PUBLICATION REGISTRY

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Publikationsdata från Europe PMC och PubMed. Följ källhänvisningar från ämnesregistret till originalpublikationerna.

Publikationer som ChEBI hänvisar till för molnupiravir. Visa hela publikationsregistret

A publication hit is not a conclusion. Publikationslistan visar bibliografiska uppgifter. Eventuella forskningsutdrag visas separat med originalunderlag. En källhänvisning visar inte i sig effekt, dosering eller säkerhet.

Publications in the selection

27 hits
Bibliografisk träff 2021-09-24

The combined treatment of Molnupiravir and Favipiravir results in a potentiation of antiviral efficacy in a SARS-CoV-2 hamster infection model.

Abdelnabi R, Foo CS, Kaptein SJF, Zhang X, Do TND, Langendries L, Vangeel L, Breuer J, Pang J, Williams R, Vergote V, Heylen E, Leyssen P, Dallmeier K, Coelmont L, Chatterjee AK, Mols R, Augustijns P, De Jonghe S, Jochmans D, Weynand B, Neyts J.

EBioMedicine · research-article; journal article · DOI 10.1016/j.ebiom.2021.103595
Bibliografisk träff 2021-08-11

Mechanism of molnupiravir-induced SARS-CoV-2 mutagenesis.

Kabinger F, Stiller C, Schmitzová J, Dienemann C, Kokic G, Hillen HS, Höbartner C, Cramer P.

Nat Struct Mol Biol · research support, non-u.s. gov't; research-article; journal article · DOI 10.1038/s41594-021-00651-0
Bibliografisk träff 2021-05-11

Molnupiravir promotes SARS-CoV-2 mutagenesis via the RNA template.

Gordon CJ, Tchesnokov EP, Schinazi RF, Götte M.

J Biol Chem · research support, non-u.s. gov't; research-article; research support, u.s. gov't, non-p.h.s.; journal article; research support, n.i.h., extramural · DOI 10.1016/j.jbc.2021.100770
Bibliografisk träff 2021-04-16

Orally delivered MK-4482 inhibits SARS-CoV-2 replication in the Syrian hamster model.

Rosenke K, Hansen F, Schwarz B, Feldmann F, Haddock E, Rosenke R, Barbian K, Meade-White K, Okumura A, Leventhal S, Hawman DW, Ricotta E, Bosio CM, Martens C, Saturday G, Feldmann H, Jarvis MA.

Nat Commun · research support, n.i.h., intramural; research support, non-u.s. gov't; research-article; journal article · DOI 10.1038/s41467-021-22580-8
Bibliografisk träff 2021-02-09

SARS-CoV-2 infection is effectively treated and prevented by EIDD-2801.

Wahl A, Gralinski LE, Johnson CE, Yao W, Kovarova M, Dinnon KH, Liu H, Madden VJ, Krzystek HM, De C, White KK, Gully K, Schäfer A, Zaman T, Leist SR, Grant PO, Bluemling GR, Kolykhalov AA, Natchus MG, Askin FB, Painter G, Browne EP, Jones CD, Pickles RJ, Baric RS, Garcia JV.

Nature · research support, non-u.s. gov't; research-article; journal article; research support, n.i.h., extramural · DOI 10.1038/s41586-021-03312-w
Bibliografisk träff 2020-10-08

A concise route to MK-4482 (EIDD-2801) from cytidine.

Vasudevan N, Ahlqvist GP, McGeough CP, Paymode DJ, Cardoso FSP, Lucas T, Dietz JP, Opatz T, Jamison TF, Gupton FB, Snead DR.

Chem Commun (Camb) · journal article · DOI 10.1039/d0cc05944g
Bibliografisk träff 2020-04-06

An orally bioavailable broad-spectrum antiviral inhibits SARS-CoV-2 in human airway epithelial cell cultures and multiple coronaviruses in mice.

Sheahan TP, Sims AC, Zhou S, Graham RL, Pruijssers AJ, Agostini ML, Leist SR, Schäfer A, Dinnon KH, Stevens LJ, Chappell JD, Lu X, Hughes TM, George AS, Hill CS, Montgomery SA, Brown AJ, Bluemling GR, Natchus MG, Saindane M, Kolykhalov AA, Painter G, Harcourt J, Tamin A, Thornburg NJ, Swanstrom R, Denison MR, Baric RS.

Sci Transl Med · research support, non-u.s. gov't; research-article; journal article; research support, n.i.h., extramural · DOI 10.1126/scitranslmed.abb5883
Bibliografisk träff 2019-10-01

Characterization of orally efficacious influenza drug with high resistance barrier in ferrets and human airway epithelia.

Toots M, Yoon JJ, Cox RM, Hart M, Sticher ZM, Makhsous N, Plesker R, Barrena AH, Reddy PG, Mitchell DG, Shean RC, Bluemling GR, Kolykhalov AA, Greninger AL, Natchus MG, Painter GR, Plemper RK.

Sci Transl Med · research support, non-u.s. gov't; research-article; research support, u.s. gov't, non-p.h.s.; journal article; research support, n.i.h., extramural · DOI 10.1126/scitranslmed.aax5866