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Publikationer i urvalet

50 träffar

Bibliografisk träff 2008-10-04

Quantitative structure-activity relationship and complex network approach to monoamine oxidase A and B inhibitors.

Santana L, González-Díaz H, Quezada E, Uriarte E, Yáñez M, Viña D, Orallo F.

J Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1021/jm800656v

Bibliografisk träff 2008-02-29

Discovery of a novel series of biphenyl benzoic acid derivatives as potent and selective human beta3-adrenergic receptor agonists with good oral bioavailability. Part I.

Imanishi M, Tomishima Y, Itou S, Hamashima H, Nakajima Y, Washizuka K, Sakurai M, Matsui S, Imamura E, Ueshima K, Yamamoto T, Yamamoto N, Ishikawa H, Nakano K, Unami N, Hamada K, Matsumura Y, Takamura F, Hattori K.

J Med Chem · journal article · DOI 10.1021/jm701324c

Bibliografisk träff 2007-12-12

Hemopressin is an inverse agonist of CB1 cannabinoid receptors.

Heimann AS, Gomes I, Dale CS, Pagano RL, Gupta A, de Souza LL, Luchessi AD, Castro LM, Giorgi R, Rioli V, Ferro ES, Devi LA.

Proc Natl Acad Sci U S A · research support, non-u.s. gov't; research-article; journal article; research support, n.i.h., extramural · DOI 10.1073/pnas.0706980105

Bibliografisk träff 2007-08-22

Transdermal penetration behaviour of drugs: CART-clustering, QSPR and selection of model compounds.

Baert B, Deconinck E, Van Gele M, Slodicka M, Stoppie P, Bodé S, Slegers G, Vander Heyden Y, Lambert J, Beetens J, De Spiegeleer B.

Bioorg Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1016/j.bmc.2007.07.050

Bibliografisk träff 2006-06-25

Coupling ligand structure to specific conformational switches in the beta2-adrenoceptor.

Yao X, Parnot C, Deupi X, Ratnala VR, Swaminath G, Farrens D, Kobilka B.

Nat Chem Biol · research support, non-u.s. gov't; journal article; research support, n.i.h., extramural · DOI 10.1038/nchembio801

Bibliografisk träff 2006-05-07

Identifying off-target effects and hidden phenotypes of drugs in human cells.

MacDonald ML, Lamerdin J, Owens S, Keon BH, Bilter GK, Shang Z, Huang Z, Yu H, Dias J, Minami T, Michnick SW, Westwick JK.

Nat Chem Biol · journal article · DOI 10.1038/nchembio790

Bibliografisk träff 2006-05-01

Biarylaniline phenethanolamines as potent and selective beta3 adrenergic receptor agonists.

Uehling DE, Shearer BG, Donaldson KH, Chao EY, Deaton DN, Adkison KK, Brown KK, Cariello NF, Faison WL, Lancaster ME, Lin J, Hart R, Milliken TO, Paulik MA, Sherman BW, Sugg EE, Cowan C.

J Med Chem · journal article · DOI 10.1021/jm0509445

Bibliografisk träff 2005-01-01

Discovery of a novel, potent and selective human beta3-adrenergic receptor agonist.

Nakajima Y, Hamashima H, Washizuka K, Tomishima Y, Ohtake H, Imamura E, Miura T, Kayakiri H, Kato M.

Bioorg Med Chem Lett · journal article · DOI 10.1016/j.bmcl.2004.11.001

Bibliografisk träff 2003-01-01

Relationship between stereochemistry and the beta3-adrenoceptor agonistic activity of 4'-hydroxynorephedrine derivative as an agent for treatment of frequent urination and urinary incontinence.

Tanaka N, Tamai T, Mukaiyama H, Hirabayashi A, Muranaka H, Ishikawa T, Kobayashi J, Akahane S, Akahane M.

J Med Chem · journal article · DOI 10.1021/jm020177z

Bibliografisk träff 2002-01-01

Synthesis and evaluation of potent and selective beta(3) adrenergic receptor agonists containing acylsulfonamide, sulfonylsulfonamide, and sulfonylurea carboxylic acid isosteres.

