DMSO-Perturbing Assay for Identifying Promiscuous Enzyme Inhibitors.
Tomohara K, Adachi I, Horino Y, Kesamaru H, Abe H, Suyama K, Nose T.
ACS Med Chem Lett · rapid-communication; journal article · DOI 10.1021/acsmedchemlett.9b00093 PUBLICATION REGISTRY
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10 hitsHSP60/10 chaperonin systems are inhibited by a variety of approved drugs, natural products, and known bioactive molecules.
Stevens M, Abdeen S, Salim N, Ray AM, Washburn A, Chitre S, Sivinski J, Park Y, Hoang QQ, Chapman E, Johnson SM.
Bioorg Med Chem Lett · research support, non-u.s. gov't; research-article; journal article; research support, n.i.h., extramural · DOI 10.1016/j.bmcl.2019.02.028From carbohydrates to drug-like fragments: Rational development of novel α-amylase inhibitors.
Al-Asri J, Fazekas E, Lehoczki G, Perdih A, Görick C, Melzig MF, Gyémánt G, Wolber G, Mortier J.
Bioorg Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1016/j.bmc.2015.09.007Radical-regulating and antiviral properties of ascorbic acid and its derivatives.
Brinkevich SD, Boreko EI, Savinova OV, Pavlova NI, Shadyro OI.
Bioorg Med Chem Lett · research support, non-u.s. gov't; journal article · DOI 10.1016/j.bmcl.2012.02.022Design of benzimidazole- and benzoxazole-2-thione derivatives as inhibitors of bacterial hyaluronan lyase.
Braun S, Botzki A, Salmen S, Textor C, Bernhardt G, Dove S, Buschauer A.
Eur J Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1016/j.ejmech.2011.07.014Lipid-like sulfoxides and amine oxides as inhibitors of mast cell activation.
Batista J, Schlechtingen G, Friedrichson T, Braxmeier T, Bajorath J.
Eur J Med Chem · journal article · DOI 10.1016/j.ejmech.2011.02.068Novel 6-O-acylated vitamin C derivatives as hyaluronidase inhibitors with selectivity for bacterial lyases.
Spickenreither M, Braun S, Bernhardt G, Dove S, Buschauer A.
Bioorg Med Chem Lett · research support, non-u.s. gov't; journal article · DOI 10.1016/j.bmcl.2006.07.087Synthesis and characterization of a series of novel monoacylated ascorbic acid derivatives, 6-O-acyl-2-O-alpha-D-glucopyranosyl-L-ascorbic acids, as skin antioxidants.
Yamamoto I, Tai A, Fujinami Y, Sasaki K, Okazaki S.
J Med Chem · journal article · DOI 10.1021/jm010379fKinetic characterisation of ene-diol-based inhibitors of alpha-amylase.
Gerrard JA, Prince MJ, Abell AD.
Bioorg Med Chem Lett · research support, non-u.s. gov't; journal article · DOI 10.1016/s0960-894x(00)00288-2Ascorbic acid-based inhibitors of alpha-amylases.
Abell AD, Ratcliffe MJ, Gerrard J.
Bioorg Med Chem Lett · research support, non-u.s. gov't; journal article · DOI 10.1016/s0960-894x(98)00298-4