: the first on-resin screening of a 4-sulfamoylphenylthiourea library.

Innocenti A, Casini A, Alcaro MC, Papini AM, Scozzafava A, Supuran CT.

J Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1021/jm049692i

Bibliografisk träff 2004-08-01

[Drug-induced liver injury; fourteenth updated edition of the bibliographic database of liver injuries and related drugs].

Biour M, Ben Salem C, Chazouillères O, Grangé JD, Serfaty L, Poupon R.

Gastroenterol Clin Biol · bibliography; journal article · DOI 10.1016/s0399-8320(04)95062-2

Bibliografisk träff 2004-07-01

Carbonic anhydrase inhibitors. Inhibition of cytosolic isozyme XIII with aromatic and heterocyclic sulfonamides: a novel target for the drug design.

Lehtonen JM, Parkkila S, Vullo D, Casini A, Scozzafava A, Supuran CT.

Bioorg Med Chem Lett · comparative study; research support, non-u.s. gov't; journal article · DOI 10.1016/j.bmcl.2004.04.106

Bibliografisk träff 2004-06-01

Carbonic anhydrase inhibitors: the first QSAR study on inhibition of tumor-associated isoenzyme IX with aromatic and heterocyclic sulfonamides.

Jaiswal M, Khadikar PV, Scozzafava A, Supuran CT.

Bioorg Med Chem Lett · journal article · DOI 10.1016/j.bmcl.2004.03.099

Bibliografisk träff 2004-05-01

Carbonic anhydrase inhibitors: inhibition of the tumor-associated isozyme IX with fluorine-containing sulfonamides. The first subnanomolar CA IX inhibitor discovered.

Vullo D, Scozzafava A, Pastorekova S, Pastorek J, Supuran CT.

Bioorg Med Chem Lett · journal article · DOI 10.1016/j.bmcl.2004.01.095

Bibliografisk träff 2004-05-01

Carbonic anhydrase inhibitors: synthesis and topical intraocular pressure lowering effects of fluorine-containing inhibitors devoid of enhanced reactivity.

de Leval X, Ilies M, Casini A, Dogné JM, Scozzafava A, Masini E, Mincione F, Starnotti M, Supuran CT.

J Med Chem · journal article · DOI 10.1021/jm031116j

Bibliografisk träff 2004-04-01

Carbonic anhydrase inhibitors. Design of selective, membrane-impermeant inhibitors targeting the human tumor-associated isozyme IX.

Casey JR, Morgan PE, Vullo D, Scozzafava A, Mastrolorenzo A, Supuran CT.

J Med Chem · journal article · DOI 10.1021/jm031079w

Bibliografisk träff 2004-02-01

Carbonic anhydrase inhibitors. Inhibition of mitochondrial isozyme V with aromatic and heterocyclic sulfonamides.

Vullo D, Franchi M, Gallori E, Antel J, Scozzafava A, Supuran CT.

J Med Chem · journal article · DOI 10.1021/jm031057+

Bibliografisk träff 2004-02-01

Carbonic anhydrase inhibitors: the first selective, membrane-impermeant inhibitors targeting the tumor-associated isozyme IX.

Pastorekova S, Casini A, Scozzafava A, Vullo D, Pastorek J, Supuran CT.

Bioorg Med Chem Lett · journal article · DOI 10.1016/j.bmcl.2003.12.029

Bibliografisk träff 2004-01-01

Carbonic anhydrase inhibitors: E7070, a sulfonamide anticancer agent, potently inhibits cytosolic isozymes I and II, and transmembrane, tumor-associated isozyme IX.

Abbate F, Casini A, Owa T, Scozzafava A, Supuran CT.

Bioorg Med Chem Lett · journal article · DOI 10.1016/j.bmcl.2003.09.062

Bibliografisk träff 2004-01-01

Carbonic anhydrase inhibitors: N-(p-sulfamoylphenyl)-alpha-D-glycopyranosylamines as topically acting antiglaucoma agents in hypertensive rabbits.

Winum JY, Casini A, Mincione F, Starnotti M, Montero JL, Scozzafava A, Supuran CT.

Bioorg Med Chem Lett · journal article · DOI 10.1016/j.bmcl.2003.09.063

Bibliografisk träff 2004-01-01

Carbonic anhydrase inhibitors: X-ray crystallographic structure of the adduct of human isozyme II with the antipsychotic drug sulpiride.

Abbate F, Coetzee A, Casini A, Ciattini S, Scozzafava A, Supuran CT.

Bioorg Med Chem Lett · journal article · DOI 10.1016/j.bmcl.2003.11.014

Bibliografisk träff 2004-01-01

Unexpected nanomolar inhibition of carbonic anhydrase by COX-2-selective celecoxib: new pharmacological opportunities due to related binding site recognition.

Weber A, Casini A, Heine A, Kuhn D, Supuran CT, Scozzafava A, Klebe G.

J Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1021/jm030912m

Bibliografisk träff 2003-12-01

Carbonic anhydrase inhibitors: inhibition of transmembrane, tumor-associated isozyme IX, and cytosolic isozymes I and II with aliphatic sulfamates.

Winum JY, Vullo D, Casini A, Montero JL, Scozzafava A, Supuran CT.

J Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1021/jm030911u