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Publikationer i urvalet

32 träffar

Bibliografisk träff 2008-09-13

Structural requirements for drug inhibition of the liver specific human organic cation transport protein 1.

Ahlin G, Karlsson J, Pedersen JM, Gustavsson L, Larsson R, Matsson P, Norinder U, Bergström CA, Artursson P.

J Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1021/jm8003152

Bibliografisk träff 2008-03-19

New approach to measure protein binding based on a parallel artificial membrane assay and human serum albumin.

Lázaro E, Lowe PJ, Briand X, Faller B.

J Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1021/jm7012826

Bibliografisk träff 2007-09-13

New series of antiprion compounds: pyrazolone derivatives have the potent activity of inhibiting protease-resistant prion protein accumulation.

Kimata A, Nakagawa H, Ohyama R, Fukuuchi T, Ohta S, Doh-ura K, Suzuki T, Miyata N.

J Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1021/jm070688r

Bibliografisk träff 2007-05-24

Synthesis and evaluation of amphiphilic cationic quinine-derived for antibacterial activity against methicillin-resistant Staphylococcus aureus.

Lv J, Qian Y, Liu T, Wang Y.

Bioorg Med Chem Lett · research support, non-u.s. gov't; journal article · DOI 10.1016/j.bmcl.2007.05.065

Bibliografisk träff 2007-05-17

Synthesis and biological studies of novel 2-aminoalkylethers as potential antiarrhythmic agents for the conversion of atrial fibrillation.

Plouvier B, Beatch GN, Jung GL, Zolotoy A, Sheng T, Clohs L, Barrett TD, Fedida D, Wang WQ, Zhu JJ, Liu Y, Abraham S, Lynn L, Dong Y, Wall RA, Walker MJ.

J Med Chem · journal article · DOI 10.1021/jm0604528

Bibliografisk träff 2007-04-25

A novel artemisinin-quinine hybrid with potent antimalarial activity.

Walsh JJ, Coughlan D, Heneghan N, Gaynor C, Bell A.

Bioorg Med Chem Lett · journal article · DOI 10.1016/j.bmcl.2007.04.054

Bibliografisk träff 2006-08-01

Biological activities and 3D QSAR studies of a series of Delisea pulchra (cf. fimbriata) derived natural products.

Wright AD, de Nys R, Angerhofer CK, Pezzuto JM, Gurrath M.

J Nat Prod · journal article; research support, n.i.h., extramural · DOI 10.1021/np050510c

Bibliografisk träff 2006-03-09

Antimalarial effect of bis-pyridinium salts, N,N'-hexamethylenebis(4-carbamoyl-1-alkylpyridinium bromide).

Fujimoto K, Morisaki D, Yoshida M, Namba T, Hye-Sook K, Wataya Y, Kourai H, Kakuta H, Sasaki K.

Bioorg Med Chem Lett · research support, non-u.s. gov't; journal article · DOI 10.1016/j.bmcl.2006.02.030

Bibliografisk träff 2005-05-01

Calculating virtual log P in the alkane/water system (log P(N)(alk)) and its derived parameters deltalog P(N)(oct-alk) and log D(pH)(alk).

Caron G, Ermondi G.

J Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1021/jm048980b

Bibliografisk träff 2004-08-01

Defining determinant molecular properties for the blockade of the apamin-sensitive SKCa channel in guinea-pig hepatocytes: the influence of polarizability and molecular geometry.

Galanakis D, Ganellin CR.

Bioorg Med Chem Lett · journal article · DOI 10.1016/j.bmcl.2004.05.031

Bibliografisk träff 2004-04-01

Pi-delocalized beta-carbolinium cations as potential antimalarials.

Takasu K, Shimogama T, Saiin C, Kim HS, Wataya Y, Ihara M.

Bioorg Med Chem Lett · research support, non-u.s. gov't; journal article · DOI 10.1016/j.bmcl.2004.01.055

Bibliografisk träff 2004-03-01

Surface activity profiling of drugs applied to the prediction of blood-brain barrier permeability.

Suomalainen P, Johans C, Söderlund T, Kinnunen PK.

J Med Chem · journal article · DOI 10.1021/jm0309001

Bibliografisk träff 2004-02-01

Conformer- and alignment-independent model for predicting structurally diverse competitive CYP2C9 inhibitors.

Afzelius L, Zamora I, Masimirembwa CM, Karlén A, Andersson TB, Mecucci S, Baroni M, Cruciani G.

J Med Chem · journal article · DOI 10.1021/jm030972s

Bibliografisk träff 2003-08-01

The imidazo[2,1-a]isoindole system. A new skeletal basis for antiplasmodial compounds.

del Olmo E, Armas MG, Ybarra M, López JL, Oporto P, Giménez A, Deharo E, San Feliciano A.

Bioorg Med Chem Lett · research support, non-u.s. gov't; journal article · DOI 10.1016/s0960-894x(03)00509-2

Bibliografisk träff 2003-07-01

Structure-activity relationships of novel anti-malarial agents. Part 7: N-(3-benzoyl-4-tolylacetylaminophenyl)-3-(5-aryl-2-furyl)acrylic acid amides with polar moieties.

Wiesner J, Mitsch A, Jomaa H, Schlitzer M.

