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Publikationer i urvalet

21 träffar

Bibliografisk träff 2020-03-20

Bioreductively Activatable Prodrug Conjugates of Combretastatin A-1 and Combretastatin A-4 as Anticancer Agents Targeted toward Tumor-Associated Hypoxia.

Winn BA, Devkota L, Kuch B, MacDonough MT, Strecker TE, Wang Y, Shi Z, Gerberich JL, Mondal D, Ramirez AJ, Hamel E, Chaplin DJ, Davis P, Mason RP, Trawick ML, Pinney KG.

J Nat Prod · research support, non-u.s. gov't; research-article; journal article; research support, n.i.h., extramural · DOI 10.1021/acs.jnatprod.9b00773

Bibliografisk träff 2012-06-01

An Amino-Benzosuberene Analogue That Inhibits Tubulin Assembly and Demonstrates Remarkable Cytotoxicity.

Tanpure RP, George CS, Sriram M, Strecker TE, Tidmore JK, Hamel E, Charlton-Sevcik AK, Chaplin DJ, Trawick ML, Pinney KG.

Medchemcomm · research-article; journal article · DOI 10.1039/c2md00318j

Bibliografisk träff 2012-01-18

Increased endothelial cell selectivity of triazole-bridged dihalogenated A-ring analogues of combretastatin A-1.

Beale TM, Bond PJ, Brenton JD, Charnock-Jones DS, Ley SV, Myers RM.

Bioorg Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1016/j.bmc.2012.01.010

Bibliografisk träff 2011-11-12

Synthesis, biological evaluation and molecular modeling of 1,2,3-triazole analogs of combretastatin A-1.

Akselsen OW, Odlo K, Cheng JJ, Maccari G, Botta M, Hansen TV.

Bioorg Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1016/j.bmc.2011.11.010

Bibliografisk träff 2011-06-30

Regioselective synthesis of water-soluble monophosphate derivatives of combretastatin A-1.

Tanpure RP, Nguyen BL, Strecker TE, Aguirre S, Sharma S, Chaplin DJ, Siim BG, Hamel E, Lippert JW, Pettit GR, Trawick ML, Pinney KG.

J Nat Prod · research support, non-u.s. gov't; research-article; research support, u.s. gov't, non-p.h.s.; journal article; research support, n.i.h., extramural · DOI 10.1021/np200104t

Bibliografisk träff 2010-06-01

Regio- and stereospecific synthesis of mono-beta-d-glucuronic acid derivatives of combretastatin A-1.

Tanpure RP, Strecker TE, Chaplin DJ, Siim BG, Trawick ML, Pinney KG.

J Nat Prod · research support, non-u.s. gov't; research support, u.s. gov't, non-p.h.s.; journal article · DOI 10.1021/np100108e

Bibliografisk träff 2010-03-17

Synthesis and biological evaluation of combretastatin analogs as cell cycle inhibitors of the G1 to S transition in Saccharomyces cerevisiae.

Coccetti P, Montano G, Lombardo A, Tripodi F, Orsini F, Pagliarin R.

Bioorg Med Chem Lett · research support, non-u.s. gov't; journal article · DOI 10.1016/j.bmcl.2010.03.066

Bibliografisk träff 2009-07-01

Isocombretastatins a versus combretastatins a: the forgotten isoCA-4 isomer as a highly promising cytotoxic and antitubulin agent.

Messaoudi S, Tréguier B, Hamze A, Provot O, Peyrat JF, De Losada JR, Liu JM, Bignon J, Wdzieczak-Bakala J, Thoret S, Dubois J, Brion JD, Alami M.

J Med Chem · comparative study; research support, non-u.s. gov't; journal article · DOI 10.1021/jm900321u

Bibliografisk träff 2009-03-01

Antineoplastic agents. 578. Synthesis of stilstatins 1 and 2 and their water-soluble prodrugs.

Pettit GR, Thornhill A, Melody N, Knight JC.

J Nat Prod · research support, non-u.s. gov't; journal article; research support, n.i.h., extramural · DOI 10.1021/np800608c

Bibliografisk träff 2008-07-24

Design, synthesis and biological evaluation of dihydronaphthalene and benzosuberene analogs of the combretastatins as inhibitors of tubulin polymerization in cancer chemotherapy.

Sriram M, Hall JJ, Grohmann NC, Strecker TE, Wootton T, Franken A, Trawick ML, Pinney KG.

Bioorg Med Chem · research support, non-u.s. gov't; research support, u.s. gov't, non-p.h.s.; journal article · DOI 10.1016/j.bmc.2008.07.050

Bibliografisk träff 2008-02-28

Combretastatin dinitrogen-substituted stilbene analogues as tubulin-binding and vascular-disrupting agents.

