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Publikationer i urvalet

13 träffar

Bibliografisk träff 2013-03-27

PPARδ agonist GW501516 inhibits PDGF-stimulated pulmonary arterial smooth muscle cell function related to pathological vascular remodeling.

Liu G, Li X, Li Y, Tang X, Xu J, Li R, Hao P, Sun Y.

Biomed Res Int · research support, non-u.s. gov't; research-article; journal article · DOI 10.1155/2013/903947

Bibliografisk träff 2013-01-01

Synthesis, mass spectrometric characterization, and analysis of the PPARδ agonist GW1516 and its major human metabolites: targets in sports drug testing.

Thevis M, Möller I, Beuck S, Schänzer W.

Methods Mol Biol · research support, non-u.s. gov't; journal article · DOI 10.1007/978-1-62703-155-4_22

Bibliografisk träff 2012-10-10

GW501516-activated PPARβ/δ promotes liver fibrosis via p38-JNK MAPK-induced hepatic stellate cell proliferation.

Kostadinova R, Montagner A, Gouranton E, Fleury S, Guillou H, Dombrowicz D, Desreumaux P, Wahli W.

Cell Biosci · research-article; journal article · DOI 10.1186/2045-3701-2-34

Bibliografisk träff 2012-09-13

PPARδ agonist GW501516 prevents uncoupling of endothelial nitric oxide synthase in cerebral microvessels of hph-1 mice.

Santhanam AV, d'Uscio LV, He T, Katusic ZS.

Brain Res · research support, non-u.s. gov't; research-article; journal article; research support, n.i.h., extramural · DOI 10.1016/j.brainres.2012.09.012

Bibliografisk träff 2012-07-19

Lipid effects of peroxisome proliferator-activated receptor-δ agonist GW501516 in subjects with low high-density lipoprotein cholesterol: characteristics of metabolic syndrome.

Olson EJ, Pearce GL, Jones NP, Sprecher DL.

Arterioscler Thromb Vasc Biol · multicenter study; randomized controlled trial; journal article · DOI 10.1161/atvbaha.112.247890

Bibliografisk träff 2011-08-01

GW501516 acts as an efficient PPARα activator in the mouse liver.

Terada M, Araki M, Ashibe B, Motojima K.

Drug Discov Ther · journal article · DOI 10.5582/ddt.2011.v5.4.176

Bibliografisk träff 2011-05-01

The role played by the peroxisome proliferator-activated receptor-β/δ (PPARβ/δ) activator, GW501516, in control of fatty acid metabolism: a new potential therapeutic target for treating metabolic syndrome.

Lee J, Chung WY.

Endocrinology · comment; journal article · DOI 10.1210/en.2011-0211

Bibliografisk träff 2009-11-28

Characterization of two major urinary metabolites of the PPARdelta-agonist GW1516 and implementation of the drug in routine doping controls.

Thevis M, Möller I, Thomas A, Beuck S, Rodchenkov G, Bornatsch W, Geyer H, Schänzer W.

Anal Bioanal Chem · research support, non-u.s. gov't; journal article · DOI 10.1007/s00216-009-3283-x

Bibliografisk träff 2007-12-01

Lipids, lipoproteins, and peroxisome proliferator activated receptor-delta.

Sprecher DL.

Am J Cardiol · review; journal article · DOI 10.1016/j.amjcard.2007.08.009

Bibliografisk träff 2006-04-01

GW-501516 GlaxoSmithKline/Ligand.

Pelton P.

Curr Opin Investig Drugs · review; journal article

Bibliografisk träff 2005-10-18

Synthesis of the PPARbeta/delta-selective agonist GW501516 and C4-thiazole-substituted analogs.

Pereira R, Gaudon C, Iglesias B, Germain P, Gronemeyer H, de Lera AR.

Bioorg Med Chem Lett · research support, non-u.s. gov't; journal article · DOI 10.1016/j.bmcl.2005.09.060

Bibliografisk träff 2004-02-01

Activation of nuclear hormone receptor peroxisome proliferator-activated receptor-delta accelerates intestinal adenoma growth.

Gupta RA, Wang D, Katkuri S, Wang H, Dey SK, DuBois RN.

Nat Med · research support, u.s. gov't, p.h.s.; research support, non-u.s. gov't; journal article · DOI 10.1038/nm993

Bibliografisk träff 2003-11-01

A short and efficient synthesis of the pharmacological research tool GW501516 for the peroxisome proliferator-activated receptor delta.

Wei ZL, Kozikowski AP.

J Org Chem · journal article · DOI 10.1021/jo035140g