The binding mode of picrotoxinin in GABA<sub>A-ρ</sub> receptors: Insight into the subunit's selectivity in the transmembrane domain.
Naffaa MM, Samad A.
Comput Biol Chem · journal article · DOI 10.1016/j.compbiolchem.2016.07.003 PUBLICATION REGISTRY
Go to research.
Publikationsdata från Europe PMC och PubMed. Följ källhänvisningar från ämnesregistret till originalpublikationerna.
Publikationer som ChEBI hänvisar till för picrotoxinin. Visa hela publikationsregistret
A publication hit is not a conclusion. Publikationslistan visar bibliografiska uppgifter. Eventuella forskningsutdrag visas separat med originalunderlag. En källhänvisning visar inte i sig effekt, dosering eller säkerhet.
Publications in the selection
9 hitsPhenylalanine in the pore of the Erwinia ligand-gated ion channel modulates picrotoxinin potency but not receptor function.
Thompson AJ, Alqazzaz M, Price KL, Weston DA, Lummis SC.
Biochemistry · research support, non-u.s. gov't; research-article; journal article · DOI 10.1021/bi5008035Binding sites for bilobalide, diltiazem, ginkgolide, and picrotoxinin at the 5-HT3 receptor.
Thompson AJ, Duke RK, Lummis SC.
Mol Pharmacol · research support, non-u.s. gov't; research-article; journal article · DOI 10.1124/mol.111.071415Relative impact of residues at the intracellular and extracellular ends of the human GABAC rho1 receptor M2 domain on picrotoxinin activity.
Carland JE, Johnston GA, Chebib M.
Eur J Pharmacol · research support, non-u.s. gov't; journal article · DOI 10.1016/j.ejphar.2007.10.036A proposed structural basis for picrotoxinin and picrotin binding in the glycine receptor pore.
Yang Z, Cromer BA, Harvey RJ, Parker MW, Lynch JW.
J Neurochem · research support, non-u.s. gov't; journal article · DOI 10.1111/j.1471-4159.2007.04850.xInvestigation of structural requirements for inhibitory activity at the rat and housefly picrotoxinin binding sites in ionotropic GABA receptors using DISCOtech and CoMFA.
Ju XL, Hao YL, Pei JF, Ozoe Y.
Chemosphere · research support, non-u.s. gov't; journal article · DOI 10.1016/j.chemosphere.2007.06.040Mechanisms for picrotoxinin and picrotin blocks of alpha2 homomeric glycine receptors.
Wang DS, Buckinx R, Lecorronc H, Mangin JM, Rigo JM, Legendre P.
J Biol Chem · comparative study; research support, non-u.s. gov't; journal article · DOI 10.1074/jbc.m701502200Differential sensitivity of two insect GABA-gated chloride channels to dieldrin, fipronil and picrotoxinin.
Le Corronc H, Alix P, Hue B.
J Insect Physiol · journal article · DOI 10.1016/s0022-1910(02)00061-6Blocking actions of picrotoxinin analogues on insect (Periplaneta americana) GABA receptors.
Anthony NM, Holyoke CW, Sattelle DB.
Neurosci Lett · journal article · DOI 10.1016/0304-3940(94)90606-8