Siles R, Ackley JF, Hadimani MB, Hall JJ, Mugabe BE, Guddneppanavar R, Monk KA, Chapuis JC, Pettit GR, Chaplin DJ, Edvardsen K, Trawick ML, Garner CM, Pinney KG.

J Nat Prod · research support, non-u.s. gov't; research support, u.s. gov't, non-p.h.s.; journal article; research support, n.i.h., extramural · DOI 10.1021/np070377j

Bibliografisk träff 2005-10-01

Antineoplastic agents. 509: synthesis of fluorcombstatin phosphate and related 3-halostilbenes(1).

Pettit GR, Minardi MD, Rosenberg HJ, Hamel E, Bibby MC, Martin SW, Jung MK, Pettit RK, Cuthbertson TJ, Chapuis JC.

J Nat Prod · research support, u.s. gov't, p.h.s.; research support, non-u.s. gov't; journal article; research support, n.i.h., extramural · DOI 10.1021/np058038i

Bibliografisk träff 2003-03-01

An adjustable release rate linking strategy for cytotoxin-peptide conjugates.

Fuselier JA, Sun L, Woltering SN, Murphy WA, Vasilevich N, Coy DH.

Bioorg Med Chem Lett · journal article · DOI 10.1016/s0960-894x(03)00016-7

Bibliografisk träff 2000-07-01

Antineoplastic agents. 443. Synthesis of the cancer cell growth inhibitor hydroxyphenstatin and its sodium diphosphate prodrug.

Pettit GR, Grealish MP, Herald DL, Boyd MR, Hamel E, Pettit RK.

J Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1021/jm000045a

Bibliografisk träff 2000-07-01

Antineoplastic agents 440. Asymmetric synthesis and evaluation of the combretastatin A-1 SAR probes (1S,2S)- and (1R,2R)-1, 2-dihydroxy- 1-(2',3'-dihydroxy-4'-methoxyphenyl)-2-(3' ',4' ',5' '-trimethoxyphenyl)-ethane.

Pettit GR, Lippert JW, Herald DL, Hamel E, Pettit RK.

J Nat Prod · research support, u.s. gov't, p.h.s.; journal article · DOI 10.1021/np0000623

Bibliografisk träff 2000-04-01

Bioactive compounds from Combretum erythrophyllum.

Schwikkard S, Zhou BN, Glass TE, Sharp JL, Mattern MR, Johnson RK, Kingston DG.

J Nat Prod · research support, u.s. gov't, p.h.s.; research support, non-u.s. gov't; journal article · DOI 10.1021/np9904410

Bibliografisk träff 1999-04-01

Antineoplastic agents. 410. Asymmetric hydroxylation of trans-combretastatin A-4.

Pettit GR, Toki BE, Herald DL, Boyd MR, Hamel E, Pettit RK, Chapuis JC.

J Med Chem · research support, u.s. gov't, p.h.s.; research support, non-u.s. gov't; research support, u.s. gov't, non-p.h.s.; journal article · DOI 10.1021/jm9807149

Bibliografisk träff 1997-11-01

Isolation, synthesis, and antiplatelet aggregation activity of resveratrol 3-O-beta-D-glucopyranoside and related compounds.

Orsini F, Pelizzoni F, Verotta L, Aburjai T, Rogers CB.

J Nat Prod · research support, non-u.s. gov't; journal article · DOI 10.1021/np970069t

Bibliografisk träff 1995-05-01

Antineoplastic agents. 291. Isolation and synthesis of combretastatins A-4, A-5, and A-6(1a)

Pettit GR, Singh SB, Boyd MR, Hamel E, Pettit RK, Schmidt JM, Hogan F.

J Med Chem · research support, u.s. gov't, p.h.s.; research support, non-u.s. gov't; research support, u.s. gov't, non-p.h.s.; journal article · DOI 10.1021/jm00010a011

Bibliografisk träff 1988-05-01

Isolation, structure, synthesis, and antimitotic properties of combretastatins B-3 and B-4 from Combretum caffrum.

Pettit GR, Singh SB, Schmidt JM, Niven ML, Hamel E, Lin CM.

J Nat Prod · research support, u.s. gov't, p.h.s.; research support, non-u.s. gov't; research support, u.s. gov't, non-p.h.s.; journal article · DOI 10.1021/np50057a011

Bibliografisk träff 1987-01-01

Isolation, structure, and synthesis of combretastatins A-1 and B-1, potent new inhibitors of microtubule assembly, derived from Combretum caffrum.

Pettit GR, Singh SB, Niven ML, Hamel E, Schmidt JM.

J Nat Prod · research support, u.s. gov't, p.h.s.; research support, non-u.s. gov't; research support, u.s. gov't, non-p.h.s.; journal article · DOI 10.1021/np50049a016