Antiplasmodial alkaloids from Desmos rostrata.
Nguyen NT, Pham VC, Litaudon M, Guéritte F, Grellier P, Nguyen VT, Nguyen VH.
J Nat Prod · research support, non-u.s. gov't; journal article · DOI 10.1021/np8004437 PUBLIKATIONSREGISTRET
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Sirisoma N, Kasibhatla S, Pervin A, Zhang H, Jiang S, Willardsen JA, Anderson MB, Baichwal V, Mather GG, Jessing K, Hussain R, Hoang K, Pleiman CM, Tseng B, Drewe J, Cai SX.
J Med Chem · journal article · DOI 10.1021/jm8003653Design, synthesis, and biological evaluation of new-generation taxoids.
Ojima I, Chen J, Sun L, Borella CP, Wang T, Miller ML, Lin S, Geng X, Kuznetsova L, Qu C, Gallager D, Zhao X, Zanardi I, Xia S, Horwitz SB, Mallen-St Clair J, Guerriero JL, Bar-Sagi D, Veith JM, Pera P, Bernacki RJ.
J Med Chem · research support, non-u.s. gov't; research-article; journal article; research support, n.i.h., extramural · DOI 10.1021/jm800086eDesign, synthesis and biological evaluation of novel fluorinated docetaxel analogues.
Lu HF, Sun X, Xu L, Lou LG, Lin GQ.
Eur J Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1016/j.ejmech.2008.04.004Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
Obach RS, Lombardo F, Waters NJ.
Drug Metab Dispos · journal article · DOI 10.1124/dmd.108.020479Cytotoxic diterpenoids and sesquiterpenoids from Pteris multifida.
Ge X, Ye G, Li P, Tang WJ, Gao JL, Zhao WM.
J Nat Prod · journal article · DOI 10.1021/np0706421Synthesis and biological evaluation of imidazol-2-one derivatives as potential antitumor agents.
Xue N, Yang X, Wu R, Chen J, He Q, Yang B, Lu X, Hu Y.
Bioorg Med Chem · journal article · DOI 10.1016/j.bmc.2007.11.048ATP-competitive inhibitors of the mitotic kinesin KSP that function via an allosteric mechanism.
Luo L, Parrish CA, Nevins N, McNulty DE, Chaudhari AM, Carson JD, Sudakin V, Shaw AN, Lehr R, Zhao H, Sweitzer S, Lad L, Wood KW, Sakowicz R, Annan RS, Huang PS, Jackson JR, Dhanak D, Copeland RA, Auger KR.
Nat Chem Biol · journal article · DOI 10.1038/nchembio.2007.34New functional assay of P-glycoprotein activity using Hoechst 33342.
Müller H, Klinkhammer W, Globisch C, Kassack MU, Pajeva IK, Wiese M.
Bioorg Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1016/j.bmc.2007.07.024Selective induction of chemotherapy resistance of mammary tumors in a conditional mouse model for hereditary breast cancer.
Rottenberg S, Nygren AO, Pajic M, van Leeuwen FW, van der Heijden I, van de Wetering K, Liu X, de Visser KE, Gilhuijs KG, van Tellingen O, Schouten JP, Jonkers J, Borst P.
Proc Natl Acad Sci U S A · research support, non-u.s. gov't; research-article; journal article · DOI 10.1073/pnas.0702955104Synthesis and antiproliferative activities of isoindigo and azaisoindigo derivatives.
Bouchikhi F, Anizon F, Moreau P.
Eur J Med Chem · journal article · DOI 10.1016/j.ejmech.2007.05.012Paclitaxel C-10 carbamates: potential candidates for the treatment of neurodegenerative tauopathies.
Ballatore C, Hyde E, Deiches RF, Lee VM, Trojanowski JQ, Huryn D, Smith AB.
Bioorg Med Chem Lett · research-article; journal article · DOI 10.1016/j.bmcl.2007.04.058Synthesis and evaluation of new arylbenzo[b]thiophene and diarylthiophene derivatives as inhibitors of the NorA multidrug transporter of Staphylococcus aureus.
Fournier Dit Chabert J, Marquez B, Neville L, Joucla L, Broussous S, Bouhours P, David E, Pellet-Rostaing S, Marquet B, Moreau N, Lemaire M.
Bioorg Med Chem · journal article · DOI 10.1016/j.bmc.2007.04.023Synthesis and evaluation of water-soluble docetaxel prodrugs-docetaxel esters of malic acid.
Du W, Hong L, Yao T, Yang X, He Q, Yang B, Hu Y.
Bioorg Med Chem · journal article · DOI 10.1016/j.bmc.2007.04.002Potentiation of mammary cancer inhibition by combination of antagonists of growth hormone-releasing hormone with docetaxel.
