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Publikationer i urvalet

29 träffar

Bibliografisk träff 2021-10-04

Flavonoid Monomers as Potent, Nontoxic, and Selective Modulators of the Breast Cancer Resistance Protein (ABCG2).

Wong ILK, Zhu X, Chan KF, Liu Z, Chan CF, Chow TS, Chong TC, Law MC, Cui J, Chow LMC, Chan TH.

J Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1021/acs.jmedchem.1c00779

Bibliografisk träff 2014-09-12

Polyoxypregnane steroids from the stems of Marsdenia tenacissima.

Yao S, To KK, Wang YZ, Yin C, Tang C, Chai S, Ke CQ, Lin G, Ye Y.

J Nat Prod · research support, non-u.s. gov't; journal article · DOI 10.1021/np500385b

Bibliografisk träff 2012-05-15

Classification of inhibitors of hepatic organic anion transporting polypeptides (OATPs): influence of protein expression on drug-drug interactions.

Karlgren M, Vildhede A, Norinder U, Wisniewski JR, Kimoto E, Lai Y, Haglund U, Artursson P.

J Med Chem · research support, non-u.s. gov't; research-article; journal article · DOI 10.1021/jm300212s

Bibliografisk träff 2012-03-27

Structure-activity relationships, ligand efficiency, and lipophilic efficiency profiles of benzophenone-type inhibitors of the multidrug transporter P-glycoprotein.

Jabeen I, Pleban K, Rinner U, Chiba P, Ecker GF.

J Med Chem · research support, non-u.s. gov't; research-article; journal article · DOI 10.1021/jm201705f

Bibliografisk träff 2012-02-22

Amine linked flavonoid dimers as modulators for P-glycoprotein-based multidrug resistance: structure-activity relationship and mechanism of modulation.

Chan KF, Wong IL, Kan JW, Yan CS, Chow LM, Chan TH.

J Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1021/jm201121b

Bibliografisk träff 2012-01-19

Cerebrospinal fluid can be used as a surrogate to assess brain exposures of breast cancer resistance protein and P-glycoprotein substrates.

Xiao G, Black C, Hetu G, Sands E, Wang J, Caputo R, Rohde E, Gan LS.

Drug Metab Dispos · journal article · DOI 10.1124/dmd.111.043703

Bibliografisk träff 2010-07-01

Design and syntheses of permethyl ningalin B analogues: potent multidrug resistance (MDR) reversal agents of cancer cells.

Zhang PY, Wong IL, Yan CS, Zhang XY, Jiang T, Chow LM, Wan SB.

J Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1021/jm100035c

Bibliografisk träff 2010-01-01

Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.

Fourches D, Barnes JC, Day NC, Bradley P, Reed JZ, Tropsha A.

Chem Res Toxicol · research-article; research support, u.s. gov't, non-p.h.s.; journal article; research support, n.i.h., extramural · DOI 10.1021/tx900326k

Bibliografisk träff 2008-04-21

Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.

Obach RS, Lombardo F, Waters NJ.

Drug Metab Dispos · journal article · DOI 10.1124/dmd.108.020479

Bibliografisk träff 2006-10-10

Differences in the transport of the antiepileptic drugs phenytoin, levetiracetam and carbamazepine by human and mouse P-glycoprotein.

Baltes S, Gastens AM, Fedrowitz M, Potschka H, Kaever V, Löscher W.

Neuropharmacology · research support, non-u.s. gov't; journal article · DOI 10.1016/j.neuropharm.2006.07.038

Bibliografisk träff 2004-03-01

Distinct groups of multidrug resistance modulating agents are distinguished by competition of P-glycoprotein-specific antibodies.

Nagy H, Goda K, Fenyvesi F, Bacsó Z, Szilasi M, Kappelmayer J, Lustyik G, Cianfriglia M, Szabó G.

Biochem Biophys Res Commun · research support, non-u.s. gov't; journal article · DOI 10.1016/j.bbrc.2004.01.156

Bibliografisk träff 2004-01-27

Broad-spectrum modulation of ATP-binding cassette transport proteins by the taxane derivatives ortataxel (IDN-5109, BAY 59-8862) and tRA96023.

Minderman H, Brooks TA, O'Loughlin KL, Ojima I, Bernacki RJ, Baer MR.

Cancer Chemother Pharmacol · research support, u.s. gov't, p.h.s.; research support, non-u.s. gov't; journal article · DOI 10.1007/s00280-003-0745-2

Bibliografisk träff 2002-06-01

Analysis of methotrexate and folate transport by multidrug resistance protein 4 (ABCC4): MRP4 is a component of the methotrexate efflux system.

Chen ZS, Lee K, Walther S, Raftogianis RB, Kuwano M, Zeng H, Kruh GD.

Cancer Res · research support, u.s. gov't, p.h.s.; research support, non-u.s. gov't; journal article

Bibliografisk träff 2001-10-01

Transport of methotrexate (MTX) and folates by multidrug resistance protein (MRP) 3 and MRP1: effect of polyglutamylation on MTX transport.

Zeng H, Chen ZS, Belinsky MG, Rea PA, Kruh GD.

Cancer Res · research support, u.s. gov't, p.h.s.; research support, non-u.s. gov't; research support, u.s. gov't, non-p.h.s.; journal article

Bibliografisk träff 2000-10-01

Selective inhibition of human cytochrome P450 3A4 by N-[2(R)-hydroxy-1(S)-indanyl]-5-[2(S)-(1, 1-dimethylethylaminocarbonyl)-4-[(furo[2, 3-b]pyridin-5-yl)methyl]piperazin-1-yl]-4(S)-hydroxy-2(R)-phenylmethy lpentanamide and P-glycoprotein by valspodar in gene transfectant systems.

