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Publikationer i urvalet

12 träffar

Bibliografisk träff 2024-07-15

Electrophile Determines Cellular Phenotypes among XPO1-Targeting Small Molecules.

Chen YF, Shen Y, Yan DF, Ghazala M, Scemama de Gialluly MA, Srinivasan R, Farrar AN, Friedrich RM, Adams DJ.

J Med Chem · research support, non-u.s. gov't; journal article; research support, n.i.h., extramural · DOI 10.1021/acs.jmedchem.4c00754

Bibliografisk träff 2019-06-05

Dual FLT3 inhibitors: Against the drug resistance of acute myeloid leukemia in recent decade.

Yuan T, Qi B, Jiang Z, Dong W, Zhong L, Bai L, Tong R, Yu J, Shi J.

Eur J Med Chem · review; journal article · DOI 10.1016/j.ejmech.2019.06.002

Bibliografisk träff 2019-03-07

Recent advancements of 4-aminoquinazoline derivatives as kinase inhibitors and their applications in medicinal chemistry.

Das D, Hong J.

Eur J Med Chem · review; journal article · DOI 10.1016/j.ejmech.2019.03.004

Bibliografisk träff 2014-05-27

Small molecule inhibitors targeting activator protein 1 (AP-1).

Ye N, Ding Y, Wild C, Shen Q, Zhou J.

J Med Chem · research support, non-u.s. gov't; review-article; journal article; research support, n.i.h., extramural · DOI 10.1021/jm5004733

Bibliografisk träff 2014-04-24

Discovery of thienopyrimidine-based FLT3 inhibitors from the structural modification of known IKKβ inhibitors.

Park CH, Lee C, Yang JS, Joe BY, Chun K, Kim H, Kim HY, Kang JS, Lee JI, Kim MH, Han G.

Bioorg Med Chem Lett · research support, non-u.s. gov't; journal article · DOI 10.1016/j.bmcl.2014.04.058

Bibliografisk träff 2009-12-11

Inhibition of IKK-beta: a new development in the mechanism of the anti-obesity effects of PTP1B inhibitors SA18 and SA32.

Bhattarai BR, Ko JH, Shrestha S, Kafle B, Cho H, Kang JH, Cho H.

Bioorg Med Chem Lett · comparative study; research support, non-u.s. gov't; journal article · DOI 10.1016/j.bmcl.2009.12.033

Bibliografisk träff 2009-02-26

IKKbeta inhibitors identification part I: homology model assisted structure based virtual screening.

Nagarajan S, Doddareddy Mr, Choo H, Cho YS, Oh KS, Lee BH, Pae AN.

Bioorg Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1016/j.bmc.2009.02.041

Bibliografisk träff 2008-12-25

Discovery of novel small molecule cell type-specific enhancers of NF-kappaB nuclear translocation.

Gong G, Xie Y, Liu Y, Rinderspacher A, Deng SX, Feng Y, Zhu Z, Tang Y, Wyler M, Aulner N, Toebben U, Smith DH, Branden L, Chung C, Schürer S, Vidović D, Landry DW.

Bioorg Med Chem Lett · journal article; research support, n.i.h., extramural · DOI 10.1016/j.bmcl.2008.12.086

Bibliografisk träff 2008-12-16

3D-QSAR studies on the inhibitors of AP-1 and NF-kappaB mediated transcriptional activation.

Qin J, Liu H, Li J, Ren Y, Yao X, Liu M.

Eur J Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1016/j.ejmech.2008.12.006

Bibliografisk träff 2008-04-29

Synthesis and structure-activity relationship of aminopyrimidine IKK2 inhibitors.

Bingham AH, Davenport RJ, Fosbeary R, Gowers L, Knight RL, Lowe C, Owen DA, Parry DM, Pitt WR.

Bioorg Med Chem Lett · journal article · DOI 10.1016/j.bmcl.2008.04.062

Bibliografisk träff 2007-10-30

Identification of N-(quinolin-8-yl)benzenesulfonamides as agents capable of down-regulating NFkappaB activity within two separate high-throughput screens of NFkappaB activation.

Xie Y, Deng S, Thomas CJ, Liu Y, Zhang YQ, Rinderspacher A, Huang W, Gong G, Wyler M, Cayanis E, Aulner N, Többen U, Chung C, Pampou S, Southall N, Vidović D, Schürer S, Branden L, Davis RE, Staudt LM, Inglese J, Austin CP, Landry DW, Smith DH, Auld DS.

Bioorg Med Chem Lett · research support, n.i.h., intramural; research-article; journal article; research support, n.i.h., extramural · DOI 10.1016/j.bmcl.2007.10.100

Bibliografisk träff 2003-11-01

The design and synthesis of novel orally active inhibitors of AP-1 and NF-kappaB mediated transcriptional activation. SAR of in vitro and in vivo studies.

Palanki MS, Erdman PE, Ren M, Suto M, Bennett BL, Manning A, Ransone L, Spooner C, Desai S, Ow A, Totsuka R, Tsao P, Toriumi W.

Bioorg Med Chem Lett · comparative study; journal article · DOI 10.1016/j.bmcl.2003.08.047