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Publikationer i urvalet

11 träffar

Bibliografisk träff 2024-06-24

Discovery of Dual MER/AXL Kinase Inhibitors as Bifunctional Small Molecules for Inhibiting Tumor Growth and Enhancing Tumor Immune Microenvironment.

Li MC, Lai YL, Kuo PH, Reddy JS, Chen CM, Manimala J, Wang PC, Wu MS, Chang CY, Yang CM, Lin CY, Huang YC, Chiu CH, Chang L, Lin WH, Yeh TK, Yen WC, Hsieh HP.

J Med Chem · research support, non-u.s. gov't; research-article; journal article · DOI 10.1021/acs.jmedchem.4c00400

Bibliografisk träff 2024-06-12

Discovery of new 1,3-diphenylurea appended aryl pyridine derivatives as apoptosis inducers through c-MET and VEGFR-2 inhibition: design, synthesis, <i>in vivo</i> and <i>in silico</i> studies.

Elsebaie HA, Nafie MS, Tawfik HO, Belal A, Ghoneim MM, Obaidullah AJ, Shaaban S, Ayed AA, El-Naggar M, Mehany ABM, Shaldam MA.

RSC Med Chem · research-article; journal article · DOI 10.1039/d4md00280f

Bibliografisk träff 2024-05-03

Recent discovery and development of AXL inhibitors as antitumor agents.

Liu Z, Chen L, Zhang J, Yang J, Xiao X, Shan L, Mao W.

Eur J Med Chem · review; journal article · DOI 10.1016/j.ejmech.2024.116475

Bibliografisk träff 2023-12-30

Structure-activity relationship study of 1,6-naphthyridinone derivatives as selective type II AXL inhibitors with potent antitumor efficacy.

Zhuo L, Guo M, Zhang S, Wu J, Wang M, Shen Y, Peng X, Wang Z, Jiang W, Huang W.

Eur J Med Chem · journal article · DOI 10.1016/j.ejmech.2023.116090

Bibliografisk träff 2023-08-11

Discovery of Novel, Thienopyridine-Based Tyrosine Kinase Inhibitors Targeting Tumorigenic RON Splice Variants.

Ryu H, Kim H, Park I, Lee M, Park YS, Jin DH, Hur SC, Park J, Lee H.

ACS Med Chem Lett · rapid-communication; journal article · DOI 10.1021/acsmedchemlett.3c00206

Bibliografisk träff 2023-06-01

Targeting MET: Discovery of Small Molecule Inhibitors as Non-Small Cell Lung Cancer Therapy.

Wang C, Lu X.

J Med Chem · research support, non-u.s. gov't; review; journal article · DOI 10.1021/acs.jmedchem.3c00028

Bibliografisk träff 2021-04-02

Progress in developing MNK inhibitors.

Jin X, Yu R, Wang X, Proud CG, Jiang T.

Eur J Med Chem · review; journal article · DOI 10.1016/j.ejmech.2021.113420

Bibliografisk träff 2020-01-07

Stepwise Evolution of Fragment Hits against MAPK Interacting Kinases 1 and 2.

Kwiatkowski J, Liu B, Pang S, Ahmad NHB, Wang G, Poulsen A, Yang H, Poh YR, Tee DHY, Ong E, Retna P, Dinie N, Kwek P, Wee JLK, Manoharan V, Low CB, Seah PG, Pendharkar V, Sangthongpitag K, Joy J, Baburajendran N, Jansson AE, Nacro K, Hill J, Keller TH, Hung AW.

J Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1021/acs.jmedchem.9b01582

Bibliografisk träff 2018-09-19

Insights into Current Tropomyosin Receptor Kinase (TRK) Inhibitors: Development and Clinical Application.

Yan W, Lakkaniga NR, Carlomagno F, Santoro M, McDonald NQ, Lv F, Gunaganti N, Frett B, Li HY.

J Med Chem · research-article; journal article; research support, n.i.h., extramural · DOI 10.1021/acs.jmedchem.8b01092

Bibliografisk träff 2017-12-01

The target landscape of clinical kinase drugs.

Klaeger S, Heinzlmeir S, Wilhelm M, Polzer H, Vick B, Koenig PA, Reinecke M, Ruprecht B, Petzoldt S, Meng C, Zecha J, Reiter K, Qiao H, Helm D, Koch H, Schoof M, Canevari G, Casale E, Depaolini SR, Feuchtinger A, Wu Z, Schmidt T, Rueckert L, Becker W, Huenges J, Garz AK, Gohlke BO, Zolg DP, Kayser G, Vooder T, Preissner R, Hahne H, Tõnisson N, Kramer K, Götze K, Bassermann F, Schlegl J, Ehrlich HC, Aiche S, Walch A, Greif PA, Schneider S, Felder ER, Ruland J, Médard G, Jeremias I, Spiekermann K, Kuster B.

Science · research support, non-u.s. gov't; research-article; journal article · DOI 10.1126/science.aan4368

Bibliografisk träff 2015-11-20

AXL Inhibitors in Cancer: A Medicinal Chemistry Perspective.

Myers SH, Brunton VG, Unciti-Broceta A.

J Med Chem · research support, non-u.s. gov't; review; journal article · DOI 10.1021/acs.jmedchem.5b01273