Bioorg Med Chem Lett · research support, non-u.s. gov't; journal article · DOI 10.1016/s0960-894x(03)00353-6

Bibliografisk träff 2003-01-01

Homology modeling of rat and human cytochrome P450 2D (CYP2D) isoforms and computational rationalization of experimental ligand-binding specificities.

Venhorst J, ter Laak AM, Commandeur JN, Funae Y, Hiroi T, Vermeulen NP.

J Med Chem · journal article · DOI 10.1021/jm0209578

Bibliografisk träff 2002-12-01

Pharmacophore model of drugs involved in P-glycoprotein multidrug resistance: explanation of structural variety (hypothesis).

Pajeva IK, Wiese M.

J Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1021/jm020941h

Bibliografisk träff 2002-10-01

Structure-activity relationships of novel anti-malarial agents. Part 4: N-(3-benzoyl-4-tolylacetylaminophenyl)-3-(5-aryl-2-furyl)acrylic acid amides.

Wiesner J, Mitsch A, Wissner P, Krämer O, Jomaa H, Schlitzer M.

Bioorg Med Chem Lett · journal article · DOI 10.1016/s0960-894x(02)00555-3

Bibliografisk träff 2002-09-01

Structure-activity relationships of the antimalarial agent artemisinin. 7. Direct modification of (+)-artemisinin and in vivo antimalarial screening of new, potential preclinical antimalarial candidates.

Avery MA, Alvim-Gaston M, Vroman JA, Wu B, Ager A, Peters W, Robinson BL, Charman W.

J Med Chem · research support, u.s. gov't, p.h.s.; research support, non-u.s. gov't; journal article · DOI 10.1021/jm020142z

Bibliografisk träff 2002-08-01

Antimalarial compounds from Parinari capensis.

Uys AC, Malan SF, van Dyk S, van Zyl RL.

Bioorg Med Chem Lett · journal article · DOI 10.1016/s0960-894x(02)00350-5

Bibliografisk träff 2002-02-01

Structure-activity relationships of novel anti-malarial agents. Part 3: N-(4-acylamino-3-benzoylphenyl)-4-propoxycinnamic acid amides.

Wiesner J, Kettler K, Jomaa H, Schlitzer M.

Bioorg Med Chem Lett · journal article · DOI 10.1016/s0960-894x(01)00798-3

Bibliografisk träff 2002-02-01

Rhodacyanine dyes as antimalarials. 1. Preliminary evaluation of their activity and toxicity.

Takasu K, Inoue H, Kim HS, Suzuki M, Shishido T, Wataya Y, Ihara M.

J Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1021/jm0155704

Bibliografisk träff 2001-12-01

Cheminformatic models to predict binding affinities to human serum albumin.

Colmenarejo G, Alvarez-Pedraglio A, Lavandera JL.

J Med Chem · journal article · DOI 10.1021/jm010960b

Bibliografisk träff 2001-09-01

New anti-malarial flavonol glycoside from Hydrangeae Dulcis Folium.

Murakami N, Mostaqul HM, Tamura S, Itagaki S, Horii T, Kobayashi M.

Bioorg Med Chem Lett · research support, non-u.s. gov't; journal article · DOI 10.1016/s0960-894x(01)00467-x

Bibliografisk träff 2001-02-01

Structure-activity relationships of novel anti-malarial agents. Part 2: cinnamic acid derivatives.

Wiesner J, Mitsch A, Wissner P, Jomaa H, Schlitzer M.

Bioorg Med Chem Lett · journal article · DOI 10.1016/s0960-894x(00)00684-3

Bibliografisk träff 2000-08-01

Synthesis of novel ferrocenyl sugars and their antimalarial activities.

Itoh T, Shirakami S, Ishida N, Yamashita Y, Yoshida T, Kim HS, Wataya Y.

Bioorg Med Chem Lett · research support, non-u.s. gov't; journal article · DOI 10.1016/s0960-894x(00)00313-9

Bibliografisk träff 2000-06-01

QSAR model for drug human oral bioavailability.

Yoshida F, Topliss JG.

J Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1021/jm0000564

Bibliografisk träff 2000-05-01

Biosensor analysis of the interaction between immobilized human serum albumin and drug compounds for prediction of human serum albumin binding levels.

Frostell-Karlsson A, Remaeus A, Roos H, Andersson K, Borg P, Hämäläinen M, Karlsson R.

J Med Chem · journal article · DOI 10.1021/jm991174y

Bibliografisk träff 1994-05-01

Synthesis and in vitro evaluation of 9-anilino-3,6-diaminoacridines active against a multidrug-resistant strain of the malaria parasite Plasmodium falciparum.

Gamage SA, Tepsiri N, Wilairat P, Wojcik SJ, Figgitt DP, Ralph RK, Denny WA.

J Med Chem · research support, non-u.s. gov't; journal article · DOI 10.1021/jm00036a014

Bibliografisk träff 1989-06-01

Antimalarial activity of new water-soluble dihydroartemisinin derivatives. 2. Stereospecificity of the ether side chain.

Lin AJ, Lee M, Klayman DL.

J Med Chem · comparative study; journal article · DOI 10.1021/jm00126a017