PUBLICATION REGISTRY

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Publikationer som ChEBI hänvisar till för molibresib. Visa hela publikationsregistret

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Publications in the selection

35 hits

Bibliografisk träff 2013-12-13

Potent antimyeloma activity of the novel bromodomain inhibitors I-BET151 and I-BET762.

Chaidos A, Caputo V, Gouvedenou K, Liu B, Marigo I, Chaudhry MS, Rotolo A, Tough DF, Smithers NN, Bassil AK, Chapman TD, Harker NR, Barbash O, Tummino P, Al-Mahdi N, Haynes AC, Cutler L, Le B, Rahemtulla A, Roberts I, Kleijnen M, Witherington JJ, Parr NJ, Prinjha RK, Karadimitris A.

Blood · research support, non-u.s. gov't; journal article · DOI 10.1182/blood-2013-01-478420

Bibliografisk träff 2013-09-25

Discovery of epigenetic regulator I-BET762: lead optimization to afford a clinical candidate inhibitor of the BET bromodomains.

Mirguet O, Gosmini R, Toum J, Clément CA, Barnathan M, Brusq JM, Mordaunt JE, Grimes RM, Crowe M, Pineau O, Ajakane M, Daugan A, Jeffrey P, Cutler L, Haynes AC, Smithers NN, Chung CW, Bamborough P, Uings IJ, Lewis A, Witherington J, Parr N, Prinjha RK, Nicodème E.

J Med Chem · journal article · DOI 10.1021/jm401088k

Bibliografisk träff 2013-09-25

The making of I-BET762, a BET bromodomain inhibitor now in clinical development.

Zhao Y, Yang CY, Wang S.

J Med Chem · comment; journal article · DOI 10.1021/jm4014407

Bibliografisk träff 2011-05-13

Discovery and characterization of small molecule inhibitors of the BET family bromodomains.

Chung CW, Coste H, White JH, Mirguet O, Wilde J, Gosmini RL, Delves C, Magny SM, Woodward R, Hughes SA, Boursier EV, Flynn H, Bouillot AM, Bamborough P, Brusq JM, Gellibert FJ, Jones EJ, Riou AM, Homes P, Martin SL, Uings IJ, Toum J, Clement CA, Boullay AB, Grimley RL, Blandel FM, Prinjha RK, Lee K, Kirilovsky J, Nicodeme E.

J Med Chem · journal article · DOI 10.1021/jm200108t

Bibliografisk träff 2010-11-10

Suppression of inflammation by a synthetic histone mimic.

Nicodeme E, Jeffrey KL, Schaefer U, Beinke S, Dewell S, Chung CW, Chandwani R, Marazzi I, Wilson P, Coste H, White J, Kirilovsky J, Rice CM, Lora JM, Prinjha RK, Lee K, Tarakhovsky A.

Nature · research support, non-u.s. gov't; research-article; journal article; research support, n.i.h., extramural · DOI 10.1038/nature09589