Palladium-Catalyzed Oxidative Direct C3- and C7-Alkenylations of Indazoles: Application to the Synthesis of Gamendazole.
Naas M, El Kazzouli S, Essassi el M, Bousmina M, Guillaumet G.
Org Lett · journal article · DOI 10.1021/acs.orglett.5b02136 PUBLICATION REGISTRY
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6 hitsToxicants target cell junctions in the testis: Insights from the indazole-carboxylic acid model.
Cheng CY.
Spermatogenesis · review-article; review; journal article · DOI 10.4161/21565562.2014.981485New approaches to male non-hormonal contraception.
Nya-Ngatchou JJ, Amory JK.
Contraception · research-article; review; journal article; research support, n.i.h., extramural · DOI 10.1016/j.contraception.2012.08.016A systematic protocol for the characterization of Hsp90 modulators.
Matts RL, Brandt GE, Lu Y, Dixit A, Mollapour M, Wang S, Donnelly AC, Neckers L, Verkhivker G, Blagg BS.
Bioorg Med Chem · research support, non-u.s. gov't; research-article; journal article; research support, n.i.h., extramural · DOI 10.1016/j.bmc.2010.10.029Gamendazole, an orally active indazole carboxylic acid male contraceptive agent, targets HSP90AB1 (HSP90BETA) and EEF1A1 (eEF1A), and stimulates Il1a transcription in rat Sertoli cells.
Tash JS, Chakrasali R, Jakkaraj SR, Hughes J, Smith SK, Hornbaker K, Heckert LL, Ozturk SB, Hadden MK, Kinzy TG, Blagg BS, Georg GI.
Biol Reprod · journal article; research support, n.i.h., extramural · DOI 10.1095/biolreprod.107.062679A novel potent indazole carboxylic acid derivative blocks spermatogenesis and is contraceptive in rats after a single oral dose.
Tash JS, Attardi B, Hild SA, Chakrasali R, Jakkaraj SR, Georg GI.
Biol Reprod · journal article; research support, n.i.h., extramural · DOI 10.1095/biolreprod.106.057810