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Publikationer som ChEBI hänvisar till för gatifloxacin. Visa hela publikationsregistret

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Publications in the selection

31 hits

Bibliografisk träff 2016-03-21

Crystal Structure of the Fab Fragment of an Anti-ofloxacin Antibody and Exploration of Its Specific Binding.

He K, Du X, Sheng W, Zhou X, Wang J, Wang S.

J Agric Food Chem · research support, non-u.s. gov't; journal article · DOI 10.1021/acs.jafc.5b05882

Bibliografisk träff 2007-11-22

Synthesis and antimycobacterial evaluation of newer 1-cyclopropyl-1,4-dihydro-6-fluoro-7-(substituted secondary amino)-8-methoxy-5-(sub)-4-oxoquinoline-3-carboxylic acids.

Senthilkumar P, Dinakaran M, Banerjee D, Devakaram RV, Yogeeswari P, China A, Nagaraja V, Sriram D.

Bioorg Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1016/j.bmc.2007.11.050

Bibliografisk träff 2007-11-09

Antimycobacterial activities of novel 2-(sub)-3-fluoro/nitro-5,12-dihydro-5-oxobenzothiazolo[3,2-a]quinoline-6-carboxylic acid.

Dinakaran M, Senthilkumar P, Yogeeswari P, China A, Nagaraja V, Sriram D.

Bioorg Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1016/j.bmc.2007.11.016

Bibliografisk träff 2007-10-26

Antimycobacterial activities of novel 1-(cyclopropyl/tert-butyl/4-fluorophenyl)-1,4-dihydro- 6-nitro-4-oxo-7-(substituted secondary amino)-1,8-naphthyridine-3-carboxylic acid.

Sriram D, Senthilkumar P, Dinakaran M, Yogeeswari P, China A, Nagaraja V.

J Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1021/jm700999n

Bibliografisk träff 2007-10-01

An atom efficient, solvent-free, green synthesis and antimycobacterial evaluation of 2-amino-6-methyl-4-aryl-8-[(E)-arylmethylidene]-5,6,7,8-tetrahydro-4H-pyrano[3,2-c]pyridine-3-carbonitriles.

Kumar RR, Perumal S, Senthilkumar P, Yogeeswari P, Sriram D.

Bioorg Med Chem Lett · comparative study; research support, non-u.s. gov't; journal article · DOI 10.1016/j.bmcl.2007.09.095

Bibliografisk träff 2007-08-21

Synthesis and antitubercular activity of lipophilic moxifloxacin and gatifloxacin derivatives.

de Almeida MV, Saraiva MF, de Souza MV, da Costa CF, Vicente FR, Lourenço MC.

Bioorg Med Chem Lett · research support, non-u.s. gov't; journal article · DOI 10.1016/j.bmcl.2007.07.073

Bibliografisk träff 2007-03-26

Activity of Garenoxacin against Macrolide-Susceptible and -Resistant Mycoplasma pneumoniae.

Yamazaki T, Sasaki T, Takahata M.

Antimicrob Agents Chemother · letter · DOI 10.1128/aac.01561-06

Bibliografisk träff 2007-02-26

Expression and purification of an active form of the Mycobacterium leprae DNA gyrase and its inhibition by quinolones.

Matrat S, Petrella S, Cambau E, Sougakoff W, Jarlier V, Aubry A.

Antimicrob Agents Chemother · research support, non-u.s. gov't; research-article; journal article · DOI 10.1128/aac.01282-06

Bibliografisk träff 2007-02-12

Fluoroquinolone resistance in Streptococcus pneumoniae: area under the concentration-time curve/MIC ratio and resistance development with gatifloxacin, gemifloxacin, levofloxacin, and moxifloxacin.

LaPlante KL, Rybak MJ, Tsuji B, Lodise TP, Kaatz GW.

Antimicrob Agents Chemother · research support, non-u.s. gov't; research-article; journal article · DOI 10.1128/aac.00646-06

Bibliografisk träff 2007-01-29

In vitro and in vivo activities of PD 0305970 and PD 0326448, new bacterial gyrase/topoisomerase inhibitors with potent antibacterial activities versus multidrug-resistant gram-positive and fastidious organism groups.

