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Publikationer i urvalet

25 träffar

Bibliografisk träff 2022-08-19

Exploring gabosine and chlorogentisyl alcohol derivatives from a marine-derived fungus as EcGUS inhibitors with informatic assisted approaches.

Ge Y, Ma Y, Zhao M, Wei J, Wu X, Zhang Z, Yang H, Lei H, Wu B.

Eur J Med Chem · journal article · DOI 10.1016/j.ejmech.2022.114699

Bibliografisk träff 2021-02-25

Structure-Activity Relationship Studies of Coumarin-like Diacid Derivatives as Human G Protein-Coupled Receptor-35 (hGPR35) Agonists and a Consequent New Design Principle.

Wei L, Hou T, Li J, Zhang X, Zhou H, Wang Z, Cheng J, Xiang K, Wang J, Zhao Y, Liang X.

J Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1021/acs.jmedchem.0c01624

Bibliografisk träff 2018-03-15

The identification of inhibitory compounds of Rickettsia prowazekii methionine aminopeptidase for antibacterial applications.

Helgren TR, Seven ES, Chen C, Edwards TE, Staker BL, Abendroth J, Myler PJ, Horn JR, Hagen TJ.

Bioorg Med Chem Lett · research-article; journal article; research support, n.i.h., extramural · DOI 10.1016/j.bmcl.2018.03.002

Bibliografisk träff 2016-12-28

Discovery of 2H-Chromen-2-one Derivatives as G Protein-Coupled Receptor-35 Agonists.

Wei L, Wang J, Zhang X, Wang P, Zhao Y, Li J, Hou T, Qu L, Shi L, Liang X, Fang Y.

J Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1021/acs.jmedchem.6b01431

Bibliografisk träff 2016-12-05

Structure-activity relationships of benzothiazole GPR35 antagonists.

Abdalhameed MM, Zhao P, Hurst DP, Reggio PH, Abood ME, Croatt MP.

Bioorg Med Chem Lett · research-article; journal article; research support, n.i.h., extramural · DOI 10.1016/j.bmcl.2016.12.012

Bibliografisk träff 2013-08-15

6-Bromo-8-(4-[(3)H]methoxybenzamido)-4-oxo-4H-chromene-2-carboxylic Acid: a powerful tool for studying orphan G protein-coupled receptor GPR35.

Thimm D, Funke M, Meyer A, Müller CE.

J Med Chem · journal article · DOI 10.1021/jm4009373

Bibliografisk träff 2013-06-17

8-Benzamidochromen-4-one-2-carboxylic acids: potent and selective agonists for the orphan G protein-coupled receptor GPR35.

Funke M, Thimm D, Schiedel AC, Müller CE.

J Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1021/jm400587g

Bibliografisk träff 2013-04-09

Structure-based identification of OATP1B1/3 inhibitors.

De Bruyn T, van Westen GJ, Ijzerman AP, Stieger B, de Witte P, Augustijns PF, Annaert PP.

Mol Pharmacol · research support, non-u.s. gov't; journal article · DOI 10.1124/mol.112.084152

Bibliografisk träff 2012-06-04

4-quinolones as noncovalent inhibitors of high molecular mass penicillin-binding proteins.

Shilabin AG, Dzhekieva L, Misra P, Jayaram B, Pratt RF.

ACS Med Chem Lett · rapid-communication; journal article · DOI 10.1021/ml3001006

Bibliografisk träff 2012-04-21

Thieno[3,2-b]thiophene-2-carboxylic acid derivatives as GPR35 agonists.

Deng H, Hu J, Hu H, He M, Fang Y.

Bioorg Med Chem Lett · journal article · DOI 10.1016/j.bmcl.2012.04.057

Bibliografisk träff 2011-10-18

Synthesis and biological effects of some kynurenic acid analogs.

Nagy K, Plangár I, Tuka B, Gellért L, Varga D, Demeter I, Farkas T, Kis Z, Marosi M, Zádori D, Klivényi P, Fülöp F, Szatmári I, Vécsei L, Toldi J.

Bioorg Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1016/j.bmc.2011.10.029

Bibliografisk träff 2007-04-08

Chemical genetics reveals a complex functional ground state of neural stem cells.

Diamandis P, Wildenhain J, Clarke ID, Sacher AG, Graham J, Bellows DS, Ling EK, Ward RJ, Jamieson LG, Tyers M, Dirks PB.

Nat Chem Biol · research support, non-u.s. gov't; journal article · DOI 10.1038/nchembio873

Bibliografisk träff 2002-05-01

Synthesis and in vitro pharmacology of substituted quinoline-2,4-dicarboxylic acids as inhibitors of vesicular glutamate transport.

Carrigan CN, Bartlett RD, Esslinger CS, Cybulski KA, Tongcharoensirikul P, Bridges RJ, Thompson CM.

