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Publikationer i urvalet

27 träffar

Bibliografisk träff 2017-03-13

In silico design of novel probes for the atypical opioid receptor MRGPRX2.

Lansu K, Karpiak J, Liu J, Huang XP, McCorvy JD, Kroeze WK, Che T, Nagase H, Carroll FI, Jin J, Shoichet BK, Roth BL.

Nat Chem Biol · research-article; journal article · DOI 10.1038/nchembio.2334

Bibliografisk träff 2009-09-06

Genetic mapping of targets mediating differential chemical phenotypes in Plasmodium falciparum.

Yuan J, Johnson RL, Huang R, Wichterman J, Jiang H, Hayton K, Fidock DA, Wellems TE, Inglese J, Austin CP, Su XZ.

Nat Chem Biol · research support, n.i.h., intramural; research-article; journal article; research support, n.i.h., extramural · DOI 10.1038/nchembio.215

Bibliografisk träff 2008-11-24

Redefining the structure-activity relationships of 2,6-methano-3-benzazocines. Part 7: syntheses and opioid receptor properties of cyclic variants of cyclazocine.

Wentland MP, Lu Q, Ganorkar R, Zhang SZ, Jo S, Cohen DJ, Bidlack JM.

Bioorg Med Chem Lett · research support, u.s. gov't, non-p.h.s.; journal article; research support, n.i.h., extramural · DOI 10.1016/j.bmcl.2008.11.076

Bibliografisk träff 2008-11-07

Syntheses and opioid receptor binding properties of carboxamido-substituted opioids.

Wentland MP, Lou R, Lu Q, Bu Y, VanAlstine MA, Cohen DJ, Bidlack JM.

Bioorg Med Chem Lett · research support, u.s. gov't, non-p.h.s.; journal article; research support, n.i.h., extramural · DOI 10.1016/j.bmcl.2008.10.134

Bibliografisk träff 2008-01-01

Development of a phospholipidosis database and predictive quantitative structure-activity relationship (QSAR) models.

Kruhlak NL, Choi SS, Contrera JF, Weaver JL, Willard JM, Hastings KL, Sancilio LF.

Toxicol Mech Methods · journal article · DOI 10.1080/15376510701857262

Bibliografisk träff 2007-11-21

Identification of new functional inhibitors of acid sphingomyelinase using a structure-property-activity relation model.

Kornhuber J, Tripal P, Reichel M, Terfloth L, Bleich S, Wiltfang J, Gulbins E.

J Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1021/jm070524a

Bibliografisk träff 2007-04-08

Chemical genetics reveals a complex functional ground state of neural stem cells.

Diamandis P, Wildenhain J, Clarke ID, Sacher AG, Graham J, Bellows DS, Ling EK, Ward RJ, Jamieson LG, Tyers M, Dirks PB.

Nat Chem Biol · research support, non-u.s. gov't; journal article · DOI 10.1038/nchembio873

Bibliografisk träff 2003-06-01

Redefining the structure-activity relationships of 2,6-methano-3-benzazocines. Part 2: 8-formamidocyclazocine analogues.

Wentland MP, Sun X, Ye Y, Lou R, Bidlack JM.

Bioorg Med Chem Lett · research support, u.s. gov't, p.h.s.; journal article · DOI 10.1016/s0960-894x(03)00295-6

Bibliografisk träff 2003-02-01

Syntheses and opioid receptor binding affinities of 8-amino-2,6-methano-3-benzazocines.

Wentland MP, Ye Y, Cioffi CL, Lou R, Zhou Q, Xu G, Duan W, Dehnhardt CM, Sun X, Cohen DJ, Bidlack JM.

J Med Chem · research support, u.s. gov't, p.h.s.; journal article · DOI 10.1021/jm020429w

Bibliografisk träff 2001-07-01

3-Carboxamido analogues of morphine and naltrexone. synthesis and opioid receptor binding properties.

Wentland MP, Lou R, Dehnhardt CM, Duan W, Cohen DJ, Bidlack JM.

Bioorg Med Chem Lett · research support, u.s. gov't, p.h.s.; journal article · DOI 10.1016/s0960-894x(01)00278-5

Bibliografisk träff 2001-03-01

8-Carboxamidocyclazocine analogues: redefining the structure-activity relationships of 2,6-methano-3-benzazocines.

Wentland MP, Lou R, Ye Y, Cohen DJ, Richardson GP, Bidlack JM.

Bioorg Med Chem Lett · research support, u.s. gov't, p.h.s.; journal article · DOI 10.1016/s0960-894x(01)00014-2

Bibliografisk träff 2000-09-01

Selective protection and functionalization of morphine: synthesis and opioid receptor binding properties of 3-amino-3-desoxymorphine derivatives.

Wentland MP, Duan W, Cohen DJ, Bidlack JM.

J Med Chem · research support, u.s. gov't, p.h.s.; journal article · DOI 10.1021/jm000119i

Bibliografisk träff 2000-06-01

Predicting blood-brain barrier permeation from three-dimensional molecular structure.

Crivori P, Cruciani G, Carrupt PA, Testa B.

J Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1021/jm990968+

Bibliografisk träff 2000-01-01

Synthesis and opioid receptor affinity of morphinan and benzomorphan derivatives: mixed kappa agonists and mu agonists/antagonists as potential pharmacotherapeutics for cocaine dependence.

Neumeyer JL, Bidlack JM, Zong R, Bakthavachalam V, Gao P, Cohen DJ, Negus SS, Mello NK.

J Med Chem · research support, u.s. gov't, p.h.s.; research support, non-u.s. gov't; journal article · DOI 10.1021/jm9903343

Bibliografisk träff 2000-01-01

8-Aminocyclazocine analogues: synthesis and structure-activity relationships.

Wentland MP, Xu G, Cioffi CL, Ye Y, Duan W, Cohen DJ, Colasurdo AM, Bidlack JM.

Bioorg Med Chem Lett · research support, u.s. gov't, p.h.s.; journal article · DOI 10.1016/s0960-894x(99)00670-8

Bibliografisk träff 1993-04-01

The role of receptor binding in drug discovery.

Sweetnam PM, Caldwell L, Lancaster J, Bauer C, McMillan B, Kinnier WJ, Price CH.

J Nat Prod · research support, u.s. gov't, p.h.s.; review; journal article · DOI 10.1021/np50094a001

Bibliografisk träff 1992-07-01

Enantiomeric N-substituted N-normetazocines: a comparative study of affinities at sigma, PCP, and mu opioid receptors.

Carroll FI, Abraham P, Parham K, Bai X, Zhang X, Brine GA, Mascarella SW, Martin BR, May EL, Sauss C.

J Med Chem · comparative study; research support, u.s. gov't, p.h.s.; journal article · DOI 10.1021/jm00093a014

Bibliografisk träff 1988-03-01

Structure-activity relationships for drugs binding to the agonist and antagonist states of the primary morphine receptor.

Cheney BV.

J Med Chem · journal article · DOI 10.1021/jm00398a007

Bibliografisk träff 1988-03-01

Synthesis and analgesic properties of N-substituted trans-4a-aryldecahydroisoquinolines.

Zimmerman DM, Cantrell BE, Swartzendruber JK, Jones ND, Mendelsohn LG, Leander JD, Nickander RC.

J Med Chem · journal article · DOI 10.1021/jm00398a011

Bibliografisk träff 1981-12-01

Analgesic narcotic antagonists. 9. 6-Methylene-8 beta-alkyl-N-(cycloalkylmethyl)-3-hydroxy- or -methoxymorphinans.

Polazzi JO, Kotick MP, Howes JF, Bousquet AR.

J Med Chem · journal article · DOI 10.1021/jm00144a029

Bibliografisk träff 1981-12-01

Analgesic narcotic antagonists. 8. 7 alpha-Alkyl-4,5 alpha-epoxymorphinan-6-ones.

Kotick MP, Leland DL, Polazzi JO, Howes JF, Bousquet AR.

J Med Chem · journal article · DOI 10.1021/jm00144a015

Bibliografisk träff 1981-06-01

Analgesic narcotic antagonists. 5. 7,7-Dimethyldihydrocodeinones and 7,7-dimethyldihydromorphinones.

Leland DL, Kotick MP.

J Med Chem · comparative study; journal article · DOI 10.1021/jm00138a015

Bibliografisk träff 1980-12-01

Analgesic narcotic antagonists. 4. 7-Methyl-N-(cycloalkylmethyl)-3-hydroxymorphinan-6-ones and -isomorphinan-6-ones.

Leland DL, Kotick MP.

J Med Chem · journal article · DOI 10.1021/jm00186a025

Bibliografisk träff 1980-02-01

Analgesic narcotic antagonists. 2. 8-Alkymorphinan-6-ones.

Polazzi JO, Schut RN, Kotick MP, Howes JF, Osgood PF, Razdan RK, Villarreal JE.

J Med Chem · journal article · DOI 10.1021/jm00176a013

Bibliografisk träff 1980-01-01

Synthesis and pharmacology of 8-amino-3-(cyclopropylmethyl)-1,2,3,4,5,6-hexahydro-cis-6,11-dimethyl-2,6-methano-3-benzazocine and related compounds.

Wentland MP, Albertson NF, Pierson AK.

J Med Chem · journal article · DOI 10.1021/jm00175a013

Bibliografisk träff 1979-10-01

(2,6-Methano-3-benzazocin-11 beta-yl)alkanones. 1. Alkylalkanones: a new series of N-methyl derivatives with novel opiate activity profiles.

Michne WF, Lewis TR, Michalec SJ, Pierson AK, Rosenberg FJ.

J Med Chem · journal article · DOI 10.1021/jm00196a002

Bibliografisk träff 1977-05-01

Synthesis and narcotic agonist-antagonist evaluation of some 2,6-methano-3-benzazocine-11 propanols. Analogues of the ring C bridged oripavine-7-mehtanols.

Michne WF, Salsbury RL, Michalec SJ.

J Med Chem · journal article · DOI 10.1021/jm00215a013