Uehling DE, Donaldson KH, Deaton DN, Hyman CE, Sugg EE, Barrett DG, Hughes RG, Reitter B, Adkison KK, Lancaster ME, Lee F, Hart R, Paulik MA, Sherman BW, True T, Cowan C.

J Med Chem · journal article · DOI 10.1021/jm0101500

Bibliografisk träff 2001-04-01

Discovery of novel N-phenylglycine derivatives as potent and selective beta(3)-adrenoceptor agonists for the treatment of frequent urination and urinary incontinence.

Tanaka N, Tamai T, Mukaiyama H, Hirabayashi A, Muranaka H, Akahane S, Miyata H, Akahane M.

J Med Chem · journal article · DOI 10.1021/jm000455z

Bibliografisk träff 2000-06-01

QSAR model for drug human oral bioavailability.

Yoshida F, Topliss JG.

J Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1021/jm0000564

Bibliografisk träff 2000-02-01

Synthesis and human beta-adrenoceptor activity of 1-(3,5-diiodo-4- methoxybenzyl)-1,2,3,4-tetrahydroisoquinolin-6-ol derivatives in vitro.

He Y, Nikulin VI, Vansal SS, Feller DR, Miller DD.

J Med Chem · research support, u.s. gov't, p.h.s.; journal article · DOI 10.1021/jm990463j

Bibliografisk träff 1999-08-01

Novel hypotensive agents from Verbesina caracasana. 6. Synthesis and pharmacology of caracasandiamide.

Carmignani M, Volpe AR, Delle Monache F, Botta B, Espinal R, De Bonnevaux SC, De Luca C, Botta M, Corelli F, Tafi A, Ripanti G, Monache GD.

J Med Chem · comparative study; research support, non-u.s. gov't; journal article · DOI 10.1021/jm991004l

Bibliografisk träff 1999-06-01

2-Amino-4-benzyl-4,5,6,7-tetrahydrothiazolo[5,4-c]pyridines: novel selective beta3-adrenoceptor agonists.

Zheng W, Nikulin VI, Konkar AA, Vansal SS, Shams G, Feller DR, Miller DD.

J Med Chem · research support, u.s. gov't, p.h.s.; research support, non-u.s. gov't; journal article · DOI 10.1021/jm990012z

Bibliografisk träff 1993-10-01

Conformationally restrained analogs of sympathomimetic catecholamines. Synthesis, conformational analysis, and adrenergic activity of isochroman derivatives.

Macchia B, Balsamo A, Breschi MC, Chiellini G, Lapucci A, Macchia M, Manera C, Martinelli A, Martini C, Scatizzi R.

J Med Chem · comparative study; research support, non-u.s. gov't; journal article · DOI 10.1021/jm00073a006

Bibliografisk träff 1992-08-01

Disodium (R,R)-5-[2-[[2-(3-chlorophenyl)-2-hydroxyethyl]-amino] propyl]-1,3-benzodioxole-2,2-dicarboxylate (CL 316,243). A potent beta-adrenergic agonist virtually specific for beta 3 receptors. A promising antidiabetic and antiobesity agent.

Bloom JD, Dutia MD, Johnson BD, Wissner A, Burns MG, Largis EE, Dolan JA, Claus TH.

J Med Chem · journal article · DOI 10.1021/jm00094a025

Bibliografisk träff 1992-05-01

Selective beta 3-adrenergic agonists of brown adipose tissue and thermogenesis. 1. [4-[2-[(2-Hydroxy-3-phenoxypropyl)amino]ethoxy]phenoxy]acetates.

Howe R, Rao BS, Holloway BR, Stribling D.

J Med Chem · journal article · DOI 10.1021/jm00088a009

Bibliografisk träff 1992-03-01

Conformational effects on the activity of drugs. 13. A revision of previously proposed models for the activation of alpha- and beta-adrenergic receptors.

