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Publikationer i urvalet

8 träffar

Bibliografisk träff 2009-01-01

Total synthesis and biological evaluation of tubulysin U, tubulysin V, and their analogues.

Balasubramanian R, Raghavan B, Begaye A, Sackett DL, Fecik RA.

J Med Chem · research support, non-u.s. gov't; research-article; research support, u.s. gov't, non-p.h.s.; journal article; research support, n.i.h., extramural · DOI 10.1021/jm8013579

Bibliografisk träff 2008-03-20

Tubulysin analogs incorporating desmethyl and dimethyl tubuphenylalanine derivatives.

Balasubramanian R, Raghavan B, Steele JC, Sackett DL, Fecik RA.

Bioorg Med Chem Lett · research support, n.i.h., intramural; comparative study; research support, non-u.s. gov't; research support, u.s. gov't, non-p.h.s.; journal article · DOI 10.1016/j.bmcl.2008.03.046

Bibliografisk träff 2008-03-04

Cytotoxic simplified tubulysin analogues.

Raghavan B, Balasubramanian R, Steele JC, Sackett DL, Fecik RA.

J Med Chem · research support, n.i.h., intramural; research support, non-u.s. gov't; research support, u.s. gov't, non-p.h.s.; journal article · DOI 10.1021/jm701321p

Bibliografisk träff 2004-11-01

Synthesis and activity of novel analogs of hemiasterlin as inhibitors of tubulin polymerization: modification of the A segment.

Yamashita A, Norton EB, Kaplan JA, Niu C, Loganzo F, Hernandez R, Beyer CF, Annable T, Musto S, Discafani C, Zask A, Ayral-Kaloustian S.

Bioorg Med Chem Lett · journal article · DOI 10.1016/j.bmcl.2004.08.024

Bibliografisk träff 2004-09-01

Synthesis and biological activity of analogues of the antimicrotubule agent N,beta,beta-trimethyl-L-phenylalanyl-N(1)-[(1S,2E)-3-carboxy-1-isopropylbut-2-enyl]- N(1),3-dimethyl-L-valinamide (HTI-286).

Zask A, Birnberg G, Cheung K, Kaplan J, Niu C, Norton E, Suayan R, Yamashita A, Cole D, Tang Z, Krishnamurthy G, Williamson R, Khafizova G, Musto S, Hernandez R, Annable T, Yang X, Discafani C, Beyer C, Greenberger LM, Loganzo F, Ayral-Kaloustian S.

J Med Chem · journal article · DOI 10.1021/jm040056u

Bibliografisk träff 2004-08-01

Tubulin inhibitors. Synthesis and biological activity of HTI-286 analogs with B-segment heterosubstituents.

Niu C, Smith D, Zask A, Loganzo F, Discafani C, Beyer C, Greenberger L, Ayral-Kaloustian S.

Bioorg Med Chem Lett · journal article · DOI 10.1016/j.bmcl.2004.05.077

Bibliografisk träff 2004-08-01

D-piece modifications of the hemiasterlin analog HTI-286 produce potent tubulin inhibitors.

Zask A, Birnberg G, Cheung K, Kaplan J, Niu C, Norton E, Yamashita A, Beyer C, Krishnamurthy G, Greenberger LM, Loganzo F, Ayral-Kaloustian S.

Bioorg Med Chem Lett · journal article · DOI 10.1016/j.bmcl.2004.05.005

Bibliografisk träff 2003-02-01

Synthesis and antimitotic/cytotoxic activity of hemiasterlin analogues.

Nieman JA, Coleman JE, Wallace DJ, Piers E, Lim LY, Roberge M, Andersen RJ.

J Nat Prod · research support, u.s. gov't, p.h.s.; research support, non-u.s. gov't; journal article · DOI 10.1021/np020375t