Buchholz S, Schally AV, Engel JB, Hohla F, Heinrich E, Koester F, Varga JL, Halmos G.
Proc Natl Acad Sci U S A · research support, non-u.s. gov't; research-article; research support, u.s. gov't, non-p.h.s.; journal article · DOI 10.1073/pnas.0610860104Cyclostreptin binds covalently to microtubule pores and lumenal taxoid binding sites.
Buey RM, Calvo E, Barasoain I, Pineda O, Edler MC, Matesanz R, Cerezo G, Vanderwal CD, Day BW, Sorensen EJ, López JA, Andreu JM, Hamel E, Díaz JF.
Nat Chem Biol · research support, non-u.s. gov't; journal article · DOI 10.1038/nchembio853Synthesis and SAR of [1,2,4]triazolo[1,5-a]pyrimidines, a class of anticancer agents with a unique mechanism of tubulin inhibition.
Zhang N, Ayral-Kaloustian S, Nguyen T, Afragola J, Hernandez R, Lucas J, Gibbons J, Beyer C.
J Med Chem · journal article · DOI 10.1021/jm060717iNovel C2-C3' N-peptide linked macrocyclic taxoids. Part 2: synthesis and biological activities of docetaxel analogues with a peptide side chain at C2 and their macrocyclic derivatives.
Larroque AL, Dubois J, Thoret S, Aubert G, Chiaroni A, Guéritte F, Guénard D.
Bioorg Med Chem · journal article · DOI 10.1016/j.bmc.2006.09.030Cytotoxic monotetrahydrofuran acetogenins from Disepalum plagioneurum.
Eparvier V, Nguyen VH, Thoison O, Martin MT, Sévenet T, Guéritte F.
J Nat Prod · research support, non-u.s. gov't; journal article · DOI 10.1021/np060168jSyntheses and evaluation of novel fatty acid-second-generation taxoid conjugates as promising anticancer agents.
Kuznetsova L, Chen J, Sun L, Wu X, Pepe A, Veith JM, Pera P, Bernacki RJ, Ojima I.
Bioorg Med Chem Lett · research support, non-u.s. gov't; journal article; research support, n.i.h., extramural · DOI 10.1016/j.bmcl.2005.10.089Modeling K(m) values using electrotopological state: substrates for cytochrome P450 3A4-mediated metabolism.
Wang YH, Li Y, Li YH, Yang SL, Yang L.
Bioorg Med Chem Lett · research support, non-u.s. gov't; journal article · DOI 10.1016/j.bmcl.2005.06.015Early absorption and distribution analysis of antitumor and anti-AIDS drugs: lipid membrane and plasma protein interactions.
Cimitan S, Lindgren MT, Bertucci C, Danielson UH.
J Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1021/jm049343oCytotoxic arylnaphthalene lignans from a Vietnamese acanthaceae, Justicia patentiflora.
Susplugas S, Hung NV, Bignon J, Thoison O, Kruczynski A, Sévenet T, Guéritte F.
J Nat Prod · research support, non-u.s. gov't; journal article · DOI 10.1021/np050028uSynthesis and biological evaluation of novel taxoids designed for targeted delivery to tumors.
Baloglu E, Miller ML, Roller EE, Cavanagh EE, Leece BA, Goldmacher VS, Chari RV.
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Matthews EJ, Kruhlak NL, Weaver JL, Benz RD, Contrera JF.
Curr Drug Discov Technol · journal article · DOI 10.2174/1570163043334794Synthesis of C2-C3'N-linked macrocyclic taxoids. Novel docetaxel analogues with high tubulin activity.
Querolle O, Dubois J, Thoret S, Roussi F, Guéritte F, Guénard D.
J Med Chem · journal article · DOI 10.1021/jm0497996Synthesis of potent taxoids for tumor-specific delivery using monoclonal antibodies.
Miller ML, Roller EE, Wu X, Leece BA, Goldmacher VS, Chari RV, Ojima I.
Bioorg Med Chem Lett · research support, u.s. gov't, p.h.s.; journal article · DOI 10.1016/j.bmcl.2004.05.027[Drug-induced liver injury; fourteenth updated edition of the bibliographic database of liver injuries and related drugs].
Biour M, Ben Salem C, Chazouillères O, Grangé JD, Serfaty L, Poupon R.
Gastroenterol Clin Biol · bibliography; journal article · DOI 10.1016/s0399-8320(04)95062-2New highly active taxoids from 9beta-dihydrobaccatin-9,10-acetals. Part 3.
Takeda Y, Yoshino T, Uoto K, Chiba J, Ishiyama T, Iwahana M, Jimbo T, Tanaka N, Terasawa H, Soga T.
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