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Publikationer i urvalet

15 träffar

Bibliografisk träff 2023-01-25

Design, synthesis and <i>in vitro</i> cytotoxicity evaluation of indolo-pyrazoles grafted with thiazolidinone as tubulin polymerization inhibitors.

Soni JP, Chilvery S, Sharma A, Reddy GN, Godugu C, Shankaraiah N.

RSC Med Chem · research-article; journal article · DOI 10.1039/d2md00442a

Bibliografisk träff 2021-12-30

Indole derivatives as tubulin polymerization inhibitors for the development of promising anticancer agents.

Hong Y, Zhu YY, He Q, Gu SX.

Bioorg Med Chem · review; journal article · DOI 10.1016/j.bmc.2021.116597

Bibliografisk träff 2021-02-05

Indolyl-α-keto-1,3,4-oxadiazoles: Synthesis, anti-cell proliferation activity, and inhibition of tubulin polymerization.

Tantak MP, Malik M, Klingler L, Olson Z, Kumar A, Sadana R, Kumar D.

Bioorg Med Chem Lett · research support, non-u.s. gov't; journal article · DOI 10.1016/j.bmcl.2021.127842

Bibliografisk träff 2020-10-22

Synthesis and biological evaluation of indolylglyoxylamide bisphosphonates, antimitotic microtubule-targeting derivatives of indibulin with improved aqueous solubility.

Brel VK, Artyushin OI, Chuprov-Netochin RN, Leonov SV, Semenova MN, Semenov VV.

Bioorg Med Chem Lett · research support, non-u.s. gov't; journal article · DOI 10.1016/j.bmcl.2020.127635

Bibliografisk träff 2019-11-11

Design, synthesis and biological evaluation of novel indole-based oxalamide and aminoacetamide derivatives as tubulin polymerization inhibitors.

Diao PC, Jian XE, Chen P, Huang C, Yin J, Huang JC, Li JS, Zhao PL.

Bioorg Med Chem Lett · research support, non-u.s. gov't; journal article · DOI 10.1016/j.bmcl.2019.126816

Bibliografisk träff 2019-09-11

Indole: A privileged scaffold for the design of anti-cancer agents.

Wan Y, Li Y, Yan C, Yan M, Tang Z.

Eur J Med Chem · review; journal article · DOI 10.1016/j.ejmech.2019.111691

Bibliografisk träff 2019-04-25

Resistance mechanisms and cross-resistance for a pyridine-pyrimidine amide inhibitor of microtubule polymerization.

Fox JC, Evans AT, Blomfield MP, Livingstone SK, Tenney SR, Webster JB, Perry K, Hill JT, Bikman BT, Hansen MDH.

Bioorg Med Chem Lett · journal article · DOI 10.1016/j.bmcl.2019.04.035

Bibliografisk träff 2017-05-03

Design and synthesis of bis(indolyl)ketohydrazide-hydrazones: Identification of potent and selective novel tubulin inhibitors.

Tantak MP, Klingler L, Arun V, Kumar A, Sadana R, Kumar D.

Eur J Med Chem · journal article · DOI 10.1016/j.ejmech.2017.04.078

Bibliografisk träff 2017-01-22

Synthesis of C<sub>5</sub>-tethered indolyl-3-glyoxylamide derivatives as tubulin polymerization inhibitors.

Guggilapu SD, Lalita G, Reddy TS, Prajapti SK, Nagarsenkar A, Ramu S, Brahma UR, Lakshmi UJ, Vegi GMN, Bhargava SK, Babu BN.

Eur J Med Chem · journal article · DOI 10.1016/j.ejmech.2017.01.026

Bibliografisk träff 2015-12-01

An Orally Bioavailable, Indole-3-glyoxylamide Based Series of Tubulin Polymerization Inhibitors Showing Tumor Growth Inhibition in a Mouse Xenograft Model of Head and Neck Cancer.

Colley HE, Muthana M, Danson SJ, Jackson LV, Brett ML, Harrison J, Coole SF, Mason DP, Jennings LR, Wong M, Tulasi V, Norman D, Lockey PM, Williams L, Dossetter AG, Griffen EJ, Thompson MJ.

J Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1021/acs.jmedchem.5b01312

Bibliografisk träff 2012-07-14

Identification of selective tubulin inhibitors as potential anti-trypanosomal agents.

Lama R, Sandhu R, Zhong B, Li B, Su B.

Bioorg Med Chem Lett · research support, non-u.s. gov't; research-article; journal article; research support, n.i.h., extramural · DOI 10.1016/j.bmcl.2012.07.023

Bibliografisk träff 2009-10-01

Indolobenzazepin-7-ones and 6-, 8-, and 9-membered ring derivatives as tubulin polymerization inhibitors: synthesis and structure--activity relationship studies.

Putey A, Popowycz F, Do QT, Bernard P, Talapatra SK, Kozielski F, Galmarini CM, Joseph B.

J Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1021/jm900476c

Bibliografisk träff 2009-07-25

Synthesis and structure-activity relationships of N-aryl(indol-3-yl)glyoxamides as antitumor agents.

Marchand P, Antoine M, Le Baut G, Czech M, Baasner S, Günther E.

Bioorg Med Chem · journal article · DOI 10.1016/j.bmc.2009.07.048

Bibliografisk träff 2008-02-16

Indole- and indolizine-glyoxylamides displaying cytotoxicity against multidrug resistant cancer cell lines.

James DA, Koya K, Li H, Liang G, Xia Z, Ying W, Wu Y, Sun L.

Bioorg Med Chem Lett · journal article · DOI 10.1016/j.bmcl.2008.02.029

Bibliografisk träff 2003-04-01

Synthesis and biological evaluation of N-heterocyclic indolyl glyoxylamides as orally active anticancer agents.

Li WT, Hwang DR, Chen CP, Shen CW, Huang CL, Chen TW, Lin CH, Chang YL, Chang YY, Lo YK, Tseng HY, Lin CC, Song JS, Chen HC, Chen SJ, Wu SH, Chen CT.

J Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1021/jm020471r