Macchia B, Balsamo A, Breschi MC, Lapucci A, Lucacchini A, Macchia F, Manera C, Martinelli A, Martini C, Martinotti E.

J Med Chem · comparative study; research support, non-u.s. gov't; journal article · DOI 10.1021/jm00084a006

Bibliografisk träff 1991-03-01

Effect of fluorine substitution on the adrenergic properties of 3-(tert-butylamino)-1-(3,4-dihydroxyphenoxy)-2-propanol.

Adejare A, Nie JY, Hebel D, Brackett LE, Choi O, Gusovsky F, Padgett WL, Daly JW, Creveling CR, Kirk KL.

J Med Chem · comparative study; journal article · DOI 10.1021/jm00107a027

Bibliografisk träff 1990-07-01

Beta-adrenoceptor control of peroxidase synthesis in nasal glands.

Watanabe K, Harada H.

Ann Otol Rhinol Laryngol · journal article · DOI 10.1177/000348949009900717

Bibliografisk träff 1989-09-01

Novel secoiridoid lactones from Jasminum multiflorum.

Shen YC, Chen CH.

J Nat Prod · research support, non-u.s. gov't; journal article · DOI 10.1021/np50065a024

Bibliografisk träff 1987-09-01

Carbostyril derivatives having potent beta-adrenergic agonist properties.

Milecki J, Baker SP, Standifer KM, Ishizu T, Chida Y, Kusiak JW, Pitha J.

J Med Chem · journal article · DOI 10.1021/jm00392a006

Bibliografisk träff 1986-12-01

Cardiotonic agents. 1. Synthesis and structure-activity relationships in a new class of 3-, 4-, and 5-pyridyl-2(1H)-quinolone derivatives.

Leclerc G, Marciniak G, Decker N, Schwartz J.

J Med Chem · comparative study; journal article · DOI 10.1021/jm00162a002

Bibliografisk träff 1986-12-01

Cardiotonic agents. 2. Synthesis and structure-activity relationships in a new class of 6-, 7-, and 8-pyridyl-2(1H)-quinolone derivatives.

Leclerc G, Marciniak G, Decker N, Schwartz J.

J Med Chem · comparative study; journal article · DOI 10.1021/jm00162a003

Bibliografisk träff 1986-05-01

Conformational effects on the activity of drugs. 11. Stereostructural models for the direct activation of the alpha- and beta-adrenergic receptor.

Macchia B, Balsamo A, Epifani E, Lapucci A, Nencetti S, Macchia F, Breschi MC, Martinotti E, Ceserani R.

J Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1021/jm00155a025

Bibliografisk träff 1986-02-01

Mapping the turkey erythrocyte beta receptor: a distance geometry approach.

Linschoten MR, Bultsma T, IJzerman AP, Timmerman H.

J Med Chem · journal article · DOI 10.1021/jm00152a017

Bibliografisk träff 1986-01-01

Stereoselective syntheses of the trans-decahydroquinoline-5-carboxylic acid epimers. Diastereomeric zwitterionic probes of gamma-aminobutyric acid related biological properties in vitro and in vivo.

Witiak DT, Patch RJ, Enna SJ, Fung YK.

J Med Chem · comparative study; research support, u.s. gov't, p.h.s.; journal article · DOI 10.1021/jm00151a001

Bibliografisk träff 1985-12-01

3,4-O-diacetylisoproterenol. Preparation, structure proof, and beta-receptor effect.

Jakobsen P, Treppendahl S, Andersen PH, Klysner R, Geisler A, Teuber L.

J Med Chem · comparative study; journal article · DOI 10.1021/jm00150a036

Bibliografisk träff 1985-10-01

Cardiotonic agents. 2. Synthesis and structure-activity relationships of 4,5-dihydro-6-[4-(1H-imidazol-1-yl)phenyl]-3(2H)-pyridazinones: a new class of positive inotropic agents.

Sircar I, Duell BL, Bobowski G, Bristol JA, Evans DB.

J Med Chem · journal article · DOI 10.1021/jm00148a006