J Med Chem · research support, u.s. gov't, p.h.s.; research support, non-u.s. gov't; research support, u.s. gov't, non-p.h.s.; journal article · DOI 10.1021/jm010261z

Bibliografisk träff 1999-09-01

Quinoline-2,4-dicarboxylic acids: synthesis and evaluation as inhibitors of the glutamate vesicular transport system.

Carrigan CN, Esslinger CS, Bartlett RD, Bridges RJ, Thompson CM.

Bioorg Med Chem Lett · research support, u.s. gov't, p.h.s.; research support, non-u.s. gov't; journal article · DOI 10.1016/s0960-894x(99)00444-8

Bibliografisk träff 1998-02-01

Transtorine, a new quinoline alkaloid from Ephedra transitoria.

al-Khalil S, Alkofahi A, el-Eisawi D, al-Shibib A.

J Nat Prod · research support, non-u.s. gov't; journal article · DOI 10.1021/np9702998

Bibliografisk träff 1995-10-01

Kynurenic acid derivatives inhibit the binding of nerve growth factor (NGF) to the low-affinity p75 NGF receptor.

Jaen JC, Laborde E, Bucsh RA, Caprathe BW, Sorenson RJ, Fergus J, Spiegel K, Marks J, Dickerson MR, Davis RE.

J Med Chem · journal article · DOI 10.1021/jm00022a008

Bibliografisk träff 1994-11-01

The glycine site on the NMDA receptor: structure-activity relationships and therapeutic potential.

Leeson PD, Iversen LL.

J Med Chem · review; journal article · DOI 10.1021/jm00050a001

Bibliografisk träff 1992-09-01

3-Phenyl-4-hydroxyquinolin-2(1H)-ones: potent and selective antagonists at the strychnine-insensitive glycine site on the N-methyl-D-aspartate receptor complex.

McQuaid LA, Smith EC, Lodge D, Pralong E, Wikel JH, Calligaro DO, O'Malley PJ.

J Med Chem · journal article · DOI 10.1021/jm00096a019

Bibliografisk träff 1992-05-01

3-(2-Carboxyindol-3-yl)propionic acid-based antagonists of the N-methyl-D-aspartic acid receptor associated glycine binding site.

Salituro FG, Harrison BL, Baron BM, Nyce PL, Stewart KT, Kehne JH, White HS, McDonald IA.

J Med Chem · journal article · DOI 10.1021/jm00088a014

Bibliografisk träff 1992-05-01

2-Carboxytetrahydroquinolines. Conformational and stereochemical requirements for antagonism of the glycine site on the NMDA receptor.

Carling RW, Leeson PD, Moseley AM, Baker R, Foster AC, Grimwood S, Kemp JA, Marshall GR.

J Med Chem · comparative study; journal article · DOI 10.1021/jm00089a003

Bibliografisk träff 1991-04-01

Kynurenic acid derivatives. Structure-activity relationships for excitatory amino acid antagonism and identification of potent and selective antagonists at the glycine site on the N-methyl-D-aspartate receptor.

Leeson PD, Baker R, Carling RW, Curtis NR, Moore KW, Williams BJ, Foster AC, Donald AE, Kemp JA, Marshall GR.

J Med Chem · comparative study; journal article · DOI 10.1021/jm00108a002

Bibliografisk träff 1990-12-01

4-[(Carboxymethyl)oxy]- and 4-[(carboxymethyl)amino]-5,7-dichloroquinoline-2-carboxylic acid: new antagonists of the strychnine-insensitive glycine binding site on the N-methyl-D-aspartate receptor complex.

Harrison BL, Baron BM, Cousino DM, McDonald IA.

J Med Chem · comparative study; journal article · DOI 10.1021/jm00174a005

Bibliografisk träff 1990-11-01

3-(2-carboxyindol-3-yl)propionic acid derivatives: antagonists of the strychnine-insensitive glycine receptor associated with the N-methyl-D-aspartate receptor complex.

Salituro FG, Harrison BL, Baron BM, Nyce PL, Stewart KT, McDonald IA.

J Med Chem · comparative study; journal article · DOI 10.1021/jm00173a003

Bibliografisk träff 1978-09-01

Structure-activity correlations for a series of antiallergy agents. Oxanilic, quinaldic, and benzopyran-2-carboxylic acids.

Cheney BV, Wright JB, Hall CM, Johnson HG.

J Med Chem · journal article · DOI 10.1021/jm00207a017

Bibliografisk träff 1978-09-01

Antiallergic activity of tetracyclic derivatives of quinoline-2-carboxylic acids. 1.

Erickson EH, Lappi LR, Rice TK, Swingle KF, Van Winkle M.

J Med Chem · journal article · DOI 10.1021/jm00207a026