Huband MD, Cohen MA, Zurack M, Hanna DL, Skerlos LA, Sulavik MC, Gibson GW, Gage JW, Ellsworth E, Stier MA, Gracheck SJ.

Antimicrob Agents Chemother · research-article; journal article · DOI 10.1128/aac.01321-06

Bibliografisk träff 2007-01-24

Synthesis and antibacterial activity of 4,5,6,7-tetrahydro-thieno[3,2-c]pyridine quinolones.

Srivastava BK, Solanki M, Mishra B, Soni R, Jayadev S, Valani D, Jain M, Patel PR.

Bioorg Med Chem Lett · journal article · DOI 10.1016/j.bmcl.2007.01.038

Bibliografisk träff 2007-01-12

First report of plasmid-mediated qnrA1 in a ciprofloxacin-resistant Escherichia coli strain in Latin America.

Castanheira M, Pereira AS, Nicoletti AG, Pignatari AC, Barth AL, Gales AC.

Antimicrob Agents Chemother · research support, non-u.s. gov't; research-article; journal article · DOI 10.1128/aac.00780-06

Bibliografisk träff 2006-11-20

Multistep resistance selection and postantibiotic-effect studies of the antipneumococcal activity of LBM415 compared to other agents.

Kosowska-Shick K, Credito KL, Pankuch GA, DeWasse B, McGhee P, Appelbaum PC.

Antimicrob Agents Chemother · comparative study; research support, non-u.s. gov't; research-article; journal article · DOI 10.1128/aac.01150-06

Bibliografisk träff 2006-11-20

Fitness costs of fluoroquinolone resistance in Streptococcus pneumoniae.

Rozen DE, McGee L, Levin BR, Klugman KP.

Antimicrob Agents Chemother · research support, non-u.s. gov't; research-article; journal article · DOI 10.1128/aac.01161-06

Bibliografisk träff 2006-11-18

Synthesis and antibacterial activities of new quinolone derivatives utilizing 1-azabicyclo[1.1.0]butane.

Ikee Y, Hashimoto K, Nakashima M, Hayashi K, Sano S, Shiro M, Nagao Y.

Bioorg Med Chem Lett · research support, non-u.s. gov't; journal article · DOI 10.1016/j.bmcl.2006.11.048

Bibliografisk träff 2006-11-01

3-aminoquinazolinediones as a new class of antibacterial agents demonstrating excellent antibacterial activity against wild-type and multidrug resistant organisms.

Ellsworth EL, Tran TP, Showalter HD, Sanchez JP, Watson BM, Stier MA, Domagala JM, Gracheck SJ, Joannides ET, Shapiro MA, Dunham SA, Hanna DL, Huband MD, Gage JW, Bronstein JC, Liu JY, Nguyen DQ, Singh R.

J Med Chem · journal article · DOI 10.1021/jm060505l

Bibliografisk träff 2006-10-16

The 6-fluoro-8-methoxy quinolone gatifloxacin down-regulates interleukin-8 production in prostate cell line PC-3.

Takeyama K, Mitsuzawa H, Nishitani C, Shimizu T, Sano H, Kunishima Y, Takahashi S, Hotta H, Matsukawa M, Shibata K, Tsukamoto T, Kuroki Y.

Antimicrob Agents Chemother · research support, non-u.s. gov't; research-article; journal article · DOI 10.1128/aac.00395-06

Bibliografisk träff 2006-10-16

Contribution of target gene mutations and efflux to decreased susceptibility of Salmonella enterica serovar typhimurium to fluoroquinolones and other antimicrobials.

Chen S, Cui S, McDermott PF, Zhao S, White DG, Paulsen I, Meng J.

Antimicrob Agents Chemother · research support, u.s. gov't, p.h.s.; research support, non-u.s. gov't; research-article; journal article · DOI 10.1128/aac.00600-06

Bibliografisk träff 2006-06-01

Discovery of new antitubercular oxazolyl thiosemicarbazones.

Sriram D, Yogeeswari P, Thirumurugan R, Pavana RK.

J Med Chem · journal article · DOI 10.1021/jm060339h

Bibliografisk träff 2006-03-22

Gatifloxacin derivatives: synthesis, antimycobacterial activities, and inhibition of Mycobacterium tuberculosis DNA gyrase.

