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Publikationer som ChEBI hänvisar till för dp001. Visa hela publikationsregistret

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Publications in the selection

8 hits

Bibliografisk träff 2020-06-24

Synthesis and Biological Activity of 2,22-Dimethylene Analogues of 19-Norcalcitriol and Related Compounds.

Sibilska-Kaminski IK, Sicinski RR, Plum LA, DeLuca HF.

J Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1021/acs.jmedchem.0c00580

Bibliografisk träff 2015-12-02

Synthesis and Biological Activity of 2-Methylene Analogues of Calcitriol and Related Compounds.

Sibilska IK, Szybinski M, Sicinski RR, Plum LA, DeLuca HF.

J Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1021/acs.jmedchem.5b01295

Bibliografisk träff 2014-10-02

Synthesis and Biological Activity of 25-Hydroxy-2-methylene-vitamin D3 analogues monohydroxylated in the A-ring.

Sibilska IK, Sicinski RR, Ochalek JT, Plum LA, DeLuca HF.

J Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1021/jm500750b

Bibliografisk träff 2012-04-22

A 20S combined with a 22R configuration markedly increases both in vivo and in vitro biological activity of 1α,25-dihydroxy-22-methyl-2-methylene-19-norvitamin D3.

Flores A, Sicinski RR, Grzywacz P, Thoden JB, Plum LA, Clagett-Dame M, DeLuca HF.

J Med Chem · research support, non-u.s. gov't; research-article; research support, u.s. gov't, non-p.h.s.; journal article; research support, n.i.h., extramural · DOI 10.1021/jm300187x

Bibliografisk träff 2010-11-24

Removal of the 26-methyl group from 19-nor-1α,25-dihydroxyvitamin D₃ markedly reduces in vivo calcemic activity without altering in vitro VDR binding, HL-60 cell differentiation, and transcription.

Grzywacz P, Chiellini G, Plum LA, Clagett-Dame M, DeLuca HF.

J Med Chem · research support, non-u.s. gov't; research-article; research support, u.s. gov't, non-p.h.s.; journal article; research support, n.i.h., extramural · DOI 10.1021/jm1010447

Bibliografisk träff 2009-09-29

Removal of the 20-methyl group from 2-methylene-19-nor-(20S)-1alpha,25-dihydroxyvitamin D(3) (2MD) selectively eliminates bone calcium mobilization activity.

Barycki R, Sicinski RR, Plum LA, Grzywacz P, Clagett-Dame M, Deluca HF.

Bioorg Med Chem · research support, non-u.s. gov't; research-article; research support, u.s. gov't, non-p.h.s.; journal article; research support, n.i.h., extramural · DOI 10.1016/j.bmc.2009.09.047

Bibliografisk träff 2006-02-01

Vitamin D receptor: ligand recognition and allosteric network.

Yamamoto K, Abe D, Yoshimoto N, Choi M, Yamagishi K, Tokiwa H, Shimizu M, Makishima M, Yamada S.

J Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1021/jm050795q

Bibliografisk träff 1998-11-01

New 1alpha,25-dihydroxy-19-norvitamin D3 compounds of high biological activity: synthesis and biological evaluation of 2-hydroxymethyl, 2-methyl, and 2-methylene analogues.

Sicinski RR, Prahl JM, Smith CM, DeLuca HF.

J Med Chem · research support, u.s. gov't, p.h.s.; research support, non-u.s. gov't; journal article · DOI 10.1021/jm9802618