The current strategies of optimization of oseltamivir against mutant neuraminidases of influenza A：A review.
Wang K, Zhang H, Tian Y.
Eur J Med Chem · review; journal article · DOI 10.1016/j.ejmech.2022.114711 PUBLICATION REGISTRY
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Publikationer som ChEBI hänvisar till för laninamivir octanoate hydrate. Visa hela publikationsregistret
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7 hitsInfluenza-existing drugs and treatment prospects.
Sarker A, Gu Z, Mao L, Ge Y, Hou D, Fang J, Wei Z, Wang Z.
Eur J Med Chem · review; journal article · DOI 10.1016/j.ejmech.2022.114189Pharmacokinetic mechanism involved in the prolonged high retention of laninamivir in mouse respiratory tissues after intranasal administration of its prodrug laninamivir octanoate.
Koyama K, Nakai D, Takahashi M, Nakai N, Kobayashi N, Imai T, Izumi T.
Drug Metab Dispos · journal article · DOI 10.1124/dmd.112.048280Laninamivir prodrug CS-8958, a long-acting neuraminidase inhibitor, shows superior anti-influenza virus activity after a single administration.
Kubo S, Tomozawa T, Kakuta M, Tokumitsu A, Yamashita M.
Antimicrob Agents Chemother · research support, non-u.s. gov't; research-article; journal article · DOI 10.1128/aac.01311-09CS-8958, a prodrug of the novel neuraminidase inhibitor R-125489, demonstrates a favorable long-retention profile in the mouse respiratory tract.
Koyama K, Takahashi M, Oitate M, Nakai N, Takakusa H, Miura S, Okazaki O.
Antimicrob Agents Chemother · research-article; journal article · DOI 10.1128/aac.00731-09Synthesis and in vivo influenza virus-inhibitory effect of ester prodrug of 4-guanidino-7-O-methyl-Neu5Ac2en.
Honda T, Kubo S, Masuda T, Arai M, Kobayashi Y, Yamashita M.
Bioorg Med Chem Lett · journal article · DOI 10.1016/j.bmcl.2009.04.067CS-8958, a prodrug of the new neuraminidase inhibitor R-125489, shows long-acting anti-influenza virus activity.
Yamashita M, Tomozawa T, Kakuta M, Tokumitsu A, Nasu H, Kubo S.
Antimicrob Agents Chemother · research support, non-u.s. gov't; research-article; journal article · DOI 10.1128/aac.00333-08