Sriram D, Aubry A, Yogeeswari P, Fisher LM.

Bioorg Med Chem Lett · research support, non-u.s. gov't; journal article · DOI 10.1016/j.bmcl.2006.02.065

Bibliografisk träff 2005-12-07

Isothiazoloquinolones containing functionalized aromatic hydrocarbons at the 7-position: synthesis and in vitro activity of a series of potent antibacterial agents with diminished cytotoxicity in human cells.

Wiles JA, Wang Q, Lucien E, Hashimoto A, Song Y, Cheng J, Marlor CW, Ou Y, Podos SD, Thanassi JA, Thoma CL, Deshpande M, Pucci MJ, Bradbury BJ.

Bioorg Med Chem Lett · journal article · DOI 10.1016/j.bmcl.2005.11.065

Bibliografisk träff 2005-08-01

A chiral benzoquinolizine-2-carboxylic acid arginine salt active against vancomycin-resistant Staphylococcus aureus.

de Souza NJ, Gupte SV, Deshpande PK, Desai VN, Bhawsar SB, Yeole RD, Shukla MC, Strahilevitz J, Hooper DC, Bozdogan B, Appelbaum PC, Jacobs MR, Shetty N, Patel MV, Jha R, Khorakiwala HF.

J Med Chem · journal article · DOI 10.1021/jm050035f

Bibliografisk träff 2005-06-01

A discriminant model constructed by the support vector machine method for HERG potassium channel inhibitors.

Tobita M, Nishikawa T, Nagashima R.

Bioorg Med Chem Lett · research support, non-u.s. gov't; journal article · DOI 10.1016/j.bmcl.2005.03.080

Bibliografisk träff 2005-03-01

A two-state homology model of the hERG K+ channel: application to ligand binding.

Rajamani R, Tounge BA, Li J, Reynolds CH.

Bioorg Med Chem Lett · research support, non-u.s. gov't; journal article · DOI 10.1016/j.bmcl.2005.01.008

Bibliografisk träff 2004-06-01

Synthesis of new fluoroquinolones and evaluation of their in vitro activity on Toxoplasma gondii and Plasmodium spp.

Anquetin G, Rouquayrol M, Mahmoudi N, Santillana-Hayat M, Gozalbes R, Greiner J, Farhati K, Derouin F, Guedj R, Vierling P.

Bioorg Med Chem Lett · journal article · DOI 10.1016/j.bmcl.2004.03.070

Bibliografisk träff 2003-08-01

Prediction of hERG potassium channel affinity by traditional and hologram qSAR methods.

Keserü GM.

Bioorg Med Chem Lett · comparative study; journal article · DOI 10.1016/s0960-894x(03)00492-x

Bibliografisk träff 2003-08-01

Discovery of (3S)-amino-(4R)-ethylpiperidinyl quinolones as potent antibacterial agents with a broad spectrum of activity and activity against resistant pathogens.

Hu XE, Kim NK, Gray JL, Almstead JI, Seibel WL, Ledoussal B.

J Med Chem · journal article · DOI 10.1021/jm030272n

Bibliografisk träff 2003-03-01

Synthesis and structure-activity relationships of 5-amino-6-fluoro-1-[(1R,2S)-2-fluorocyclopropan-1-yl]-8-methylquinolonecarboxylic acid antibacterials having fluorinated 7-[(3R)-3-(1-aminocyclopropan-1-yl)pyrrolidin-1-yl] substituents.

Inagaki H, Miyauchi S, Miyauchi RN, Kawato HC, Ohki H, Matsuhashi N, Kawakami K, Takahashi H, Takemura M.

J Med Chem · journal article · DOI 10.1021/jm020328y

Bibliografisk träff 2002-08-01

Toward a pharmacophore for drugs inducing the long QT syndrome: insights from a CoMFA study of HERG K(+) channel blockers.

Cavalli A, Poluzzi E, De Ponti F, Recanatini M.

J Med Chem · journal article · DOI 10.1021/jm0208875

Bibliografisk träff 2000-03-01

Artificial neural network applied to prediction of fluorquinolone antibacterial activity by topological methods.

Jaén-Oltra J, Salabert-Salvador MT, García-March FJ, Pérez-Giménez F, Tomás-Vert F.

J Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1021/jm980448z