Structure-based identification of OATP1B1/3 inhibitors.
De Bruyn T, van Westen GJ, Ijzerman AP, Stieger B, de Witte P, Augustijns PF, Annaert PP.
Mol Pharmacol · research support, non-u.s. gov't; journal article · DOI 10.1124/mol.112.084152 PUBLICATION REGISTRY
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14 hitsAntiviral activity of 2,3'-anhydro and related pyrimidine nucleosides against hepatitis B virus.
Srivastav NC, Mak M, Agrawal B, Tyrrell DL, Kumar R.
Bioorg Med Chem Lett · research support, non-u.s. gov't; journal article · DOI 10.1016/j.bmcl.2010.08.120Deoxyribonucleoside kinases activate nucleoside antibiotics in severely pathogenic bacteria.
Sandrini MP, Shannon O, Clausen AR, Björck L, Piskur J.
Antimicrob Agents Chemother · research support, non-u.s. gov't; research-article; journal article · DOI 10.1128/aac.00081-07Sensitivity of monkey B virus (Cercopithecine herpesvirus 1) to antiviral drugs: role of thymidine kinase in antiviral activities of substrate analogs and acyclonucleosides.
Focher F, Lossani A, Verri A, Spadari S, Maioli A, Gambino JJ, Wright GE, Eberle R, Black DH, Medveczky P, Medveczky M, Shugar D.
Antimicrob Agents Chemother · research support, non-u.s. gov't; research-article; journal article; research support, n.i.h., extramural · DOI 10.1128/aac.01284-06Probing the anticancer activity of nucleoside analogues: a QSAR model approach using an internally consistent training set.
Helguera AM, Rodríguez-Borges JE, García-Mera X, Fernández F, Cordeiro MN.
J Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1021/jm061445mThymidine and thymidine-5'-O-monophosphate analogues as inhibitors of Mycobacterium tuberculosis thymidylate kinase.
Vanheusden V, Van Rompaey P, Munier-Lehmann H, Pochet S, Herdewijn P, Van Calenbergh S.
Bioorg Med Chem Lett · research support, non-u.s. gov't; journal article · DOI 10.1016/s0960-894x(03)00643-7Synthesis and antiviral activity of novel 5-(1-cyanamido-2-haloethyl) and 5-(1-hydroxy(or methoxy)-2-azidoethyl) analogues of uracil nucleosides.
Kumar R, Rai D, Sharma SK, Sharma SK, Saffran HA, Blush R, Tyrrell DL.
J Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1021/jm010226sSynthesis of new acyclic pyrimidine nucleoside analogs as potential antiviral drugs.
Eger K, Klünder EM, Schmidt M.
J Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1021/jm00045a010Synthesis and antiviral activity of novel 5-(1-azido-2-haloethyl) and 5-(1-azido-, amino-, or methoxyethyl) analogs of 2'-deoxyuridine.
Kumar R, Wiebe LI, Knaus EE.
J Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1021/jm00069a004Synthesis and antiviral activity of phosphonoacetic and phosphonoformic acid esters of 5-bromo-2'-deoxyuridine and related pyrimidine nucleosides and acyclonucleosides.
Lambert RW, Martin JA, Thomas GJ, Duncan IB, Hall MJ, Heimer EP.
J Med Chem · journal article · DOI 10.1021/jm00122a014Synthesis and biological activities of 4-O-(difluoromethyl)-5-substituted-uracil nucleoside analogues.
Reefschläger J, Pein CD, Cech D.
J Med Chem · journal article · DOI 10.1021/jm00397a022Synthesis and antitumor and antiviral properties of 5-alkyl-2'-deoxyuridines, 3',5'-cyclic monophosphates, and neutral cyclic triesters.
Bères J, Bentrude WG, Balzarini J, De Clercq E, Otvös L.
J Med Chem · research support, u.s. gov't, p.h.s.; research support, non-u.s. gov't; journal article · DOI 10.1021/jm00154a012Synthesis and antiviral activity of the carbocyclic analogues of 5-ethyl-2'-deoxyuridine and of 5-ethynyl-2'-deoxyuridine.
Shealy YF, O'Dell CA, Arnett G, Shannon WM.
J Med Chem · comparative study; research support, u.s. gov't, p.h.s.; journal article · DOI 10.1021/jm00151a013Thymidine phosphorylase. Substrate specificity for 5-substituted 2'-deoxyuridines.
Nakayama C, Wataya Y, Meyer RB, Santi DV, Saneyoshi M, Ueda T.
J Med Chem · research support, u.s. gov't, p.h.s.; journal article · DOI 10.1021/jm00182a029