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Publikationer i urvalet

16 träffar

Bibliografisk träff 2020-12-03

Synthesis and Biological Characterization of Cyclic Disulfide-Containing Peptide Analogs of the Multifunctional Opioid/Neuropeptide FF Receptor Agonists That Produce Long-Lasting and Nontolerant Antinociception.

Zhang M, Xu B, Li N, Liu H, Shi X, Zhang Q, Shi Y, Xu K, Xiao J, Chen D, Zhu H, Sun Y, Zhang T, Zhang R, Fang Q.

J Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1021/acs.jmedchem.0c01367

Bibliografisk träff 2017-03-13

In silico design of novel probes for the atypical opioid receptor MRGPRX2.

Lansu K, Karpiak J, Liu J, Huang XP, McCorvy JD, Kroeze WK, Che T, Nagase H, Carroll FI, Jin J, Shoichet BK, Roth BL.

Nat Chem Biol · research-article; journal article · DOI 10.1038/nchembio.2334

Bibliografisk träff 2015-01-06

CNS drug design: balancing physicochemical properties for optimal brain exposure.

Rankovic Z.

J Med Chem · review; journal article · DOI 10.1021/jm501535r

Bibliografisk träff 2013-11-19

Comparison of the accuracy of experimental and predicted pKa values of basic and acidic compounds.

Settimo L, Bellman K, Knegtel RM.

Pharm Res · comparative study; journal article · DOI 10.1007/s11095-013-1232-z

Bibliografisk träff 2011-06-12

Synthesis and biological evaluation of analogues of M6G.

Trécant C, Dlubala A, George P, Pichat P, Ripoche I, Troin Y.

Eur J Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1016/j.ejmech.2011.05.076

Bibliografisk träff 2010-12-13

Measurement of unbound drug exposure in brain: modeling of pH partitioning explains diverging results between the brain slice and brain homogenate methods.

Fridén M, Bergström F, Wan H, Rehngren M, Ahlin G, Hammarlund-Udenaes M, Bredberg U.

Drug Metab Dispos · comparative study; journal article · DOI 10.1124/dmd.110.035998

Bibliografisk träff 2009-10-01

Structure-brain exposure relationships in rat and human using a novel data set of unbound drug concentrations in brain interstitial and cerebrospinal fluids.

Fridén M, Winiwarter S, Jerndal G, Bengtsson O, Wan H, Bredberg U, Hammarlund-Udenaes M, Antonsson M.

J Med Chem · journal article · DOI 10.1021/jm901036q

Bibliografisk träff 2009-05-01

Synthesis, conformation, and biological characterization of a sugar derivative of morphine that is a potent, long-lasting, and nontolerant antinociceptive.

Arsequell G, Salvatella M, Valencia G, Fernández-Mayoralas A, Fontanella M, Venturi C, Jiménez-Barbero J, Marrón E, Rodríguez RE.

J Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1021/jm8011245

Bibliografisk träff 2008-04-21

Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.

Obach RS, Lombardo F, Waters NJ.

Drug Metab Dispos · journal article · DOI 10.1124/dmd.108.020479

Bibliografisk träff 2005-03-01

Synthesis and in vitro biological evaluation of a carbon glycoside analogue of morphine-6-glucuronide.

MacDougall JM, Zhang XD, Polgar WE, Khroyan TV, Toll L, Cashman JR.

Bioorg Med Chem Lett · journal article · DOI 10.1016/j.bmcl.2005.01.072

Bibliografisk träff 2005-01-12

UDP-glucuronosyltransferases and clinical drug-drug interactions.

Kiang TK, Ensom MH, Chang TK.

Pharmacol Ther · research support, non-u.s. gov't; review; journal article · DOI 10.1016/j.pharmthera.2004.10.013

Bibliografisk träff 2004-11-01

Design, chemical synthesis, and biological evaluation of thiosaccharide analogues of morphine- and codeine-6-glucuronide.

MacDougall JM, Zhang XD, Polgar WE, Khroyan TV, Toll L, Cashman JR.

J Med Chem · journal article · DOI 10.1021/jm049554t

Bibliografisk träff 2003-03-01

Structure-activity relationships of some opiate glycosides.

Stachulski AV, Scheinmann F, Ferguson JR, Law JL, Lumbard KW, Hopkins P, Patel N, Clarke S, Gloyne A, Joel SP.

Bioorg Med Chem Lett · journal article · DOI 10.1016/s0960-894x(03)00056-8

Bibliografisk träff 2000-06-01

Predicting blood-brain barrier permeation from three-dimensional molecular structure.

Crivori P, Cruciani G, Carrupt PA, Testa B.

J Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1021/jm990968+

Bibliografisk träff 1996-10-01

Octanol-, chloroform-, and propylene glycol dipelargonat-water partitioning of morphine-6-glucuronide and other related opiates.

Avdeef A, Barrett DA, Shaw PN, Knaggs RD, Davis SS.

J Med Chem · journal article · DOI 10.1021/jm960073m

Bibliografisk träff 1991-04-01

Morphine 6-glucuronide and morphine 3-glucuronide as molecular chameleons with unexpected lipophilicity.

Carrupt PA, Testa B, Bechalany A, el Tayar N, Descas P, Perrissoud D.

J Med Chem · comparative study; research support, non-u.s. gov't; journal article · DOI 10.1021/jm00108a005