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Publikationer som ChEBI hänvisar till för GSK1016790A. Visa hela publikationsregistret

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Publications in the selection

14 hits

Bibliografisk träff 2018-03-22

TRPV4 is functionally expressed in oligodendrocyte precursor cells and increases their proliferation.

Ohashi K, Deyashiki A, Miyake T, Nagayasu K, Shibasaki K, Shirakawa H, Kaneko S.

Pflugers Arch · research support, non-u.s. gov't; journal article · DOI 10.1007/s00424-018-2130-3

Bibliografisk träff 2018-02-07

Transient Receptor Potential Vanilloid 4 Activation-Induced Increase in Glycine-Activated Current in Mouse Hippocampal Pyramidal Neurons.

Qi M, Wu C, Wang Z, Zhou L, Men C, Du Y, Huang S, Chen L, Chen L.

Cell Physiol Biochem · journal article · DOI 10.1159/000487350

Bibliografisk träff 2018-01-02

Pharmacological activation of TRPV4 produces immediate cell damage and induction of apoptosis in human melanoma cells and HaCaT keratinocytes.

Olivan-Viguera A, Garcia-Otin AL, Lozano-Gerona J, Abarca-Lachen E, Garcia-Malinis AJ, Hamilton KL, Gilaberte Y, Pueyo E, Köhler R.

PLoS One · research support, non-u.s. gov't; research-article; journal article · DOI 10.1371/journal.pone.0190307

Bibliografisk träff 2017-10-01

PROPERTIES OF THE TRPV4 AGONIST GSK1016790A AND the TRPV4 ANTAGONIST GSK2193874.

Thorneloe KS, Cheung M, Holt DA, Willette RN.

Physiol Rev · letter; comment · DOI 10.1152/physrev.00019.2017

Bibliografisk träff 2017-06-15

Activation of Transient Receptor Potential Vanilloid 4 Impairs the Dendritic Arborization of Newborn Neurons in the Hippocampal Dentate Gyrus through the AMPK and Akt Signaling Pathways.

Tian Y, Qi M, Wang Z, Wu C, Sun Z, Li Y, Sha S, Du Y, Chen L, Chen L.

Front Mol Neurosci · research-article; journal article · DOI 10.3389/fnmol.2017.00190

Bibliografisk träff 2017-03-27

TRPV4 regulates insulin mRNA expression and INS-1E cell death via ERK1/2 and NO-dependent mechanisms.

Billert M, Skrzypski M, Sassek M, Szczepankiewicz D, Wojciechowicz T, Mergler S, Strowski MZ, Nowak KW.

Cell Signal · research support, non-u.s. gov't; journal article · DOI 10.1016/j.cellsig.2017.03.018

Bibliografisk träff 2016-10-17

Enhanced Oxidative Stress Is Responsible for TRPV4-Induced Neurotoxicity.

Hong Z, Tian Y, Yuan Y, Qi M, Li Y, Du Y, Chen L, Chen L.

Front Cell Neurosci · research-article; journal article · DOI 10.3389/fncel.2016.00232

Bibliografisk träff 2016-08-26

Transient Receptor Potential Vanilloid 4 Inhibits γ-Aminobutyric Acid-Activated Current in Hippocampal Pyramidal Neurons.

Hong Z, Tian Y, Qi M, Li Y, Du Y, Chen L, Liu W, Chen L.

Front Mol Neurosci · research-article; journal article · DOI 10.3389/fnmol.2016.00077

Bibliografisk träff 2016-01-19

NO synthase inhibition attenuates EDHF-mediated relaxation induced by TRPV4 channel agonist GSK1016790A in the rat pulmonary artery: Role of TxA2.

Addison MP, Singh TU, Parida S, Choudhury S, Kasa JK, Sukumaran SV, Darzi SA, Kandasamy K, Singh V, Kumar D, Mishra SK.

Pharmacol Rep · journal article · DOI 10.1016/j.pharep.2016.01.003

Bibliografisk träff 2014-08-22

Role of MMP2 and MMP9 in TRPV4-induced lung injury.

Villalta PC, Rocic P, Townsley MI.

Am J Physiol Lung Cell Mol Physiol · research-article; journal article; research support, n.i.h., extramural · DOI 10.1152/ajplung.00113.2014

Bibliografisk träff 2013-11-01

Analysis of responses to the TRPV4 agonist GSK1016790A in the pulmonary vascular bed of the intact-chest rat.

Pankey EA, Zsombok A, Lasker GF, Kadowitz PJ.

Am J Physiol Heart Circ Physiol · research-article; journal article · DOI 10.1152/ajpheart.00303.2013

Bibliografisk träff 2012-06-11

Optical recording reveals novel properties of GSK1016790A-induced vanilloid transient receptor potential channel TRPV4 activity in primary human endothelial cells.

Sullivan MN, Francis M, Pitts NL, Taylor MS, Earley S.

Mol Pharmacol · research-article; journal article; research support, n.i.h., extramural · DOI 10.1124/mol.112.078584

Bibliografisk träff 2011-02-14

Determinants of TRPV4 activity following selective activation by small molecule agonist GSK1016790A.

Jin M, Wu Z, Chen L, Jaimes J, Collins D, Walters ET, O'Neil RG.

PLoS One · research-article; journal article; research support, n.i.h., extramural · DOI 10.1371/journal.pone.0016713

Bibliografisk träff 2008-05-22

N-((1S)-1-{[4-((2S)-2-{[(2,4-dichlorophenyl)sulfonyl]amino}-3-hydroxypropanoyl)-1-piperazinyl]carbonyl}-3-methylbutyl)-1-benzothiophene-2-carboxamide (GSK1016790A), a novel and potent transient receptor potential vanilloid 4 channel agonist induces urinary bladder contraction and hyperactivity: Part I.

Thorneloe KS, Sulpizio AC, Lin Z, Figueroa DJ, Clouse AK, McCafferty GP, Chendrimada TP, Lashinger ES, Gordon E, Evans L, Misajet BA, Demarini DJ, Nation JH, Casillas LN, Marquis RW, Votta BJ, Sheardown SA, Xu X, Brooks DP, Laping NJ, Westfall TD.

J Pharmacol Exp Ther · research support, non-u.s. gov't; journal article · DOI 10.1124/jpet.108.139295