Kawahara I, Kato Y, Suzuki H, Achira M, Ito K, Crespi CL, Sugiyama Y.

Drug Metab Dispos · research support, non-u.s. gov't; journal article

Bibliografisk träff 2000-10-01

Role of breast cancer resistance protein in the bioavailability and fetal penetration of topotecan.

Jonker JW, Smit JW, Brinkhuis RF, Maliepaard M, Beijnen JH, Schellens JH, Schinkel AH.

J Natl Cancer Inst · research support, non-u.s. gov't; journal article · DOI 10.1093/jnci/92.20.1651

Bibliografisk träff 2000-06-01

Pharmacological inhibition of P-glycoprotein transport enhances the distribution of HIV-1 protease inhibitors into brain and testes.

Choo EF, Leake B, Wandel C, Imamura H, Wood AJ, Wilkinson GR, Kim RB.

Drug Metab Dispos · research support, u.s. gov't, p.h.s.; research support, non-u.s. gov't; journal article · DOI 10.1016/s0090-9556(24)15144-6

Bibliografisk träff 1999-12-01

Effect of multidrug resistance-reversing agents on transporting activity of human canalicular multispecific organic anion transporter.

Chen ZS, Kawabe T, Ono M, Aoki S, Sumizawa T, Furukawa T, Uchiumi T, Wada M, Kuwano M, Akiyama SI.

Mol Pharmacol · research support, non-u.s. gov't; journal article · DOI 10.1124/mol.56.6.1219

Bibliografisk träff 1999-08-01

OATP and P-glycoprotein transporters mediate the cellular uptake and excretion of fexofenadine.

Cvetkovic M, Leake B, Fromm MF, Wilkinson GR, Kim RB.

Drug Metab Dispos · research support, u.s. gov't, p.h.s.; research support, non-u.s. gov't; journal article · DOI 10.1016/s0090-9556(24)15235-x

Bibliografisk träff 1999-04-01

PSC833, cyclosporin A, and dexniguldipine effects on cellular calcein retention and inhibition of the multidrug resistance pump in human leukemic lymphoblasts.

Wigler PW.

Biochem Biophys Res Commun · journal article · DOI 10.1006/bbrc.1999.0475

Bibliografisk träff 1998-11-01

Expression of the apical conjugate export pump, Mrp2, in the polarized hepatoma cell line, WIF-B.

Nies AT, Cantz T, Brom M, Leier I, Keppler D.

Hepatology · research support, non-u.s. gov't; journal article · DOI 10.1002/hep.510280523

Bibliografisk träff 1998-11-01

Inhibitory effects of a cyclosporin derivative, SDZ PSC 833, on transport of doxorubicin and vinblastine via human P-glycoprotein.

Kusunoki N, Takara K, Tanigawara Y, Yamauchi A, Ueda K, Komada F, Ku Y, Kuroda Y, Saitoh Y, Okumura K.

Jpn J Cancer Res · research support, non-u.s. gov't; research-article; journal article · DOI 10.1111/j.1349-7006.1998.tb00518.x

Bibliografisk träff 1998-05-01

Effect of the Mdr1a P-glycoprotein gene disruption on the tissue distribution of SDZ PSC 833, a multidrug resistance-reversing agent, in mice.

Desrayaud S, De Lange EC, Lemaire M, Bruelisauer A, De Boer AG, Breimer DD.

J Pharmacol Exp Ther · journal article · DOI 10.1016/s0022-3565(24)37447-6

Bibliografisk träff 1998-01-01

The drug transporter P-glycoprotein limits oral absorption and brain entry of HIV-1 protease inhibitors.

Kim RB, Fromm MF, Wandel C, Leake B, Wood AJ, Roden DM, Wilkinson GR.

J Clin Invest · research support, u.s. gov't, p.h.s.; research support, non-u.s. gov't; research-article; journal article · DOI 10.1172/jci1269

Bibliografisk träff 1997-11-01

P-Glycoprotein mediates the efflux of quinidine across the blood-brain barrier.

Kusuhara H, Suzuki H, Terasaki T, Kakee A, Lemaire M, Sugiyama Y.

J Pharmacol Exp Ther · journal article · DOI 10.1016/s0022-3565(24)37075-2

Bibliografisk träff 1997-09-01

Interaction of cyclosporin derivatives with the ATPase activity of human P-glycoprotein.

Watanabe T, Kokubu N, Charnick SB, Naito M, Tsuruo T, Cohen D.

Br J Pharmacol · comparative study; research-article; journal article · DOI 10.1038/sj.bjp.0701377

Bibliografisk träff 1997-01-01

Reversal of P-glycoprotein-associated multidrug resistance by ivermectin.

Pouliot JF, L'Heureux F, Liu Z, Prichard RK, Georges E.

Biochem Pharmacol · research support, non-u.s. gov't; journal article · DOI 10.1016/s0006-2952(96)00656-9

Bibliografisk träff 1996-07-01

Ranking of P-glycoprotein substrates and inhibitors by a calcein-AM fluorometry screening assay.

Tiberghien F, Loor F.

Anticancer Drugs · comparative study; research support, non-u.s. gov't; journal article · DOI 10.1097/00001813-199607000-00012

Bibliografisk träff 1994-11-01

The MRP gene encodes an ATP-dependent export pump for leukotriene C4 and structurally related conjugates.

Leier I, Jedlitschky G, Buchholz U, Cole SP, Deeley RG, Keppler D.

J Biol Chem · comparative study; research support, non-u.s. gov't; journal article · DOI 10.1016/s0021-9258(18)46856-1